Carbamates and crop protection agents containing them

ABSTRACT

Carbamates of the formula I                    
     where the substituents have the following meanings: 
     Z is methoxy, NH 2 , NHCH 3 , N(CH 3 ) 2 , CH 3 , C 2 H 5 , CF 3  or CCl 3 , 
     X and Y are identical or different and each is hydrogen, F, Cl, Br, CF 3 , CN, NO 2 , alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may be condensed together to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, 
     R 1  may also be substituted or unsubstituted and is O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O—CO 2 -alkyl, 
     A is —O—, —S—, —CR 2 ═CR 3 —, CHR 2 —O—, —CHR 2 —S—, —CHR 2 —O—N═C(R 4 )—, —CR 2 ═N—O—, —O—N═C(R 4 )—, —C≡C—, —CHR 2 —CHR 3 —, —CHR 2 —O—CO—, —O—CHR 2 — or a single bond, 
     B is substituted or unsubstituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, substituted or unsubstituted alkylaryl, substituted or unsubstituted alkylhetaryl, substituted or unsubstituted alkylcycloalkyl, substituted or unsubstituted alkylcycloalkenyl, 
     R 2  and R 3  are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, 
     R 4  is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl, 
     R 5  is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl and plant-tolerated acid and base adducts thereof, and fungicides containing them.

This application is a Division of application Ser. No. 09/275,767 filed on Mar. 25, 1999 now U.S. Pat. No. 6,075,148, which is a divisional of Ser. No. 09/110,884, filed Jul. 7, 1998 now U.S. Pat. No. 5,981,532, which is a continuation of Ser. No. 08/256,628, filed Jul. 29, 1994 now U.S. Pat. No. 5,824,705, which is a continuation of PCT/EP93/00104, filed on Jan. 18, 1993.

DESCRIPTION

The present invention relates to carbamates and crop protection agents, in particular for controlling fungi, insects, nematodes and spider mites.

It is known that aniline derivatives, for example isopropyl N-phenylcarbamate or the corresponding 3-chlorophenyl ester (GB 574 995) or methyl N-3,4-dichlorophenylcarbamate (BE 612 550) can be used as crop protection agents. However, their fungicidal action is unsatisfactory.

It has now been found, surprisingly, that carbamates of the formula I

where the substituents have the following meanings:

Z is methoxy, NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂H₅, CF₃ or CCl₃,

X and Y independently of one another are each hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ is unsubstituted or substituted alkyl, alkenyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, —CN₃—CN, —CH₂OCH₃, —CO₂CH₃ or —S—R⁵, O-alkyl, O-alkenyl, O-alkynyl, O-cycloalkyl, O-cycloalkenyl or O—CO₂-alkyl,

A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl, hydrogen, unsubstituted or substituted alkylaryl, unsubstituted or substituted alkylhetaryl, unsubstituted or substituted alkylcycloalkyl or unsubstituted or substituted alkylcycloalkenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is hydrogen, CN, alkyl, alkenyl, alkynyl, alkoxy or cycloalkyl,

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products have a good fungicidal, acaricidal, insecticidal and nematocidal action.

Acids for addition products are, for example, mineral acids, such as hydrochloric acid, hydrobromic acid, phosphoric acid, sulfuric acid or nitric acid, or carboxylic acids, such as formic acid, acetic acid, oxalic acid, malonic acid, lactic acid, malic acid, succinic acid, tartaric acid, citric acid, salicylic acid, p-toluenesulfonic acid or dodecylbenzenesulfonic acid, as well as proton-acidic compounds generally, for example saccharin.

Bases for base addition products are, for example, potassium hydroxide, sodium hydroxide, potassium carbonate, sodium carbonate and ammonium hydroxide.

The novel compounds of the formula I may be obtained in the preparation as mixtures of stereoisomers (E/Z isomers, diastereomers, enantiomers), which can be separated into the individual components in a conventional manner, for example by crystallization or chromatography. Both the individual isomers and mixtures thereof may be used as fungicides, acaricides, nematocides or insecticides, and form the subject of the present invention.

The abovementioned alkyl radicals may be substituted and are of 1 to 6 carbon atoms.

The abovementioned alkenyl and alkynyl radicals may be substituted and are of 2 to 6 carbon atoms.

The abovementioned cycloalkyl radicals are of 3 to 10 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned aryl radicals are of 6, 10 or 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different subutituents R⁶.

The abovementioned hetaryl radicals have 5 to 14 ring atoms, including from 1 to 4 hetero atoms selected from the group consisting of N, O and S, are unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned heterocyclyl radicals have 5 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S, are saturated or partially unsaturated and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

The abovementioned cycloalkenyl radicals are of 5 to 14 carbon atoms and are unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁶.

Two adjacent substituents R⁶, together with the carbon atoms of which they are substituents, may form a carbocyclic hydrogenated, partially unsaturated or aromatic ring having 3 to 14 carbon atoms or a heterocyclic hydrogenated, partially unsaturated or heteroaromatic ring having 3 to 14 carbon atoms, including 1 to 4 hetero atoms selected from the group consisting of N, O and S.

R⁶ may be unsubstituted or substituted, for example by 1 to 4 identical or different substituents R⁷, and R⁶ is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoxyimino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl, alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

R⁷ is is any substituent and is, for example, hydrogen, halogen, cyano, nitro, haloalkyl, alkyl, haloalkoxy, alkenyl, alkynyl, cycloalkyl, aryl, hetaryl, heterocyclyl, cycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, aryloxy, hetaryloxy, heterocyclyloxy, cycloalkenyloxy, alkoximino, alkenyloximino, alkynyloximino, cycloalkoximino, cycloalkenyloximino, aryloximino, hetaryloximino, heterocyclyloximino, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, cycloalkyloxycarbonyl, aryloxycarbonyl, hetaryloxycarbonyl, heterocyclyloxycarbonyl, cycloalkenyloxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkenylaminocarbonyl, dialkenylaiminocarbonyl, alkylthio, alkenylthio, alkynylthio, cycloalkylthio, arylthio, hetarylthio, heterocyclylthio, cycloalkenylthio, alkylamino, alkenylamino, alkynylamino, cycloalkylamino, arylamino, hetarylamino, heterocyclylamino, cycloalkenylamino, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, arylcarbonyl, hetarylcarbonyl, heterocyclylcarbonyl, cycloalkenylcarbonyl, alkylsulfoxyl; alkenylsulfoxyl, alkynylsulfoxyl, cycloalkylsulfoxyl, arylsulfoxyl, hetarylsulfoxyl, heterocyclylsulfoxyl, cycloalkenylsulfoxyl, alkylsulfonyl, alkenylsulfonyl, alkynylsulfonyl, cycloalkylsulfonyl, arylsulfonyl, hetarylsulfonyl, heterocyclylsulfonyl, cycloalkenylsulfonyl, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, cycloalkylsulfinyl, arylsulfinyl, hetarylsulfinyl, heterocyclylsulfinyl or cycloalkenylsulfinyl.

The abovementioned alkyl radicals may be substituted, are preferably of 1 to 6 carbon atoms and are, in particular, methyl, ethyl, propyl, such as n-propyl or isopropyl, butyl, such as n-butyl, isobutyl, tert-butyl or sec-butyl, pentyl or hexyl.

The abovementioned alkenyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethenyl, propenyl, such as prop-1-enyl, prop-2-enyl or prop-1-en-2-yl, butenyl, such as but-1-enyl, but-2-enyl, but-3-enyl, but-1-en-3-yl, but-2-en-2-yl, but-1-en-2-yl, 2-methyl-1-propenyl or 2-methyl-2-propenyl, pentenyl or hexenyl.

The abovementioned alkynyl radicals may be substituted, are preferably of 2 to 6 carbon atoms and are, in particular, ethynyl, propynyl, such as prop-1-ynyl or prop-3-ynyl, butynyl, such as but-1-ynyl, but-2-ynyl, but-3-ynyl or 1-methylprop-2-ynyl, pentynyl or hexynyl.

The abovementioned halogens are fluorine, chlorine, bromine or iodine.

The abovementioned cycloalkyl radicals are preferably cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl, cyclononyl, cyclodecyl, bornanyl, norbornanyl, dicyclohexyl, bicyclo[3.3.0]octyl, bicyclo[3.2.1]octyl, bicyclo[2.2.2]octyl or bicyclo[3.3.1]nonyl.

The abovementioned cycloalkenyl radicals are preferably cyclopropenyl, cyclobutenyl, cyclopentenyl, cyclohexenyl, cycloheptenyl, cyclooctenyl, cyclononenyl, cyclodecenyl, bornenyl, norbornenyl, bicyclo[3.3.0]octenyl, bicyclo[3.2.1]octenyl, bicyclo[2.2.2]octenyl or bicyclo[3.3.1]nonenyl.

The abovementioned haloalkyl radicals are preferably C₁-C₄-haloalkyl, in particular C₁- or C₂-haloalkyl, such as chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The abovementioned haloalkoxy radicals are preferably C₁-C₄-haloalkoxy, in particular C₁- or C₂-haloalkoxy, such as chloromethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or pentafluoroethoxy.

The abovementioned aryl radicals are preferably phenyl, 1-naphthyl, 2-naphtyl, 1-anthracenyl, 2-anthracenyl or 9-anthracenyl.

The abovementioned hetaryl radicals are preferably furyl, such as 2-furyl or 3-furyl, thienyl, such as 2-thienyl or 3-thienyl, pyrrolyl, such as 1-pyrrolyl, 2-pyrrolyl or 3-pyrrolyl, isoxazolyl, such as 3-isoxazolyl, 4-isoxazolyl or 5-isoxazolyl, isothiazolyl, such as 3-isothiazolyl, 4-isothiazolyl or 5-isothiazolyl, pyrazolyl, such as 1-pyrazolyl, 3-pyrazolyl, 4-pyrazolyl or 5-pyrazolyl, oxazolyl, such as 2-oxazolyl, 4-oxazolyl or 5-oxazolyl, thiazolyl, such as 2-thiazolyl, 4-thiazolyl or 5-thiazolyl, imidazolyl, such as 1-imidazolyl, 2-imidazolyl, 4-imidazolyl or 5-imidazolyl, 1,2,3-thiadiazolyl, 1,2,4-thiadiazolyl, 1,2,5-thiadiazolyl, 1,3,4-thiadiazolyl, tetrazolyl, 1,2,3,4-thiatriazolyl, 1,2,3,4-oxatriazolyl, pyridyl, such as 2-pyridyl or 4-pyridyl, pyridazinyl, such as 3-pyridazinyl or 4-pyridazinyl, pyrimidinyl, such as 2-pyrimidinyl, 4-pyrimidinyl or 5-pyrimidinyl, pyrazinyl, such as 2-pyrazinyl or 3-pyrazinyl, 1,2,4-triazinyl, 1,3,5-triazinyl or 1,2,4,5-tetrazinyl.

Adjacent substituents of the hetero atoms may be condensed to form an aromatic or heteroaromatic ring, so that hetaryl also comprises fused ring systems, eg. benzofuranyl, isobenzofuranyl, 1-benzothienyl, 2-benzothienyl, indolyl, isoindolyl, benzisoxazolyl, benzoxazolyl, benzisothiazolyl, benzothiazolyl, such as 2-benzothiazolyl, 4-benzothiazolyl, 5-benzothiazolyl, 6-benzothiazolyl or 7-benzothiazolyl, indazolyl, benzimidazolyl, benzofurazanyl, dibenzofuranyl, dibenzothienyl, acridinyl, phenanthridinyl, carbazolyl, quinolyl, isoquinolyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl, 1,5-naphthyridinyl, 1,6-naphthyridinyl, 1,7-naphthyridinyl, 1,8-naphthyridinyl, pteridinyl, pyrrolopyridinyl, pyrrolopyridazinyl, pyrrolopyrimidinyl, pyrrolopyrazinyl, pyrrolotriazinyl, furopyridyl, furopyridazinyl, furopyrimidinyl, furopyrazinyl, furotriazinyl, thienopyridyl, thienopyridazinyl, thienopyrimidinyl, thienopyrazinyl, thienotriazinyl, imidazopyridazinyl, imidazopyrimidinyl, imidazopyrazinyl, pyrazolopyridyl, pyrazolopyridazinyl, pyrazolopyrimidinyl, pyrazopyrazinyl, isoxazolopyrazinyl, oxazolopyridyl, oxazolopyridazinyl, oxazolopyrimidinyl, oxazolopyrazinyl, thiazolopyridyl, thiazolopyridazinyl, isothiazolopyrazinyl, triazolopyridyl, triazolopyridazinyl, triazolopyrimidinyl or triazolopyrazinyl.

The abovementioned heterocycyl radicals are preferably 2-tetrahydrofuranyl, oxiranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1,2,4-oxadiazolidin-3-yl, 1,2,4-oxadiazolidin-5-yl, 1,2,4-thiadiazolidin-3-yl, 1,2,4-thiadiazolidin-5-yl, 1,2,5-triazolidin-3-yl, 1,3,4-oxadiazolidin-2-yl, 1,3,4-thiadiazolidin-2-yl, 1,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,5-dihydrofur-2-yl, 2,5-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,3-dihydrothieno-2-yl, 2,3-dihydrothien-3-yl, 2,5-dihydrothien-2-yl, 2,4-pyrrolin-2-yl, 2,3-pyrrolin-3-yl, 2,5-pyrrolin-2-yl, 2,5-pyrrolin-3-yl, 2,3-isoxazolidin-3-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-2-yl, 2,3-isoxazolin-4-yl, 3,4-isoxazolin-3-yl, 4,5-isoxazolin-4-yl, 2,3-isoxazolin-5-yl, 3,4-isoxazolin-5-yl, 4,5-isoxazolin-5-yl, 2,3-isothiazolin-3-yl, 3,4-isothiazolin-3-yl, 4,5-isothiazolin-3-yl, 2,3-isothiazolin-4-yl, 3,4-isothiazolin-4-yl, 4,5-isothiazolin-4-yl, 2,3-isothiazolin-5-yl, 3,4-isothiazolin-5-yl, 4,5-isothiazolin-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3- dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1-yl, 3,4-dihydropyrazol-2-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 3,4-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4-yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 3-tetrahydropyridazinyl, 4-tetrahydropyridazinyl, 2-tetrahydropyrimidinyl, 4-tetrahydropyrimidinyl, 5-tetrahydropyrimidinyl, 2-tetrahydropyrazinyl, 1,3,5-tetrahydrotriazin-2-yl, 1,2,4-tetrahydrotriazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, oxazol-2-in-2-yl, 2-tetrahydropyranyl, 1,3-dioxolan-2-yl, thiazol-2-in-2-yl, 3,4,5,6-tetrahydropyridin-2-yl, 4H-1,3-thiazin-2-yl, 4H-3,1-benzothiazin-2-yl, 1,1-dioxo-2,3,4,5-tetrahydrothien-2-yl, 2H-1,4-benzothiazin-3-yl, 2H-1,4-benzoxazin-3-yl, 1,3-dihydrooxazin-2-yl, 1,3-dithian-2-yl, N-morpholinyl or dihydroquinazolinyl.

The invention furthermore relates to carbamates of the formula I

where the substituents have the following meanings:

Z is methoxy, NH₂, NHCH₃ or CH₃,

X and Y independently of one another are each hydrogen, F, Cl, Br, CF, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form a phenyl ring,

R¹ is hydrogen, alkyl, alkenyl alkynyl cyclopropyl, cyclopropylmethyl, cyclobutyl, —CH₂—CN, —CH₂—O—CH₃, —CO₂CH₃ or —S—R⁵,

A in —O—, —CR²═CR³, —C≡C—, —CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O— or —O—N═C(R⁴)—,

a) B is substituted phenyl when A is —CR²≡CR³—, —C═C—, —CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O— or —O—N═C(R⁴),

b) or B is unsubstituted or substituted cyclolalkyl, unsubstituted or substituted cycloalkenyl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted hetaryl, unsubstituted or substituted naphthyl, unsubstituted or substituted arylalkyl, unsubstituted or substituted hetarylalkyl, unsubstituted or substituted cycloalkylalkyl, unsubstituted or substituted cycloalkenylalkyl or unsubstituted or substituted anthracenyl,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl,

R⁴ is CN, alkyl, alkenyl, alkynyl or cycloalkyl and

R⁵ is alkyl, cyclopropyl, cyclopropylmethyl or cyclobutyl, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula II

where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula III

where X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula I as claimed in claim 2, where A is —CH═CH— and X, Y, R¹ and B have the meanings stated in claim 2.

The invention furthermore relates to carbamates of the formula VII

where the substituents have the following meanings:

X and Y independently of one another are each hydrogen, Fe Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or X and Y may be condensed together to form an unsubstituted or substituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring,

R¹ can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or —CO₂-alkyl,

A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond,

B can be unsubstituted or substituted and is alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, cycloalkynyl, aryl, hetaryl, heterocyclyl or hydrogen,

R² and R³ independently of one another are each hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R₁ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, and their plant-tolerated acid addition products and base addition products.

The invention furthermore relates to carbamates of the formula VIII

where A, B and R¹ have the meanings stated in claim 9.

The invention furthermore relates to carbamates of the formula IX

where R¹ and B have the meanings stated in claim 1.

The invention furthermore relates to carbamates of the formula X

where R¹ and B have the meanings stated in claim 1.

The novel compounds can be prepared, for example, by the following processes:

The nitrobenzenes 1 obtainable by standard processes are reduced to the anilines 2, for example with hydrogen or hydrogen transfer agents, such as ammonium formate, in the presence of suitable catalysts, such as Pd, Pt or Ni, with complex reducing agents, eg. Collman's reagent (Na₂Fe(CO)₄) or by other methods known from the literature (J. March, Advanced Organic Chemistry, 3rd Edition, 1985, page 1103 et seq.). The anilines 2 are reacted under alkaline conditions with methyl chloroformate to give the carbamates 3. The reaction of the carbamates 3 under alkaline conditions with the corresponding alkylating agents, acylating agents or R⁵—S—S(═O)₂—R⁵ gives the derivatives 4 (Scheme 1).

The nitrobenzenes 5 can be converted into the carbamates 6 similarly to Scheme 1. The halogen derivatives 7 (Z=Cl or Br) are obtainable by acidic cleavage of the methyl ether of 6 (Scheme 2).

Alternatively, the halogen derivatives 7 (Z=Cl or Br) are obtainable from the derivatives 9 by free radical halogenation. The carbamates 9 are in turn prepared from the corresponding starting materials 8, similarly to Scheme 1 (Scheme 3).

The halogen derivatives 7 (Z=Cl or Br) can be converted into the active ingredients 10 under alkaline conditions. Alternatively, the compounds 7 are converted into the phosphorus compounds 11a and 11b by reaction with P(C₆H₅)₃ or P(O-Alkyl)₃, or into the carbonyl compounds 12 by oxidation (for example with N-methylmorpholine N-oxide) (Scheme 4).

A=—CHR²—O—

—CHR²—S—

—CHR²—O—N═C (R⁴)—

The corresponding stilbenes 13 are obtainable from the phosphonium salts 11a or phosphonates 11b or carbonyl compounds 12 by a Wittig reaction (Scheme 5).

Partial reduction of the nitroaromatics 21 (for example with zinc (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278) or with hydrogen in the presence of suitable catalysts such as platinum (similarly to European Patent 85,890)) gives the hydroxylamines 22, which can be reacted under alkaline conditions with an acylating agent (eg. propionyl chloride) or a carbamoylating agent (eg. methyl isocyanate) to give the compound 23 and then with an electrophile, for example with an alkylating agent, to give the active ingredients 24 (scheme 11).

In addition, the hydroxylamine 25 can be acylated or aminoacylated (for example with methyl isocyanate) (similarly to Bamberger et al., Ann. Chem. 316 (1901), 278; European Patent 85,890) to give the compound 26, which can then be alkylated or alkoxyacylated (for example with chloroformates) to give the hydroxylamine derivative 27. The free radical halogenation of 27, for example with N-bromosuccinamide, bromine, chlorine or So₂Cl₂ in the presence of free radical initiator, eg. azobisisobutyronitrile, or with exposure to UV light, then gives the halide 28 (Hal=Cl or Br; Scheme 12).

The halides 28 can then be converted into the compounds 29 with the corresponding nucelphiles (Scheme 13).

In addition, the halides 28 can be converted b free radical reaction to the dihalide 30 and then converted by with H₂O/MeOH in the presence of AgNO₃ into the carbonyl compound 31 or reacted directly with N-methylmorpholine N-oxide to give the carbonyl compound 11. Furthermore, the phosphonates, phosphonium salts or phosphine oxides 32 (P is the particular organophosphorus radical) are obtainable from the halides 8 (Scheme 14).

The carbonyl compounds 31 can then be reacted with the corresponding hydroxylamines to give the oximes 33 or can be subjected to a Wittig reaction to give the olefins 34, The olefins 34 are also obtainable by a Wittig reaction starting from the phosphonates, phosphonium salts or phosphine oxides 32 (Scheme 15).

The saturated compounds 35 can be prepared from the olefins 34 by reduction or, where R² and R³ are each the acetylenes 3 6 can be prepared from said olefins by halogen addition-(Hal=Cl, Br or I) and subsequent twofold elimination of hydrogen halide (Scheme 16).

Alternatively, the ureas 39 can be synthesized by acylation of the hydroxylamines 22 to the compounds 37, subsequent alkylation or acylation to the compounds 38 and substitution of the nucleofugic leaving group V (V is, for example, OCH₃, OCCl₃, CCl₃, O-phenyl or O-p-nitrophenyl) by NH₃, H₂N—CH₃ or HN(CH₃)₂ (Scheme 17).

Alternatively, ureas of the formula 39 can also be obtained by alkylating ureas of the formula 41, which in turn are obtainable from 17 by reacting 17 with the corresponding amines, or directly from 22 by aminocarbonylation (for example with dimethylcarbamoyl chloride or methyl isocyanate) (cf. for example Houben-Weyl, volume E16a, page 208).

Furthermore, ureas of the formula 39 can also be obtained from the N-aryl-O-alkylhydroxylamines of the formula 42 in a similar manner by aminocarbonylation.

The compounds of the formula 42 arc in turn obtainable by methods known from the literature, from hydroxylamines of the formula 2 (cf. for example Houben-Weyl, volume E16a, pages 271 and 282-289).

In addition, the hydroxylamines 22 are obtainable from the anilines 43 by formation of the imines 44, oxidation of the compounds 44 with the m-chloroperbenzoic acid and reaction of the oxaziridines 45 with hydroxylamine (Scheme 18; similarly to G. Grundke et al., Synthesis 1987, 1115).

The Examples which follow illustrate the preparation of the novel compounds.

EXAMPLES Example 1 Methyl N-ethyl-N-(2-(2′-methylphenoxymethyl)-phenyl)carbamate (Table 7, No. 2)

a) Methyl N-(o-methylphenyl)-carbamate

50 g (0.53 mol) of methyl chloroformate are added dropwise to 53 g (0.5 mol) of o-toluidene in 500 ml of methylene chloride. During this procedure, the reaction solution heats up to the boiling point and a colorless solid is precipitated.

Stirring is carried out for one hour, after which 200 ml of 10% strength sodium hydroxide solution are added dropwise, the colorless solid going into solution. The organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The remaining solid is stirred with n-hexane and filtered off under suction. 84 g (0.5 mol, quantitative yield) of the title compound are obtained as a colorless solid.

mp.=61-62° C.

¹H-NMR (DMSO-d₆; δ (ppm)): 8.85 (s, 1H, NH); 7.35 (d, broad, 1H, aromatic); 7.1 (m, 3H, aromatic); 3.6 (s, 3H, OCH₃); 2.2 (s, 3H, CH₃)

b) Methyl N-ethyl-N-(o-methylphenyl)-carbamate

5.1 g (0.2 mol) of sodium hydride are added a little at a time to 30 g (0.18 mol) of methyl N-(o-methylphenyl)-carbamate (Example 1a) in 200 ml of dimethylformamide. After the evolution of gas has ceased, 30 g (0.2 mol) of ethyl iodide are added dropwise, the reaction mixture being lightly cooled in a water bath. A white solid is precipitated. After about 4 hours, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is dried over MgSO₄ and evaporated down. The residue is distilled. 32.5 g (0.17 mol=93%) of the title compound are obtained as a colorless oil.

bp.^(0.5)=74° C.

¹H-NMR (CDCl₃; δ (ppm): 7.2 (m, 3H, aromatic); 7.1 (m, 1H, aromatic); 3.8 (m, 1H, N—CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N—CH_(B)); 2.2 (s, 3H, CH₃); 1.1 (t, 3H, CH₃)

c) Methyl N-ethyl-N-(o-bromomethylphenyl)-carbamate

A mixture of 30 g (0.155 mol) of methyl N-ethyl-N-(o-methylphenyl)-carbamate (Example 1b), 33 g (0.185 mol) of N-bromosuccinimide and 0.1 g of azoisobutyronitrile in 300 ml of carbon tetrachloride is exposed to a 300 W UV lamp for 6 hours. During this procedure, the contents of the flask heat up to about 70° C. Thereafter, the reaction mixture is washed four times with water, dried and evaporated down. The residue obtained comprises 41 g of a brown oil which contains the title compound in about 50% purity and is used without further purification in the next reaction.

¹H-NMR (CDCl₃; δ (ppm)): 7.2 (m, 4H, aromatic); 4.45 (s, 2H, CH₂—Br); 3.8 (m, 1H, N—CH_(A)); 3.6 (s, 3H, OCH₃); 3.5 (m, 1H, N—CH_(B)); 1.15 (t, 3H, J=8 Hz, CH₃)

d) Methyl N-ethyl-N-(2-(2′-methylphenoxymethyl)phenyl)-carbamate (Table 7, No. 2)

2.4 g (17 mmol) of sodium hydride are added a little at a time to 8.6 g (80 mmol) of o-cresol in 100 ml of dimethylformamide. Stirring is carried out for 30 minutes at room temperature (20° C.), after which 20.5 g of methylN-ethyl-N-(o-bromomethylphenyl)-carbamate (Example 1c, about 50% purity, about 37 mmol) are added. Stirring is carried out overnight at room temperature, after which the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The combined ether phases are dried over MgSO₄ and evaporated down. The residue is distilled in a kugelrohr (bulb tube) apparatus. 10 g of a yellow oil are obtained at 220° C. and 0.2 mbar, and the oil is then purified by chromatography with cyclohexane/ethyl acetate mixtures over silica gel and then over alumina. The product thus obtained is purified again by kugelrohr distillation. 3.6 g (12 mmol=32%) of the title compound are obtained as a colorless oil.

¹H-NMR (CDCl₃; δ (ppm)): 7.6 (m, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (dd, broad, 2H, O—CH₂); 3.8 (m, 1H, N—CH_(A)); 3.6 (s, 3H, O—CH₃); 3.5 (m, 1H, N—CH_(B)); 2.3 (s, 3H, CH₃); 1.15 (t, 3H, J=8 Hz, CH₃)

Example 2 Methyl N-[2-(2′-methylphenoxymethyl)-phenyl]-N-methylthiocarbamate (Table 7, No. 89)

a) 2-(2′-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide are stirred for 5 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and filtered off under suction. 73 g (0.300 mol=88%) of the title compound are obtained as a colorless solid.

mp.=83° C.

¹H-NMR (CDCl₃; δ (ppm)): 8.15 (d, 1H, J=8 Hz, aromatic); 7.95 (d, 1H, J=8 Hz, aromatic); 7.7 (t, 1H, J=8 Hz, aromatic); 7.45 (t, 1H, J=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O—CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2′-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2′-methylphenoxymethyl)nitrobenzene (Example 2a) and 10 g of 5% strength Pt/C (platinum adsorbed onto active carbon) in 50 ml of methanol are stirred vigorously for two hours under an H₂ atmosphere. Thereafter, a further 2 g of 5% strength Pt/C are added and stirring is continued overnight. The catalyst is then filtered off under suction and is replaced with 10 g of fresh catalyst. Stirring is continued overnight, the mixture is filtered under suction and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography using hexane/ethyl acetate mixtures. 61 g (0.286 mol=93%) of the title compound are obtained as a colorless solid.

mp.=56° C.

¹H-NMR (CDCl₃; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, J=8 Hz, aromatic); 6.9 (t, 1H, J=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (s, 2H, O—CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) Methyl N-[2-(2′-methylphenoxymethyl)-phenyl]carbamate (Table 7, No. 3)

6 g (63 mmol) of methyl chloroformate are added dropwise to 10 g (47 mmol) of 2-(2′-methylphenoxymethyl)aniline in 500 of methylene chloride at 20-30° C. Stirring is carried out for 3 hours at room temperature, a white solid being precipitated, and the reaction mixture is then stirred with 20 ml of 10% strength sodium hydroxide solution. The organic phase is filtered off under suction over silica gel, the filtrate is evaporated down and the remaining residue is stirred thoroughly with methanol and filtered under suction. 10.5 g (39 mmol=82%) of the title compound are obtained as a colorless solid.

mp.=111° C.

¹H-NMR (CDCl₃; δ (ppm)): 8.0 (d, broad, 1H, aromatic); 7.7 (s, broad, 1H, aromatic); 7.7 (s, broad, 1H, NH); 6.8-7.5 (m, 6H, aromatic); 5.0 (s, 2H, O—CH₂); 3.75 (s, 3H, O—CH₃); 2.25 (s, 3H, CH₃)

d) Methyl N-[2-(2′-methylphenoxymethyl)-phenyl]-N-methylthiocarbamate (Table 7, No. 89)

0.5 g (20.8 mmol) of sodium hydride is added a little et a time to 4.9 g (17.3 mmol) of methyl N-[2-(2′-methylphenoxymethyl)]-phenylcarbamate (Example 2c) in 80 ml of toluene. After the end of gas evolution, 2.4 g (19 mmol) of methyl methanethiosulfonate are added and stirring is carried out overnight at room temperature.

Thereafter, the reaction mixture is extracted with water, dried over MgSO₄ and evaporated down under reduced pressure. The residue is purified by column chromatography with hexane/ethyl acetate mixtures over silica gel. 3 g (9.1 mmol=53%) of the title compound are obtained as a yellow oil.

¹H-NMR (CDCl₃; δ (ppm)): 7.65 (d, broad, 1H, aromatic); 7.35 (m, 2H, aromatic); 7.15 (m, 3H, aromatic); 6.85 (m, 2H, aromatic); 5.0 (m, 2H, O—CH₂); 3.75 (s, 3H, O—CH₃); 2.55 (s, 3H, S—CH₃); 2.3 (s, 3H, CH₃)

Example 3 Methyl N-allyl-N-[2-(3″-bromophenylmethyliminoxymethyl)phenyl]-carbamate (Table 7, No. 91)

a) o-Methoxymethylnitrobenzene

125 g of 30% strength sodium methylate solution (0.69 mol) in methanol are added dropwise to 130 g (0.6 mol) of o-nitrobenzyl bromide in 200 ml of methanol. During this procedure, the reaction mixture heats up to about 50° C. Stirring is continued for a further 3 hours, the reaction mixture being cooled to room temperature, after which ice water is added to the reaction vessel and the reaction mixture is neutralized by adding dilute hydrochloric acid. The aqueous phase is extracted with three times with ether, and the organic phase is dried over MgSO₄ and evaporated down. 101 g (0.6 mol, quantitative yield) of the title compound are obtained as a residue in the form of a brownish oil.

¹H-NMR (CDCl₃; δ (ppm)): 8.1 (d, broad, 1H, aromatic); 7.8 (d, broad, 1H, aromatic); 7.65 (t, broad, 1H, aromatic); 7.45 (t, broad, 1H, aromatic); 4.85 (s, 2H, O—CH₂); 3.5 (s, 3H, OCH₃)

b) Methyl N-(2-methoxymethylphenyl)-carbamate

528 g of 21.8% strength Na₂[Fe(CO)₄] solution (0.6 mol; 1 kg of the solution contains 633 g of water, 218 g of Na₂[Fe(CO)₄], 108 g of Na₂CO₃ and 41 g of NaOH) are added dropwise to 101 g (0.6 mol) of o-methoxymethylnitrobenzene (Example 3a) in 1 l of methanol at 20-30° C. Stirring is carried out for 1 hour at room temperature, after which the reaction mixture is diluted with ether. A brown oil separates out in the reaction vessel. The total reaction mixture is poured onto a silica gel column and is eluted with ether. Thereafter, the ether phase is evaporated, the residue is taken up in methylene chloride and the solution is dried over MgSO₄. It is filtered under suction over silica gel and the solvent is then evaporated off under reduced pressure. The residue is purified by column chromatography with hexane and methylene chloride. 83.8 g of o-methoxymethylaniline are obtained as a brown oil, which is directly reacted further.

The resulting crude product is dissolved in 700 ml of methylene chloride, 62.4 g (0.66 mol) of methyl chloroformate are added and 52.2 g (0.66 mol) of pyridine are then added dropwise. Stirring is carried out overnight at room temperature and the reaction mixture is then extracted with dilute hydrochloric acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with hexane/ethyl acetate mixtures. 89.4 g (0.41 mol=69%, based on 2-methoxymethylnitrobenzene) of the title compound are obtained as a yellow oil in a purity of about 90%.

¹H-NMR (CDCl₃; δ (ppm)): 8.0 (m, 2H, 1×aromatic, NH); 7.35 (t, broad, 1H, aromatic); 7.15 (d, broad, 1H, aromatic); 7.0 (t, broad, 1H, aromatic); 4.5 (s, 2H, OCH₂); 3.8 (s, broad, 3H, OCH₃); 3.4 (s, broad, 3H, OCH₃)

c) Methyl N-(2-bromomethylphenyl)-carbamate

38.6 g (150 mmol) of boron tribromide are added dropwise to 10 g (51 mmol) of methyl N-(2-methoxymethylphenyl)-carbamate (Example 2b) in 100 ml of methylene chloride. Stirring is carried out for 2 hours, after which the vigorously stirred reaction mixture is added dropwise to a solution of 11.8 g (0.17 mol) of NaHCO₃ in water. The organic phase is separated off and the aqueous phase is extracted once with methylene chloride and once with ethyl acetate. The combined organic phases are dried over MgSO₄ and evaporated down. 9.5 g (39 mmol=76%) of the title compound are obtained as a colorless solid.

mp.=132° C.

¹H-NMR (CDCl₃; δ (ppm)): 7.85 (d, broad, 1H, aromatic); 7.3 (m, 2H, aromatic); 7.1 (t, broad, 1H, aromatic); 6.9 (s, broad, 1H, NH); 4.5 (s, 2H, CH₂—Br); 3.8 (s, 3H, OCH₃)

d) Methyl N-[2-(3″-bromophenylmethyliminoxymethyl)phenyl]-carbamate (Table 7, No. 88)

0.95 g (39 mmol) of sodium hydride is added a little at a time to 7 g (33 mmol) of m-bromoacetophenone oxime in 100 ml of dimethylformamide. When the evolution of gas has ended, 8 g (33 mmol) of methyl N-(2-bromomethylphenyl)-carbamate (Example 3c), dissolved in 10 ml of dimethylformamide, are added dropwise. Stirring is carried out for 3 hours at room temperature, the reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The organic phase is washed three times with water, dried and evaporated down. The residue crystallizes and is stirred thoroughly with methanol. 5.1 g (13.5 mmol=41%) of the title compound are obtained as a colorless solid.

mp.=124-125° C.

¹H-NMR (CDCl₃; δ (ppm)): 8.6 (s, broad, 1H, NH); 7.8-8.1 (m, 2H, aromatic); 7-7.6 (m, 6H, aromatic); 5.2 (s, 2H, O—CH₂); 3.8 (s, 3H, O—CH₃); 2.2 (s, 3H, CH₃)

e) Methyl N-allyl-N-[2-(3″-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Table 7, No. 91)

0.1 g (4.1 mmol) of sodium hydride is added a little at a time to 1.3 g (3.5 mmol) of methyl N-[2-(3″-bromophenylmethyliminoxymethyl)-phenyl]-carbamate (Example 3d) in 20 ml of dimethylformamide. After gas evolution has ended, 0.5 g (3.8 mmol) of allyl bromide are added and stirring is carried out overnight at room temperature. Thereafter, the reaction mixture is diluted with water and extracted three times with ether. The combined ether phases are washed three times with water, dried over MgSO₄ and evaporated down. 1.5 g (quantitative yield) of the title compound are obtained as a residue in the form of a yellow oil.

¹H-NMR (CDCl₃; δ (ppm)): 7.8 (s, broad, 1H, aromatic); 7.1-7.6 (m, 7H, aromatic); 6.0 (m, 1H, C—CH═C); 5.1 (m, 4H, O—CH₂ and C═CH₂); 4.4 (m, 1H, N—CH_(A)); 4.0 (m, 1H, N—CH_(B)) 3.6-3.8 (2s, broad, O—CH₃); 2.2 (s, 3H, CH₃)

The compounds described in the Tables below can be prepared in a similar manner.

TABLE 1

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-s-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—H₃ 293 3-CO—CH₂—H₃ 294 4-CO—CH₂—H₃ 295 2-CO—CH₂—H₂—CH₃ 296 3-CO—CH₂—H₂—CH₃ 297 4-CO—CH₂—H₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—H₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—CO₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H II: R¹ = CH₃ III: R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂—CN VII: R¹ = CH₂—O—CH₃ VIII: R¹ = CO—OCH₃

TABLE 2

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyi-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH₃-Oxazolyl-4 234 3-C₆H₅-Oxazolyl-4 235 3-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 3-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 3-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 3-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 3-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 3-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 3-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 3-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 3-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 3-(4′-CN—C₆H₄)-Oxazolyl-4 245 3-(3′-CN—C₆H₄)-Oxazolyl-4 246 3-(2′-CN—C₆H₄)-Oxazolyl-4 247 3-(4′-Cl—C₆H₄)-Oxazolyl-4 248 3-(3′-Cl—C₆H₄)-Oxazolyl-4 249 3-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazo1y1-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl I: R¹ = H II: R¹ = CH₃ III: R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂—CN VII: R¹ = CH₂—O—CH₃ VIII: R¹ = CO—OCH₃

TABLE 3

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4- (2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-C-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)-CH₃ 299 3-CO—CH(CH₃)-CH₃ 300 4-CO—CH(CH₃)-CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH (CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-C-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NCAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—CO₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H II: R¹ = CH₃ III: R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂—CN VII: R¹ = CH₂—O—CH₃ R¹ = CO—OCH₃

TABLE 4

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₄-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazoiyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl I: R¹ = H II: R¹ = CH₃ III: = R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂CN VII: R¹ = CH₂—O—CH₃ VIII: R¹ = CO—OCH₃

TABLE 5

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉ ₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-C-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₆H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-C(₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₂H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F-C₆H₄) 387 2-(3′-F-C₆H₄) 388 2-(4′-F-C₆H₄) 389 3-(2′-F-C₆H₄) 390 3-(3′-F-C₆H₄) 391 3-(4′-F-C₆H₄) 392 4-(2′-F-C₆H₄) 393 4-(3′-F-C₆H₄) 394 4-(4′-F-C₆H₄) 395 2-(2′-Cl-C₆H₄) 396 2-(3′-Cl-C₆H₄) 397 2-(4′-Cl-C₆H₄) 398 3-(2′-Cl-C₆H₄) 399 3-(3′-Cl-C₆H₄) 400 3-(4′-Cl-C₆H₄) 401 4-(2′-Cl-C₆H₄) 402 4-(3′-Cl-C₆H₄) 403 4-(4′-Cl-C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NoAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄ 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃C—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃C—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 478 3-O—C₆H₅ 476 4-C—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NO—C₆H₄) 552 2-O-(3′-NO—C₆H₄) 553 2-O-(4′-NO—C₆H₄) 554 3-O-(2′-NO—C₆H₄) 555 3-O-(3′-NO—C₆H₄) 556 3-O-(4′-NO—C₆H₄) 557 4-O-(2′-NO—C₆H₄) 558 4-O-(3′-NO—C₆H₄) 559 4-O-(4′-NO—C₆H₄) 560 2-O-(2′-CF₃—C₆H₅) 561 2-O-(3′-CF₃—C₆H₅) 562 2-O-(4′-CF₃—C₆H₅) 563 3-O-(2′-CF₃—C₆H₅) 564 3-O-(3′-CF₃—C₆H₅) 565 3-O-(4′-CF₃—C₆H₅) 566 4-O-(2′-CF₃—C₆H₅) 567 4-O-(3′-CF₃—C₆H₅) 568 4-O-(4′-CF₃—C₆H₅) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isozazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = H II: R¹ = CH₃ III: R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂—CN VII: R¹ = CH₂—O—CH₃ VIII: R¹ = CO—OCH₃

TABLE 6

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 I: R¹ = H II: R¹ = CH₃ III: R¹ = Allyl IV: R¹ = Propargyl V: R¹ = S—CH₃ VI: R¹ = CH₂—CN VII: R¹ = CH₂—O—CH₃ VIII: R¹ = CO—OCH₃

TABLE 7 Selected physical data of some compounds No. Compound mp/° C. IR/cm⁻¹ 4 1

— 1707, 1484, 1457 1447, 1303, 1277 2

— 1708, 1495, 1457 1449, 1304, 1241 3

111 4

 73 5

 54 6

— 1706, 1496, 1456 1447, 1294, 1241 7

 73 8

 57 9

 86 10

— 1709, 1599, 1497 1453, 1346, 1241 11

— 1708, 1599, 1497 1455, 1447, 1397 1238 12

— 1740, 1593, 1527 1489, 1456, 1252 1225 13

— 1710, 1603, 1584 1490, 1451, 1364 1254 14

— 1709, 1490, 1456, 1447, 1379, 1300, 1258 15

— 1712, 1490, 1456 1447, 1378, 1298 1259 16

 88 17

— 1710, 1511, 1451 1364, 1302, 1238 18

— 1709, 1511, 1456 1447, 1379, 1301 1236 19

— 1712, 1511, 1447 1378, 1298, 1233 20

— 1738, 1723, 1582 1522, 1452, 1223 21

— 1711, 1492, 1480 1447, 1362, 1303 1192, 1159 22

— 1708, 1491, 1479 1446, 1376, 1300 1277, 1150 23

— 1712, 1511, 1447 1378, 1298, 1233 24

— 1736, 1582, 1523 1453, 1221 25

— 1706, 1495, 1485 1363, 1303, 1193 1160 26

— 1706, 1484, 1447 1377, 1301, 1280 1150 27

— 1710, 1495, 1483 1446, 1376, 1299 1233 28

 92 29

— 1709, 1489, 1447 1362, 1303, 1192 1159 30

— 1706, 1484, 1447 1377, 1301, 1280 1150 31

— 1711, 1488, 1446 1375, 1299, 1232 32

132 33

— 1709, 1495, 1486 1451, 1366, 1161 1008 34

— 1708, 1487, 1455, 1447, 1379, 1300, 1009 35

— 1711, 1488, 1447 1378, 1297, 1232 1023, 1008 36

— 1696, 1532, 1515 1453, 1267, 1245 1069 37

— 1712, 1486, 1447 1361, 1303, 1191 1160 38

— 1708, 1485, 1446 1376, 1300, 1274 39

— 1709, 1484, 1446 1374, 1297, 1277 1232 40

— 1712, 1495, 1457 1447, 1378, 1298 1237 41

110 42

— 1739, 1593, 1528 1511, 1457, 1226 1035 43

102 44

— 1708, 1513, 1457 1447, 1378, 1302 1246, 1035 45

102 46

 74 47

— 1709, 1606, 1512 1364, 1245, 1228 1171, 1162, 1033 1005 48

 59 1709, 1447, 1364 1261, 1157, 1034 1007 49

— 1709, 1576, 1446 1379, 1300, 1260 1239, 1156, 1037 50

— 51

 89 52

— 1740, 1593, 1575 1527, 1457, 1316 1300, 1224, 1067 1029 53

 81 54

— 1711, 1574, 1447 1365, 1322, 1303 1213, 1160, 1033 1008 55

— 1709, 1574, 1446, 1378, 1321, 1301, 1284, 1213, 1034 56

— 1711, 1505, 145 1365, 1304, 124 1160, 1143, 1035 1007 57

 63 58

— 1710, 1487, 1450 1364, 1301, 1246 1160, 1030, 1006 59

— 1708, 1487, 1449 1378, 1300, 1247 1030, 1009 60

— 1743, 1593, 1528 1502, 1457, 1301 1255, 1190, 1066 1006 61

 77 62

— 1712, 1503, 1453 1363, 1303, 1259 1244, 1160, 1136 1006 63

— 1711, 1503, 1457 1447, 1380, 1301 1258, 1239, 1136 1015 64

 92 1743, 1593, 1528 1502, 1457, 1301 1255, 1190, 1066 1006 65

 90 66

 70 67

 75 68

108 69

 93 70

 74 71

— 1712, 1504, 1450 1363, 1303, 1255 1222, 1159, 1134 72

— 1712, 1510, 149 1450, 1365, 132 1246, 1150, 103 1005 73

 60 74

— 1711, 1509, 149 1451, 1363, 130 1264, 1193, 115 1129 75

— 1710, 1496, 1475 1149, 1365, 1301 1263, 1195, 1159 76

 66 77

 86 78

 91 79

100 80

— 1710, 1593, 1497 1452, 1364, 1323 1297, 1193, 1165 1153 81

— 1715, 1510, 1447 1367, 1324, 1299 1243, 1149, 1027 996 82

— 1710, 1509, 1456 1446, 1377, 1326 1300, 1241, 1149 1306 83

— 1723, 1509, 1453 1437, 1316, 1292 1241, 1149, 1064 1036 84

— 1738, 1611, 1581 1539, 1446, 1312 1301, 1231, 1201 1067 85

— 1713, 1504, 1447 1375, 1313, 1300 1233, 1143, 1027 86

— 1711, 1486, 1447 1376, 1300, 1281 1150, 1034, 1013 87

— 1714, 1487, 1447 1376, 1300, 1231 1023, 999 88

— 1733, 1594, 1533 1457, 1306, 1231 1013, 984 89

— 1721, 1495, 1453 1437, 1313, 1290 1239, 1123 90

— 1709, 1453, 1366 1303, 1228, 1160 1014 91

— 1708, 1455, 1447 1378, 1299, 1282 1015, 996 92

— 1710, 1447, 1378 1296, 1232, 1045 1023, 995 93

108 94

— 1717, 1495, 1457 1444, 1376, 1298 1241, 1228, 1193 95

— 1739, 1614, 1603 1542, 1450, 1262 129, 1179 96

170 97

180 98

173 99

150 100

129 101

112 102

116 103

127 104

108 105

— 1710, 1486, 1447 1363, 1307, 1193 1159, 1031, 1006 919 106

— 1706, 1448, 1447 1376, 1302, 1279 1150, 1031, 1011 923 107

— 1711, 1484, 1446 1376, 1298, 1232 1144, 1024, 995, 922 108

147 109

1716, 1455, 1445 1376, 1297, 1279 1097, 1069, 1017 1008 110

1718, 1487, 1447 1394, 1374, 1306 1232, 1025, 1008 111

109 112

1706, 1487, 1450 1387, 1304, 1276 1155, 1022, 1009 769 113

1706, 1487, 1453 1383, 1312, 1301 1274, 1155, 1033 1008 114

115 115

167 116

1729, 1575, 1565 1545, 1523, 1445 1434, 1224, 1060 117

110 118

 77 119

1712, 1494, 1447 1378, 1298, 1232 1045, 1024, 818, 771 120

115 121

1717, 1455, 1445 1376, 1298, 1278 1097, 1068, 1016 999 122

 81 123

1712, 1493, 1447, 1378, 1297, 1232, 1047, 1024, 998, 772 124

107 125

1717, 1455, 1445 1376, 1298, 1279 1096, 1068, 1017 999 126

128 127

1712, 1492, 1447 1378, 1298, 1232 1096, 1044, 1023 128

119 129

1717, 1492, 1455 1445, 1376, 1298 1096, 1068, 1012 1000 130

133 131

1712, 1511, 1494 1447, 1378, 1298 1232, 1045, 1024 837 132

113 133

1716, 1511, 1455 1445, 1376, 1298 1228, 1097, 1068 999 134

1737, 1592, 1529 1509, 1489, 1455 1303, 1231, 1067 1014 135

1712, 1586, 1507 1489, 1454, 1378 1297, 1239, 1023 136

148 137

1716, 1587, 1507 1490, 1455, 1375 1298, 1240, 1068 138

 90 139

1719, 1495, 1464 1446, 1375, 1295 1239, 1104, 1075 1014 140

1715, 1495, 1463 1448, 1376, 1298 1239 141

134 142

1744, 1583, 1522 1503, 1458, 1442 1223, 1304, 1035 1004 143

1720, 1465, 1446 1372, 1296, 1280 1243, 1144, 1035 1014 144

1716, 1505, 1465 1448, 1374, 1298 1279, 1241, 1141 999 145

109 146

158 147

1718, 1463, 1445 1376, 1294, 1104 1073, 1024, 1010 148

1714, 1462, 1447 1377, 1297, 1238 1025, 1009 149

140

Example 4 Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14, No. 1)

a) Methyl N-(2-methylphenyl)-N-hydroxy-carbamate

At 25-30° C., 14.0 g (0.148 mol) of methyl Chloroocarbonate is added dropwise to 16.4 g of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Ann. Chem. 316 (1901), 278) and 12.9 g (0.163 mol) of pyridine in 100 ml of methylene Chloroide. The mixture is stirred overnight at room temperature (20° C.) and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 7 g (39 mmol) of the title compound as a yellow oil.

¹H-NMR (CDCl₃; δ (ppm): 8.6 (s, broad, OH); 7.3 (m, 4H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

b) Methyl N-(2-methylphenyl)-N-methoxy-carbamate (Table 14 No. 1)

At 20-30° C., 1.1 g (44.1 mmol) of sodium hydride is added in portions to 6.6 g (36.5 mmol) of the hydroxyl compound from Example 4a in 50 ml of dimethylformamide. Upon conclusion of gas evolution 5.7 g (40.1 mmol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is the diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtains 40 5.2 g (27 mmol=73%) of the title compound as a yellow oil.

¹H-NMR (CDCl₃; δ in ppm):

7.25 (m, 4H, phenyl); 3.8; 3.75 (s, 3H, OCH₃; 3.75 (s, 3H, OCH₃); 2.3 (s, 3H , CH₃)

Example 5 Methyl N-(2-bromomethylphenyl)-N-methoxy-carbamate (Table 14, No. 2)

2.5 g (12.8 mmol) of the N-methoxycarbamate from Example 4b, 2.5 g (14.1 mmol) of N-bromosuccinimide and a spatula-tip (1 g) of azoisobutyrodinitrile in 20 ml of carbon tetrachlo roide were irradiated with a 300 W UV lamp; the reaction mixture heated up to 30-40° C. After three hours the reaction mixture is extracted twice with water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.4 g (5.1 mmol=40%) of the title compound as a yellow oil.

¹H-NMR (CDCl₃; δ in ppm): 7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.55 (s, 2H, CH₂—Br); 3.8 (2s, 6H, 2xOCH₃)

Example 6 Methyl N-[2-(2′-methylphenoxymethyl)-phenyl]-N-methoxy-carbamate (Table 14, No. 3)

1.2 g (4.4 mmol) of the methyl bromide from Example 5, 0.4 g (4.2 mmol) o-cresol and 0.7 g (4.8 mmol) of K₂CO₃ in 30 ml of dimethylformamide are stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl-t-butyl ether. The combined organic phases are dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 1.2 g of the title compound containing o-cresol as impurity. The mixture is heated in a furnace at about 1 mbar for about 1 hour at 125° C. The residue obtained is 0.9 g (3 mmol=68%) of the title compound as a yellow oil.

¹NMR (CDCl₃; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 7.15 (m, 2H, phenyl); 6.9 (t, broad, 2H, phenyl); 5.15 (s, 2H, O—CH₂); 3.8 (s, 3H, OCH₃), 3.75 (s, 3H, OCH₃); 2.3 (s, 3H, CH₃)

TABLE 8

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F5 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C2H5)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH3, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO2 251 2-NO2, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl2, 5-NO2 254 2,4-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, 4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO₂CH₃ 260 3-CO2CH3 261 4-CO2CH3 262 2-CO2(C2H5) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH_(2O)(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH3O2C—C6H4) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C6H5 476 4-O—C6H5 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O-—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₄ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = CH₃ II: R¹ = CH₂—CH₃

TABLE 9

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Fury1-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃ II: R¹ = CH₂—CH₃

TABLE 10

I: II: R¹ = CH₃ R¹ = CH₂—CH₃ No. X_(m)  1 H  2 2-F  3 3-F  4 4-F  5 2,4-F₂  6 2,4,6-F₃  7 2,3,4,5,6-F₅  8 2,3-F₂  9 2-Cl  10 3-Cl  11 4-Cl  12 2,3-Cl₂  13 2,4-Cl₂  14 2,5-Cl₂  15 2,6-Cl₂  16 3,4-Cl₂  17 3,5-Cl₂  18 2,3,4-Cl₃  19 2,3,5-Cl₃  20 2,3,6-Cl₃  21 2,4,5-Cl₃  22 2,4,6-Cl₃  23 3,4,5-Cl₃  24 2,3,4,6-Cl₄  25 2,3,5,6-Cl₄  26 2,3,4,5,6-Cl₅  27 2-Br  28 3-Br  29 4-Br  30 2,4-Br₂  31 2,5-Br₂  32 2,6-Br₂  33 2,4,6-Br₃  34 2,3,4,5,6-Br₅  35 2-I  36 3-I  37 4-I  38 2,4-I₂  39 2-Cl, 3-F  40 2-Cl, 4-F  41 2-Cl, 5-F  42 2-Cl, 6-F  43 2-Cl, 3-Br  44 2-Cl, 4-Br  45 2-Cl, 5-Br  46 2-Cl, 6-Br  47 2-Br, 3-Cl  48 2-Br, 4-Cl  49 2-Br, 5-Cl  50 2-Br, 3-F  51 2-Br, 4-F  52 2-Br, 5-F  53 2-Br, 6-F  54 2-F, 3-Cl  55 2-F, 4-Cl  56 2-F, 5-Cl  57 3-Cl, 4-F  58 3-Cl, 5-F  59 3-Cl, 4-Br  60 3-Cl, 5-Br  61 3-F, 4-Cl  62 3-F, 4-Br  63 3-Br, 4-Cl  64 3-Br, 4-F  65 2,6-Cl₂, 4-Br  66 2-CH₃  67 3-CH₃  68 4-CH₃  69 2,3-(CH₃)₂  70 2,4-(CH₃)₂  71 2,5-(CH₃)₂  72 2,6-(CH₃)₂  73 3,4-(CH₃)₂  74 3,5-(CH₃)₂  75 2,3,5-(CH₃)₃  76 2,3,4-(CH₃)₂  77 2,3,6-(CH₃)₃  78 2,4,5-(CH₃)₃  79 2,4,6-(CH₃)₃  80 3,4,5-(CH₃)₃  81 2,3,4,6-(CH₃)₄  82 2,3,5,6-(CH₃)₄  83 2,3,4,5,6-(CH₃)₅  84 2-C₂H₅  85 3-C₂H₅  86 4-C₂H₅  87 2,4-(C₂H₅)₂  88 2,6-(C₂H₅)₂  89 3,5-(C₂H₅)₂  90 2,4,6-(C2H5)3  91 2-n-C₃H₇  92 3-n-C₃H₇  93 4-n-C₃H₇  94 2-i-C₃H₇  95 3-i-C₃H₇  96 4-i-C₃H₇  97 2,4-(i-C₃H₇)₂  98 2,6-(i-C₃H₇)₂  99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇), 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O-C₂H₅ 164 4-O-C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F2, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂-OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)-CH₃ 299 3-CO—CH(CH₃)-CH₃ 300 4-CO—CH(CH₃)-CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃-CH₂—CH₂—CO 305 2-Me-4-CH₃-CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃₎—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃--CH(CH₃₎—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 34i 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH_(3-4-(C) ₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃-C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃-C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃-C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃-C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃-C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃-C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N-C₆H₄) 451 2-(3′-O₂N-C₆H₄) 452 2-(4′-O₂N-C₆H₄) 453 3-(2′-O₂N-C₆H₄) 454 3-(3′-O₂N-C₆H₄) 455 3-(4′-O₂N-C₆H₄) 456 4-(2′-O₂N-C₆H₄) 457 4-(3′-O₂N-C₆H₄) 458 4-(4′-O₂N-C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C6H5 476 4-O—C6H5 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N-C₆H₄) 543 2-O-(3′-O₂N-C₆H₄) 544 2-O-(4′-O₂N-C₆H₄) 545 3-O-(2′-O2N-C6H4) 546 3-O-(3′-O₂N-C₆H₄) 547 3-O-(4′-O₂N-C₆H₄) 548 4-O-(2′-O₂N-C₆H₄) 549 4-O-(3′-O₂N-C₆H₄) 550 4-O-(4′-O₂N-C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 664 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-l′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 63i 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-S-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₉ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C)H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 11

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Fury1-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazoiyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-.CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄′)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃-C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1, 2, 4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH_(3-1,2,4-Triazolyl-5) 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃ II: R¹ = CH₂—CH₃

TABLE 12

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-Cl₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH_(3‘—CH) ₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chlorallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—O(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = CH₃ II: R¹ = CH₂—CH₃

TABLE 13

I: R¹ = CH₃ II: R¹ = CH₂—CH₃ No. B 1 Pyrrolyl-3 2 N-CH₃-Pyrrolyl-3 3 N-C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅-N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)-N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)-N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)-N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)-N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)-N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)-N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 257 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3

TABLE 14 Selected physical data of some compounds No. Compound ¹H-NMR (ppm) 1

3.8(s, 3H); 3.75(s, 3H) 2

3.8(2s, 2 × 3H) 3

3.8(s, 3H); 3.75(s, 3H) 4

3.95(q, 2H, I = 7.5Hz); 3.8(s, 3H) 5

4.05(q, 2H, I = 7.5Hz); 3.85(s, 3H) 6

4.0(q, 2H, I = 7.5Hz); 3.8(s, 3H) 7

3.8(s, 3H); 3.75(s, 3H) 8

3.8(s, 3H); 3.75(s, 3H) 9

3.85(s, 3H); 3.8 (s, 3H) 10

4.0(s, 3H); 3.8(s, 3H), 3.75(s, 3H) 11

3.8(s, 3H); 3.75(s, 3H) 12

3.8(s, 3H); 3.75(s, 3H) 13

3.8(s, 3H); 3.75(s, 3H) 14

3.8(s, 3H); 3.75(s, 3H) 66 15

3.8(s, 3H); 3.75(s, 3H) 16

4.0(q, 2H, I = 7.5Hz); 3.8(s, 3H) 17

3.8(2s, each 3H) 18

3.8(2s, each 3H) 19

3.8(s, 3H); 3.75(s, 3H) 20

3.8(s, 3H); 3.75(s, 3H) 21

3.8(s, 3H); 3.75(s, 3H) 22

3.8(s, 3H); 3.75(s, 3H) 23

3.8(s, 3H); 3.75(s, 3H) 24

3.8(s, 6H) 25

3.75(2s, each 3H) 26

3.8(s, 3H); 3.75(s, 3H) 27

3.8(s, 3H); 3.75(s, 3H) 28

3.8(s, 3H); 3.75(s, 3H) 29

3.8(s, 3H); 3.75(s, 3H) 30

3.8(s, 6H)

TABLE 52 Selected physical data of some compounds

¹H-NMR (ppm) or IR No. X_(m) mp (° C.) (cm⁻¹) 1 H 3.75(2s, each 3H) 2 2-CH₃ 3.75(2s, each 3H) 3 3-CH₃ 3.75(2s, each 3H) 4 2,4-(CH₃)₂ 3.75(2s, each 3H) 5 4-C₂H₅ 3.75(2s, each 3H) 6 4-i-C₃H₇ 3.75(2s, each 3H) 7 4-t-C₄H₉ 3.75(2s, each 3H) 8 3,4-(CH₃)₂ 3.75(2s, each 3H) 9 3-Cl 3.75(2s, each 3H) 10 3-Br 3.75(2s, each 3H) 11 3-CF₃ 3.75(2s, each 3H) 12 4-Br 3.75(2s, each 3H) 13 4-F 3.75(2s, each 3H) 14 4-CF₃ 3.75(2s, each 3H) 15 4-OCH₃ 3.8(s, 3H); 3.75(2s, each 3H) 16 4-CN 3.75(2s, each 3H) 17 3-CH₃-4-O-i-C₃H₇ 3.75(2s, each 3H) 18 3,4-Cl₂ 3.75(2s, each 3H) 19 3-CH₃-4-OCH₃ 3.85(s, 3H); 3.75 (2s, each 3H) 20 4-NO₂ 112 21 3,5-(CH₃)₂ 3.75(2s, each 3H) 22 3-CH₃-4-Cl 3.75(2s, each 3H) 23 3-Cl-4-CH₃ 3.75(2s, each 3H)

TABLE 53 Selected physical data of some compounds

mp ¹H-NMR (ppm) or No. X_(m) (° C.) IR (cm⁻¹) 1 2-CH₃-4-C(CH₃)═N—O—C₂H₅ 3.8(s, 3H); 3.75(s, 3H) 2 2-CH₃-4-C(CH₃)═N—O- 3.8(s, 3H); 3.75(s, 3H) (trans-CH₂—CH═CHCl) 3 2,5-(CH₃)₂-4-C(CH₃)═N— 3.95(s, 3H); 3.8(s, 3H); OCH₃ 3.75(s, 3H) 4 2,5-(CH₃)₂-4-C(CH₃)═N— 3.8(s, 3H); 3.75(s, 3H) OC₂H₅ 5 2,5-(CH₃)₂-4-C(CH₃)═N—O- 3.85(s, 3H); 3.75(s, 3H) (trans-CH₂—CH═CHCl) 6 2-CH₃-4-C(C₂H₅)═N—OCH₃ 3.95(s, 3H); 3.8(s, 3H); 3.75(s, 3H) 7 2-CH₃-4-C(C₂H₅)═N— 3.8(s, 3H); 3.75(s, 3H) O—C₂H₅ 8 2-CH₃-4-C(C₂H₅)═N—O- 3.8(s, 3H); 3.75(s, 3H) Allyl 9 2-CH₃-4-C(C₂H₅)═N—O- 3.8(s, 3H); 3.75(s, 3H) (trans-CH₂—CH═CHCl) 10 2,5-(CH₃)₂-4-C(C₂H₅)═N— 3.95(s, 3H); 3.8(s, 3H); OCH₃ 3.75(s, 3H) 11 2,5-(CH₃)₂-4-C(C₂H₅)═N— 3.8(s, 3H); 3.75(s, 3H) O—C₂H₅ 12 2,5-(CH₃)₂-4-C(C₂H₅)═N— 3.8(s, 3H); 3.75(s, 3H) O-Allyl 13 2-Cl 3.8(s, 3H); 3.75(s, 3H) 14 4-Cl 3.8(s, 3H); 3.75(s, 3H) 15 2-CH₃-4-Cl 3.8(s, 3H); 3.75(s, 3H) 16 2-Cl-4-CH₃ 3.8(s, 3H); 3.75(s, 3H) 17 2-Cl-5-CH₃ 3.8(s, 3H); 3.75(s, 3H) 18 2,5-(CH₃)₂-4-C(CH₃)═N— 3.8(s, 3H); 3.75(s, 3H) O-Allyl 19 2,5-(CH₃)₂-4-C(C₂H₅)═N— 3.8(s, 3H): 3.75(s, 3H) O-(trans-CH₃—CH═CHCl)

TABLE 54

No. B 1 2-Pyridyl 2 3-Trifluormethyl-2-pyridyl 3 5-Trifluormethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-4-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimi- dazo[5,4-a]-pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl I: R¹ = CH₃ II: R¹ = C₂H₅

TABLE 55 Selected physical data of some compounds

No. X_(m) mp (° C.) ¹H-NMR (ppm) or IR (cm⁻¹) 1 H 3.75(s, 3H); 3.65(s, 3H) 2 4-OCH₃ 3.8(s, 3H); 3.75(s, 3H); 3.65(s, 3H) 3 4-CH₃ 3.75(s, 3H); 3.65(s, 3H) 4 4-Cl 3.75(s, 3H); 3.65(s, 3H) 5 4-CF₃ 3.75(s, 3H); 3.65(s, 3H) 6 3,5-(CF₃)₂ 3.75(s, 3H); 3.65(s, 3H) 7 2,4-Cl₂ 3.75(s, 3H); 3.65(s, 3H) 8 3,4-Cl₂ 3.75(s, 3H); 3.65(s, 3H)

Example 6 O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

a) N-(2-Methylphenyl)-N-propionyl-hydroxylamine

At 25 to 30° C., 12,5 g (0.135 mol) of propionyl Chloroide and then 10.7 g (0.135 mol) of pyridine are dripped into 30 g of N-(2-methylphenyl)-hydroxylamine (crude product, prepared according to Bamberger et al., Anm. Chem. 316 (1901), 278; content approx. 80%{circumflex over (=)}0.2 mol) in 500 ml of methylene Chloroide. The mixture is stirred for 30 minutes at room temperature, and is then extracted with dilute hydroChloroic acid and water. The organic phase is dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 22.7 g (0.127 mol{circumflex over (=)}63%) of the title compound as a yellow oil.

¹H-NMR (COCl₃; δ in ppm): 9.4 (s, broad, 1H, OH); 7.2 (m, 4H, phenyl); 2.4 (s, 3H, CH₃); 2.1 (q, broad, 2H, CH₂); 1.1 (t, 3H, I=7 Hz, CH₃)

b) O-Methyl-N-(2-methylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 1)

At 25 to 30° C., a solution of 22.7 g (0.127 mol) (Example 6a) of N-(2-methylphenyl)-N-propionyl-hydroxylamine in 50 ml of dimethylformamide is dripped into a stirred mixture of 3.4 g (0.14 mol) of NaH in 150 ml of dimethylformamide. After completion of gas evolution (15 mins) 18.4 g (0.13 mol) of methyl iodide is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 18 g (0.081 mol{circumflex over (=)}64%) of the title compound as a yellow oil.

¹H-NMR (COCl₃; δ in ppm): 7.2 (m, 4H, phenyl); 3.7 (s, broad, 3H, OCH₃); 2.6 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (s, broad, 3H, CH₃)

Example 7 O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine (Table 21, No. 2)

A mixture of 10 g (51.8 mmol) of the hydroxylamine derivative from Example 1, 11 g (61 mmol) of N-bromosuccinimide and 0.1 g of azoisobutyrodinitrile in 100 ml of CCl₄ is refluxed. One drop of bromine is added and the mixture is refluxed for a further 2.5 hours. The reaction mixture is cooled to room temperature, washed with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained in this sequence 3.4 g (7.9 mmol{circumflex over (=)}15%) of O-methyl-N-(2-bromomethylphenyl)-d-(α,α-dibromopropionyl)-hydroxylamine, 3.8 g (10.8 mmol{circumflex over (=)}21%) of O-methyl-N-(2-bromomethylphenyl)-N-(α-bromopropionyl)-hydroxylamine, 2.3 g (8.5 g (8.5 mmol{circumflex over (=)}16%) of the title compound and 3.5 g of starting material, each as brown oils.

a) O-Methyl-N-(2-bromomethylphenyl)-N-(α,α-dibromopropionyl)-hydroxylamine

7.55 (m, 1H, phenyl); 7.4 (m, 3H, phenyl); 4.5 (s, 2H, CH₂, Br); 3.8 (s, 3H, OCH₃); 2.75 (s, 3H, CH₃)

b) O-Methyl-N-(2-bromomethylphenyl)-N-(δ-bromopropionyl)-hydroxylamine

7.5 (s, broad, 1H, phenyl); 7.4 (s, broad, 3H, phenyl); 5.15 (s, broad, 1H, CH—Br); 4.5 (dd, broad, 2H, CH₂—Br); 3.8 (s, 3H, OCH₃); 1.85 (s, broad, 3H, CH₃)

c) O-Methyl-N-(2-bromomethylphenyl)-N-propionyl-hydroxylamine

7.5 (m, 1H, phenyl); 7.35 (m, 3H, phenyl); 4.5 (s, broad, 2H, CH₂—Br); 3.75 (s, 3H, OCH₃); 2.55 (s, very broad, CH₂); 1.2 (t, 3H, I=7 Hz, CH₃)

Example 8 O-Methyl-N-(2-(2′-methylphenyloxymethyl)-phenyl)-N-propionyl-hydroxylamine (Table 21, No. 3)

0.12 g (5 mmol) of sodium hydride is added to a solution of 0.4 g (3.7 mmol) of o-cresol in 5 ml of dimethylformamide. Upon completion of gas evolution, 1 g (3.6 mmol) of the benzyl bromide from Example 2c is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is diluted with water and extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MgSO₄ and evaporated down. The residue is chromatographed with mixtures of cyclohexane and ethyl acetate using Al₂O₃ and silica gel. There is obtained 0.4 g (1.33 mmol{circumflex over (=)}37%) of the title compound as a yellow oil.

¹H-NMR (COCl₃; δ in ppm): 7.7 (d, broad, 1H, phenyl); 7.35 (m, 3H, phenyl); 7.1 (m, 2H, phenyl); 6.85 (t, broad, 2H, phenyl); 5.05 (s, 2H, OCH₃); 3.7 (s, 3H, OCH₃); 2.55 (s, very broad, 2H, CH₂); 2.3 (s, 3H, CH₃); 1.2 (t, broad, 3H, CH₃)

Example 9 N-Methyl-N′-methoxy-N′-2-methylphenylurea (Table 21, No. 5)

a) Phenyl N-hydroxy-N-(2-methylphenyl)-carbamate

A mixture of 2.5 g (20 mmol) of N-(2-methylphenyl)-hydroxylamine (crude product, obtained according to Bamberger et al., Anm. Chem. 316 (1901), 278), 3.5 g (25 mmol) of K₂CO₃ and 3.5 g (22 mmol) of phenyl Chlorooformate in 20 ml of CH₂Cl₂ is stirred for 2 hours at room temperature. The reaction mixture is then extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 2.0 g (8.2 mmol{circumflex over (=)}42%) of the title compound as a colorless solid (mp=98° C.).

¹H-NMR (COCl₃; δ in ppm): 7-7.6 (m, 10H, phenyl, OH); 2.35 (s, 3H, CH₃)

b) Phenyl N-methoxy-N-(2-methylphenyl)-carbamate

A mixture of 2.0 g (8.2 mmol) of the phenyl carbamate from Example 4a, 2 g (15 mmol) of K₂CO₃ and 1.3 g (10 mmol) of dimethyl sulfate in 20 ml of acetone is stirred for 3 hours at room temperature. The reaction mixture is then filtered and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.5 g (5.8 mmol{circumflex over (=)}71%) of the title compound as a colorless oil, which slowly crystallizes (mp=60° C.).

¹H-NMR (COCl₃; δ in ppm): 7.1-7.5 (m, 9H, phenyl); 3.8 (s, 3H, OCH₃); 2.4 (s, 3H, CH₃)

c) N-Methyl-N′-methoxy-N′-2-methylphenylurea (Table 21, No. 5)

1.5 g (5.8 mmol) of the phenyl carbamate from Example 4b in 20 ml of 40% strength aqueous methylamine solution is stirred for 1 hour at 50° C. The reaction mixture is then cooled and extracted with CH₂Cl₂. The combined organic phases are dried over MgCO₄ and evaporated down. The residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 0.6 g (3.1 mmol{circumflex over (=)}53%) of the title compound as a colorless solid (mp=99° C.).

¹H-NMR (COCl₃; δ in ppm): 7.2 (m, 4H, phenyl); 5.9 (s, broad, 1H, NH); 3.6 (s, 3H, OCH₃); 2.9 (d, 3H, I=approx. 2 Hz, N—CH₃); 2.3 (s, 3H, CH₃)

Example 18 N-Methyl-N′-methoxy-N′-(2-2′,5′-dimethylphenoxymethyl)phenyl)-urea

a) Phenyl N-methoxy-N-(2-bromomethylphenyl)-carbamate

A mixture of 125 g (0.486 mol) of methyl N-methoxy-N-(2-methylphenyl)-carbamate (Example 4b), 88 g (0.494 mol) of N-bromosuccinimide and 1 g of azoisobutyrodinitrile (AIBN) in 800 ml of CCl₄ is refluxed for about 12 hours. 10 g of N-bromosuccinimide is then added and the mixture is refluxed for about 4 hours. The reaction mixture is extracted with water and sodium thiosulfate solution, and the organic phase is dried over MgSO₄ and evaporated down under reduced pressure. The residue crystallizes, is stirred with hexane/methyl tert-butyl ether and suction dried. There is obtained 107 g (63%) of the title compound as a colorless solid.

¹H-NMR CDCl₃; δ in ppm): 7.1-7.6 (m, 9H, phenyl); 4.65 (s, 2H, CH₂Br); 3.9 (s, 3H, OCH₃)

b) Phenyl N-methoxy-N-(2-(2′,5′-dimethylphenoxymethyl)-phenyl)-carbamate

A mixture of 7 g (20 mmol) of the bromide of Example 5a and 3.3 g (22 mmol) of sodium iodide in 50 ml of acetone is refluxed for 30 minutes. The precipitated solid is then filtered off and the organic phase is evaporated down under reduced pressure. The crude product obtain is the iodide corresponding to Example 5a, which is used in the next reaction without any further purification.

The crude product obtained above is dissolved in 100 ml of dimethylformamide, 3 g (21.6 mmol) of K₂CO₃ and 7.3 g (60 mmol) of 2,5-dimethylphenol are added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography using methylene chloride/cyclohexane (1:2) over Al₂O₃. There is obtained 7.3,g (94%) of the title compound as a yellow oil.

¹H-NMR CDCl₃; δ in PPM): 7.7 (d, broad, 1H, phenyl); 7-7.6 (m, 9H, phenyl); 6.7 (m, 2H, phenyl); 5.2 (s, 2H, OCH₂); 3.85 (s, 3H, OCH₃); 2.3 (s, 6H, 2xCH₃).

c) N-Methyl-N′-methoxy-N′-(2-(2′,5′-dimethylphenoxymethyl)phenyl)-urea (Table 1, No. V.71)

A mixture of 3.4 g (8.8 mmol) of the phenyl carbamate of Example 5b and 20 ml of 40% strength aqueous methylamine solution is stirred for 2 hours at 50° C. The mixture is allowed to cool and is then extracted with methylene chloride. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of cyclohexane/ethyl acetate. There is obtained 1 g (36%) of the title compound as a colorless solid (mp=101° C.).

¹H-NMR CDCl₃; δ in PPM): 7.75 (m, 1H, phenyl); 6.6-7.4 (m, 6H, phenyl); 6.0 (s, broad, NH); 5.15 (s, 2H, OCH₂); 3.65 (s, 3H, OCH₃); 2.9 (d, 3H, N—CH₃); 2.3 (s, 3H, CH₃); 2.25 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared analogously. Compound I.1 from Table 15 has for instance the following formula

TABLE 15

I: II: III: IV: V: VI: R¹ = CH₃, Z = CH₃ R¹ = CH₂—CH₃, Z = CH₃ R¹ = CH₃, Z = C₂H₅ R¹ = CH₂—CH₃, Z = C₂H₅ R¹ = CH₃, Z = NHCH₃ # R¹ = CH₂—CH₃, Z = NHCH₃ No. Xm  1 H  2 2-F  3 3-F  4 4-F  5 2,4-F₂  6 2,4,6-F₃  7 2,3,4,5,6-F5  8 2,3-F₂  9 2-Cl  10 3-Cl  11 4-Cl  12 2,3-Cl₂  13 2,4-Cl₂  14 2,5-Cl₂  15 2,6-Cl₂  16 3,4-Cl₂  17 3,5-Cl₂  18 2,3,4-Cl₃  19 2,3,5-Cl₃  20 2,3,6-Cl₃  21 2,4,5-Cl₃  22 2,4,6-Cl₃  23 3,4,5-Cl₃  24 2,3,4,6-Cl₄  25 2,3,5,6-Cl₄  26 2,3,4,5,6-Cl₅  27 2-Br  28 3-Br  29 4-Br  30 2,4-Br₂  31 2,5-Br₂  32 2,6-Br₂  33 2,4,6-Br₃  34 2,3,4,5,6-Br₅  35 2-I  36 3-I  37 4-I  38 2,4-I₂  39 2-Cl, 3-F  40 2-Cl, 4-F  41 2-Cl, 5-F  42 2-Cl, 6-F  43 2-Cl, 3-Br  44 2-Cl, 4-Br  45 2-Cl, 5-Br  46 2-Cl, 6-Br  47 2-Br, 3-Cl  48 2-Br, 4-Cl  49 2-Br, 5-Cl  50 2-Br, 3-F  51 2-Br, 4-F  52 2-Br, 5-F  53 2-Br, 6-F  54 2-F, 3-Cl  55 2-F, 4-Cl  56 2-F, 5-Cl  57 3-Cl, 4-F  58 3-Cl, 5-F  59 3-Cl, 4-Br  60 3-Cl, 5-Br  61 3-F, 4-Cl  62 3-F, 4-Br  63 3-Br, 4-Cl  64 3-Br, 4-F  65 2,6-Cl₂, 4-Br  66 2-CH₃  67 3-CH₃  68 4-CH₃  69 2,3-(CH₃)₂  70 2,4-(CH₃)₂  71 2,5-(CH₃)₂  72 2,6-(CH₃)₂  73 3,4-(CH₃)₂  74 3,5-(CH₃)₂  75 2,3,5-(CH₃)₃  76 2,3,4-(CH₃)₃  77 2,3,6-(CH₃)₃  78 2,4,5-(CH₃)₃  79 2,4,6-(CH₃)₃  80 3,4,5-(CH₃)₃  81 2,3,4,6-(CH₃)₄  82 2,3,5,6-(CH₃)₄  83 2,3,4,5,6-(CH₃)₅  84 2-C₂H₅  85 3-C₂H₅  86 4-C₂H₅  87 2,4-(C2H5)₂  88 2,6-(C₂H₅₎ ₂  89 3,5-(C₂H₅₎ ₂  90 2,4,6-(C₂H₅₎ ₃  91 2-n-C₃H₇  92 3-n-C₃H₇  93 4-n-C₃H₇  94 2-i-C₃H₇  95 3-i-C₃H₇  96 4-i-C₃H₇  97 2,4-(i-C₃H₇)₂  98 2,6-(i-C₃H₇)₂  99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O-C₂H₅ 164 4-O-C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O-CH₂C₆H₅ 178 3-O-CH₂C₆H₅ 179 4-O-CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)_(3, 4-F) 244 2,3,6-(CH₃)_(3, 4-Cl) 245 2,3,6-(CH₃)_(3, 4-Br) 246 2,4-(CH₃)_(2, 6-F) 247 2,4-(CH₃)_(2, 6-Cl) 248 2,4-(CH₃)_(2, 6-Br) 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO2 251 2-NO2, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl2, 5-NO2 254 2,4-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, ,4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO₂CH₃ 260 3-CO2CH3 261 4-CO2CH3 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO-CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃——CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 2-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH3-4-(CH3—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C6H5 475 3-O—C6H5 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—C—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Proparoyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 16

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiaiolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1.3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazbiyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃, Z = CH₃ II: R¹ = CH₂—CH₃, Z = CH₃ III: R¹ = CH₃, Z = C₂H₅ IV: R¹ = CH₂—CH₃, Z = C₂H₅ V: R¹ = CH₃, Z = NHCH₃ VI: R¹ = CH₂—CH₃, Z = NHCH₃

TABLE 17

I: II: III: IV: V: VI: R¹ = CH₃, Z = CH₃ R¹ = CH₂—CH₃, Z = CH₃ R¹ = CH₃, Z = C₂H₅ R¹ = CH₂—CH₃, Z = C₂H₅ R¹ = CH₃, Z = NHCH₃ # R¹ = CH₂—CH₃, Z = NHCH₃ No. X_(m)  1 H  2 2-F  3 3-F  4 4-F  5 2,4-F₂  6 2,4,6-F₃  7 2,3,4,5,6-F₅  8 2,3-F₂  9 2-Cl  10 3-Cl  11 4-Cl  12 2,3-Cl₂  13 2,4-Cl₂  14 2,5-Cl₂  15 2,6-Cl₂  16 3,4-Cl₂  17 3,5-Cl₂  18 2,3,4-Cl₃  19 2,3,5-Cl₃  20 2,3,6-Cl₃  21 2,4,5-Cl₃  22 2,4,6-Cl₃  23 3,4,5-Cl₃  24 2,3,4,6-Cl₄  25 2,3,5,6-Cl₄  26 2,3,4,5,6-Cl₅  27 2-Br  28 3-Br  29 4-Br  30 2,4-Br₂  31 2,5-Br₂  32 2,6-Br₂  33 2,4,6-Br₃  34 2,3,4,5,6-Br₅  35 2-I  36 3-I  37 4-I  38 2,4-I₂  39 2-Cl, 3-F  40 2-Cl, 4-F  41 2-Cl, 5-F  42 2-Cl, 6-F  43 2-Cl, 3-Br  44 2-Cl, 4-Br  45 2-Cl, 5-Br  46 2-Cl, 6-Br  47 2-Br, 3-Cl  48 2-Br, 4-Cl  49 2-Br, 5-Cl  50 2-Br, 3-F  51 2-Br, 4-F  52 2-Br, 5-F  53 2-Br, 6-F  54 2-F, 3-Cl  55 2-F, 4-Cl  56 2-F, 5-Cl  57 3-Cl, 4-F  58 3-Cl, 5-F  59 3-Cl, 4-Br  60 3-Cl, 5-Br  61 3-F, 4-Cl  62 3-F, 4-Br  63 3-Br, 4-Cl  64 3-Br, 4-F  65 2,6-Cl₂, 4-Br  66 2-CH₃  67 3-CH₃  68 4-CH₃  69 2,3-(CH₃ ₂  70 2,4-(CH₃ ₂  71 2,5-(CH₃ ₂  72 2,6-(CH₃ ₂  73 3,4-(CH₃ ₂  74 3,5-(CH₃ ₂  75 2,3,5-(CH₃)₃  76 2,3,4-(CH₃)₃  77 2,3,6-(CH₃)₃  78 2,4,5-(CH₃)₃  79 2,4,6-(CH₃)₃  80 3,4,5-(CH₃)₃  81 2,3,4,6-(CH₃)₄  82 2,3,5,6-(CH₃)₄  83 2,3,4,5,6-(CH₃)₅  84 2-C₂H₅  85 3-C₂H₅  86 4-C₂H₅  87 2,4-(C₂H₅)₂  88 2,6-(C₂H₅)₂  89 3,5-(C₂H₅)₂  90 2,4,6-(C2H5)3  91 2-n-C₃H₇  92 3-n-C₃H₇  93 4-n-C₃H₇  94 2-i-C₃H₇  95 3-i-C₃H₇  96 4-i-C₃H₇  97 2,4-(i-C₃H₇)₂  98 2,6-(i-C₃H₇)₂  99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl,6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃ ₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H_(5, 4-Cl) 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O-C₂H₅ 164 4-O-C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-C-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O-CH₂C₆H₅ 178 3-O-CH₂C₆H₅ 179 4-O-CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃——CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NC-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇) 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═No-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃-C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃-C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C6H5 385 4-C6H5 386 2-(2′-F—C6H4) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C6H4) 399 3-(3′-Cl—C6H4) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH3O2C—C6H4) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF3—C6H4) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF3—C6H4) 476 4-(4′-CF3—C6H4) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 62i 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₂-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 18

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazo1yl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 257 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃, Z = CH₃ II: R¹ = CH₂—CH₃, Z = CH₃ III: R¹ = CH₃, Z = C₂H₅ IV: R¹ = CH₂—CH₃, Z = C₂H₅ V: R¹ = CH₃, Z = NHCH₃ VI: R¹ = CH₂—CH₃, Z = NHCH₃

TABLE 19

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃,)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—O 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—O 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄( 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃C₂C—C₆H₄) 527 3-O-(2′-CH₃C₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = CH₃, Z = CH₃ II: R¹ = CH₂—CH₃, Z = CH₃ III: R¹ = CH₃, Z = C₂H₅ IV: R¹ = CH₂—CH₃, Z = C₂H₅ V: R¹ = CH₃, Z = NHCH₃ VI: R¹ = CH₂—CH₃, Z = NHCH₃

TABLE 20

I: R¹ = CH₃, Z = CH₃ II: R¹ = CH₂—CH₃, Z = CH₃ III: R¹ = CH₃, Z = C₂H₅ IV: R¹ = CH₂—CH₃, Z = C₂H₅ V: R¹ = CH₃, Z = NHCH₃ VI: R¹ = CH₂—CH₃, Z = NHCH₃ No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃-N-Methylpyrazolyl-4 144 3-C₆H₅-N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl-C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(4′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-l,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-l,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-l,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-l,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-l,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl-C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3

TABLE 21 Selected physical data of some compounds No. Compound ¹H-NMR(ppm) m.p. 1

3,7(s, broad, 3H); 1,2(s, broad, 3H) 2

3,75(s, 3H); 1,2(t, 3H) 3

3,7(s, 3H); 1,2(t, 3H) 4

3,95(s, 3H); 3,7(s, 3H); 1,2(t, 3H) 5

3,6(s, 3H); 2,9(d, 3H) 6

123 7

118 8

3.7(s, 3H); 2.55 (s, very broad, 2H)

TABLE 56 Selected physical data of some compounds

¹H-NMR(ppm) or IR No. X_(m) mp (° C.) (cm⁻¹) 1 H 90 2 2-CH₃ 80 3 2,5-(CH₃)₂ 101  4 2-CH₃-4-C(CH₃)═N—OCH₃ 3.95(s, 3H); 3.65(s, 3H); 2.9(d, 3H) 5 2,5-(CH₃)₂-4-C(CH₃)═N— 3.65(s, 3H); 2.9(d, O-Allyl 3H)

TABLE 22

No. X Z A 1 H CH₃ —CH₂O— 2 H CH₃ —CH₂O—N═C(CH₃)— 3 H CH₃ —CH═CH— 4 H NH₂ —CH₂O— 5 H NH₂ —CH₂O—N═C(CH₃)— 6 H NH₂ —CH═CH— 7 H N(CH₃)₂ —CH₂O— 8 H N(CH₃)₂ —CH₂O—N═C(CH₃)— 9 H N(CH₃)₂ —CH═CH— 10 H CCl₃ —CH₂O— 11 H CCl₃ —CH₂O—N═C(CH₃)— 12 H CCl₃ —CH═CH— 13 H CF₃ —CH₂O— 14 H CF₃ —CH₂O—N═C(CH₃)— 15 H CF₃ —CH═CH— 16 CH₃ CH₃ —CH₂O— 17 CH₃ CH₃ —CH₂O—N═C(CH₃)— 18 CH₃ CH₃ —CH═CH— 19 CH₃ NH₂ —CH₂O— 20 CH₃ NH₂ —CH₂O—N═C(CH₃)— 21 CH₃ NH₂ —CH═CH— 22 CH₃ N(CH₃)₂ —CH₂O— 23 CH₃ N(CH₃)₂ —CH₂O—N═C(CH₃)— 24 CH₃ N(CH₃)₂ —CH═CH— 25 CH₃ CCl₃ —CH₂O— 26 CH₃ CCl₃ —CH₂O—N═C(CH₃)— 27 CH₃ CCl₃ —CH═CH— 28 CH₃ CF₃ —CH₂O— 29 CH₃ CF₃ —CH₂O—N═C(CH₃)— 30 CH₃ CF₃ —CH═CH— 31 Cl CH₃ —CH₂O— 32 Cl CH₃ —CH₂C—N—C(CH₃)— 33 Cl CH₃ —CH═CH— 34 Cl NH₂ —CH₂O— 35 Cl NH₂ —CH₂O—N═C(CH₃)— 36 Cl NH₂ —CH═CH— 37 Cl N(CH₃)₂ —CH₂O— 38 Cl N(CH₃)₂ —CH₂O—N═C(CH₃)— 39 Cl N(CH₃)₂ —CH═CH— 40 Cl CCl₃ —CH₂O— 41 Cl CCl₃ —CH₂O—N═C(CH₃)— 42 Cl CCl₃ —CH═CH— 43 Cl CF₃ —CH₂O— 44 Cl CF₃ —CH₂O—N═C(CH₃)— 45 Cl CF₃ —CH═CH—

TABLE 23

No. B 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluormethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-4-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimi- dazo[5,4-a]-pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl I: R¹ = CH₃, Z = CH₃ II: R¹ = CH₂—CH₃, Z = CH₃ III: R¹ = CH₃, Z = C₂H₅ IV: R¹ = CH₂—CH₃, Z = C₂H₅ V: R¹ = CH₃, Z = NHCH₃ VI: R¹ = CH₂—CH₃, Z = NHCH₃

Example 10 N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-o-methyl-hydroxylamine (Table 30, No. 1)

a) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-hydroxylamine

At 0 to 5° C., 7.0 g (70 mmol) of methyl chloroformate is added dropwise to 11.3 g (80 mmol) of N-2,6-dimethylphenyl-hydroxylamine (prepared analogously to Bamberger et 10 al., Ann. Chem. 316 (1901), 278) and 12.5 g (90 mmol) of K₂CO₃ in 30 ml of methylene chloride. The mixture is stirred for 30 mins at 0-5° C., the insoluble solid is filtered off and the filtrate is evaporated down under reduced pressure. The residure is purified by column chromatography with mixtures of cyclohexand and ethyl acetate. There is obtained 1.4 g (7.2 mmol=9%) of the title compound as a dark oil.

¹H-NMR (CDCl₃; δ in ppm): 8.85 (s, broad, 1H, OH); 7.1 (m, 3H, phenyl); 3.75 (s, 3H, OCH₃); 2.3 (s, 6H, 2xCH₃)

b) N-(2,6-Dimethylphenyl)-N-methoxycarbonyl-O-methylhydroxylamine (Table 7, No. 1)

A mixture of 1.4 g (7.2 mmol) of N-(2,6-dimethylphenyl)-N-methoxycarbonyl-hydroxylamine (Example 1a), 1.3 g (9 mmol) of K₂CO₃ and 10 g (8 mmol) of dimethyl sulfate in 10 ml of acetone is stirred overnight at room temperature. The reaction mixture is then diluted with CH₂Cl₂ and stirred with dilute NH₃ solution. The phases are then separated and the organic phase is extracted another twice with water. The organic phase is dried over MgSO₄ and evaporated down, and the residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 1.2 g (6 mmol=83%)) of the title compound as a colorless solid (mp=81° C.)

¹H-NMR (CDCl₃; δ in ppm): 7.1 (m, 3H, phenyl); 3.75 (s, broad, 6H, 2xOCH₃); 2.3 (s, 3H, CH₃)

The compounds listed in the following tables may be prepared similarly. Compound I, No. 1 from Table 24, No. 1 has for example the following formula:

TABLE 24

a I: R¹ = CH₃, X = CH₃ b II: R¹ = CH₂ − CH₃, X = CH₃ c III: R¹ = CH₃, X = Cl b IV: R¹ = CH₂ − CH₃, X = Cl No. T_(m)  1 H  2 2-F  3 3-F  4 4-F  5 2,4-F₂  6 2,4,6-F₃  7 2,3,4,5,6-F5  8 2,3-F₂  9 2-Cl  10 3-Cl  11 4-Cl  12 2,3-Cl₂  13 2,4-Cl₂  14 2,5-Cl₂  15 2,6-Cl₂  16 3,4-Cl₂  17 3,5-Cl₂  18 2,3,4-Cl₃  19 2,3,5-Cl₃  20 2,3,6-Cl₃  21 2,4,5-Cl₃  22 2,4,6-Cl₃  23 3,4,5-Cl₃  24 2,3,4,6-Cl₄  25 2,3,5,6-Cl₄  26 2,3,4,5,6-Cl₅  27 2-Br  28 3-Br  29 4-Br  30 2,4-Br₂  31 2,5-Br₂  32 2,6-Br₂  33 2,4,6-Br₃  34 2,3,4,5,6-Br₂  35 2-I  36 3-I  37 4-I  38 2,4-I₂  39 2-Cl, 3-F  40 2-Cl, 4-F  41 2-Cl, 5-F  42 2-Cl, 6-F  43 2-Cl, 3-Br  44 2-Cl, 4-Br  45 2-Cl, 5-Br  46 2-Cl, 6-Br  47 2-Br, 3-Cl  48 2-Br, 4-Cl  49 2-Br, 5-Cl  50 2-Br, 3-F  51 2-Br, 4-F  52 2-Br, 5-F  53 2-Br, 6-F  54 2-F, 3-Cl  55 2-F, 4-Cl  56 2-F, 5-Cl  57 3-Cl, 4-F  58 3-Cl, 5-F  59 3-Cl, 4-Br  60 3-Cl, 5-Br  61 3-F, 4-Cl  62 3-F, 4-Br  63 3-Br, 4-Cl  64 3-Br, 4-F  65 2,6-Cl₂, 4-Br  66 2-CH₃  67 3-CH₃  68 4-CH₃  69 2,3-(CH₃)₂  70 2,4-(CH₃)₂  71 2,5-(CH₃)₂  72 2,6-(CH₃)₂  73 3,4-(CH₃)₂  74 3,5-(CH₃)₂  75 2,3,5-(CH₃)₃  76 2,3,4-(CH₃)₃  77 2,3,6-(CH₃)₃  78 2,4,5-(CH₃)₃  79 2,4,6-(CH₃)₃  80 3,4,5-(CH₃)₃  81 2,3,4,6-(CH₃)₄  82 2,3,5,6-(CH₃)₄  83 2,3,4,5,6-(CH₃)₅  84 2-C₂H₅  85 3-C₂H₅  86 4-C₂H₅  87 2,4-(C₂H₅)₂  88 2,6-(C₂H₅)₂  89 3,5-(C₂H₅)₂  90 2,4,6-(C₂H₅)₃  91 2-n-C₃H₇  92 3-n-C₃H₇  93 4-n-C₃H₇  94 2-i-C₃H₇  95 3-i-C₃H₇  96 4-i-C₃H₇  97 2,4-(i-C₃H₇)₂  98 2,6-(i-C₃H₇)₂  99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-Cl₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH2—C₆H₅ 138 3-CH2—C₆H₅ 139 4-CH2—C₆H₅ 140 2-CH2—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-O—C₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-9-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C6H13 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-CH₃, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO2, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl2, 5-NO2 254 2,4-Cl2, 6-NO2 255 2,6-Cl2, 4-NO2 256 2,6-Br2, 4-NO2 257 2,6-I2, 4-NO2 258 2-CH3, 5-i-C3H7, 4-Cl 259 2-CO₂CH₃ 260 3-CO2CH3 261 4-CO2CH3 262 2-CO2(C2H5) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂-OCH₃ 275 3-CH₂-OCH₃ 276 4-CH₂-OCH₃ 277 2-CH_(2O)(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂C(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH3—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C-NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO-C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C2H5—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂-C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C6H5 476 4-O—C6H5 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-C-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH_(3—C) ₆H₄) 498 2-O-(3′-CH_(3—C) ₆H₄) 499 2-O-(4′-CH_(3—C) ₆H₄) 500 3-O-(2′-CH_(3—C) ₆H₄) 501 3-O-(3′-CH_(3—C) ₆H₄) 502 3-O-(4′-CH_(3—C) ₆H₄) 503 4-O-(2′-CH_(3—C) ₆H₄) 504 4-O-(3′-CH_(3—C) ₆H₄) 505 4-O-(4′-CH_(3—C) ₆H₄) 506 2-O-(2′-CH_(3—CO—C) ₆H₄) 507 2-O-(3′-CH_(3—CO—C) ₆H₄) 508 2-O-(4′-CH_(3—CO—C) ₆H₄) 509 3-O-(2′-CH_(3—CO—C) ₆H₄) 510 3-O-(3′-CH_(3—CO—C) ₆H₄) 511 3-O-(4′-CH_(3—CO—C) ₆H₄) 512 4-O-(2′-CH_(3—CO—C) ₆H₄) 513 4-O-(3′-CH_(3—CO—C) ₆H₄) 514 4-O-(4′-CH_(3—CO—C) ₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C6H4) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H5) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-b-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-b-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-6-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 25

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH_(3—C) ₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃, X = CH₃ II: R¹ = CH₂—CH₃, X = CH₃ III: R¹ = CH₃, X = Cl IV: R¹ = CH₂—CH₃, X = Cl

TABLE 26

I: R₁ = CH₃, X = CH₃ II: R₁ = CH₂—CH₃, X = CH₃ III: R₁ = CH₃, X = Cl IV: R₁ = CH₂—CH₃, X = Cl No. T_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C2H5)3 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₃C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH3 211 2-Cl, 5-CH3 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH3 226 3-Br, 4-CH3 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇₎ 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH²—C⁶H⁵)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroal- lyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C6H5 385 4-C6H5 386 2-(2′-F—C6H4) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C6H4) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH3O2C—C6H4) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF3—C6H4) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C6H5 476 4-O—C6H5 478 2-O-(2′-F—C6H4) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH3—CO—C6H4) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O2N—C6H4) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 27

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrr9ly1-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₂H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chioroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₅)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Cxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3 385 1-Naphthyl 386 2-Naphthyl I: R¹ = CH₃, X = CH₃ II: R¹ = CH₂—CH₃, X = CH₃, III: R¹ = CH₃, X = Cl IV: R¹ = CH₂—CH₃, X = Cl

TABLE 28

No. T_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C4H9)2, 4-CH3 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C6H11 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═No-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = CH₃, X = CH₃ II: R¹ = CH₂—CH₃, X = CH₃ III: R¹ = CH₃, X = Cl IV: R¹ = CH₂—CH₃, X = Cl

TABLE 29

I: R¹ = CH₃, X = CH₃ II: R¹ = CH₂—CH₃, X = CH₃ III: R¹ = CH₃, X = Cl IV: R¹ = CH₂—CH₃, X = Cl No. B  1 Pyrrolyl-3  2 N—CH₃-Pyrrolyl-3  3 N—C₆H₅-Pyrrolyl-3  4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3  5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3  6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3  7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3  8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3  9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3  10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3  11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3  12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3  13 N-(4′-CN—C₆H₄)-Pyrrolyl-3  14 N-(3′-CN—C₆H₄)-Pyrrolyl-3  15 N-(2′-CN—C₆H₄)-Pyrrolyl-3  16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3  17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3  18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3  19 Pyrrolyl-2  20 N—CH₃-Pyrrolyl-2  21 N—C₆H₅-Pyrrolyl-2  22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2  23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2  24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2  25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2  26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2  27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2  28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2  29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2  30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2  31 N-(4′-CN—C₆H₄)-Pyrrolyl-2  32 N-(3′-CN—C₆H₄)-Pyrrolyl-2  33 N-(2′-CN—C₆H₄)-Pyrrolyl-2  34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2  35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2  36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2  37 Furyl-2  38 5-CH₃-Furyl-2  39 5-C₆H₅-Furyl-2  40 5-(4′-CH₃—C₆H₄)-Furyl-2  41 5-(3′-CH₃—C₆H₄)-Furyl-2  42 5-(2′-CH₃—C₆H₄)-Furyl-2  43 5-(4′-CH₃O—C₆H₄)-Furyl-2  44 5-(3′-CH₃O—C₆H₄)-Furyl-2  45 5-(2′-CH₃O—C₆H₄)-Furyl-2  46 5-(4′-NO₂—C₆H₄)-Furyl-2  47 5-(3′-NO₂—C₆H₄)-Furyl-2  48 5-(2′-NO₂—C₆H₄)-Furyl-2  49 5-(4′-CN—C₆H₄)-Furyl-2  50 5-(3′-CN—C₆H₄)-Furyl-2  51 5-(2′-CN—C₆H₄)-Furyl-2  52 5-(4′-Cl—C₆H₄)-Furyl-2  53 5-(3′-Cl—C₆H₄)-Furyl-2  54 5-(2′-Cl—C₆H₄)-Furyl-2  55 4-CH₃-Furyl-2  56 4-C₆H₅-Furyl-2  57 4-(4′-CH₃—C₆H₄)-Furyl-2  58 4-(3′-CH₃—C₆H₄)-Furyl-2  59 4-(2′-CH₃—C₆H₄)-Furyl-2  60 4-(4′-CH₃O—C₆H₄)-Furyl-2  61 4-(3′-CH₃O—C₆H₄)-Furyl-2  62 4-(2′-CH₃O—C₆H₄)-Furyl-2  63 4-(4′-NO₂—C₆H₄)-Furyl-2  64 4-(3′-NO₂—C₆H₄)-Furyl-2  65 4-(2′-NO₂—C₆H₄)-Furyl-2  66 4-(4′-CN—C₆H₄)-Furyl-2  67 4-(3′-CN—C₆H₄)-Furyl-2  68 4-(2′-CN—C₆H₄)-Furyl-2  69 4-(4′-Cl—C₆H₄)-Furyl-2  70 4-(3′-Cl—C₆H₄)-Furyl-2  71 4-(2′-Cl—C₆H₄)-Furyl-2  72 Thienyl-2  73 5-CH₃-Thienyl-2  74 5-C₆H₅-Thienyl-2  75 5-(4′-CH₃—C₆H₄)-Thienyl-2  76 5-(3′-CH₃—C₆H₄)-Thienyl-2  77 5-(2′-CH₃—C₆H₄)-Thienyl-2  78 5-(4′-CH₃O—C₆H₄)-Thienyl-2  79 5-(3′-CH₃O—C₆H₄)-Thienyl-2  80 5-(2′-CH₃O—C₆H₄)-Thienyl-2  81 5-(4′-NO₂—C₆H₄)-Thienyl-2  82 5-(3′-NO₂—C₆H₄)-Thienyl-2  83 5-(2′-NO₂—C₆H₄)-Thienyl-2  84 5-(4′-CN—C₆H₄)-Thienyl-2  85 5-(3′-CN—C₆H₄)-Thienyl-2  86 5-(2′-CN—C₆H₄)-Thienyl-2  87 5-(4′-Cl—C₆H₄)-Thienyl-2  88 5-(3′-Cl—C₆H₄)-Thienyl-2  89 5-(2′-Cl—C₆H₄)-Thienyl-2  90 4-CH₃-Thienyl-2  91 4-C₆H₅-Thienyl-2  92 4-(4′-CH₃—C₆H₄)-Thienyl-2  93 4-(3′-CH₃—C₆H₄)-Thienyl-2  94 4-(2′-CH₃—C₆H₄)-Thienyl-2  95 4-(4′-CH₃O—C₆H₄)-Thienyl-2  96 4-(3′-CH₃O—C₆H₄)-Thienyl-2  97 4-(2′-CH₃O—C₆H₄)-Thienyl-2  98 4-(4′-NO₂—C₆H₄)-Thienyl-2  99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 2-CH₃-Oxazolyl-4 234 2-C₆H₅-Oxazolyl-4 235 2-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 2-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 2-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 2-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 2-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 2-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 2-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 2-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 2-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 2-(4′-CN—C₆H₄)-Oxazolyl-4 245 2-(3′-CN—C₆H₄)-Oxazolyl-4 246 2-(2′-CN—C₆H₄)-Oxazolyl-4 247 2-(4′-Cl—C₆H₄)-Oxazolyl-4 248 2-(3′-Cl—C₆H₄)-Oxazolyl-4 249 2-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5′ 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,2,3-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-,3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 Pyridinyl-3

TABLE 30 Selected physical data of some compounds IR(cm⁻¹) or No. Compound ¹H-NMR (ppm) m.p 1

81 2

60 3

3.85(s, broad, 3H); 3.7(s, broad, 3H) 4

3.85(s, broad, 3H); 3.75(s, broad, 3H) 5

3.75(2s, broad, each 3H) 6

91 7

3.8(s, 3H); 3.75(s, broad, 3H) 8

3.85(s, 3H); 3.8(s, broad, 3H)

TABLE 31

I: R¹ = CH₃, X = CH₃ II: R¹ = C₂H₅, X = CH₃ III: R¹ = CH₃, X = Cl IV: R¹ = C₂H₅, X = Cl No. B 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10  5-Chloro-1-methyl-2-benzimidazolyl 11  2-Benzoxazolyl 12  1-Methyl-5-trifluoromethylimidazo- [5,4-a]-pyridin-2-yl 13  5-Chloro-2-pyrimidinyl 14  4-Methyl-5-phenyl-2-thiazolin-2-yl 15  4-Methyl-5-phenyl-2-oxazolin-2-yl 16  7-Trifluoromethyl-4-quinolinyl

TABLE 57 Selected physical data of some compounds

mp ¹H-NMR (ppm) No. X T_(m) (° C.) or IR (cm⁻¹) 1 Cl 2-CH₃ 3.8(s, broad, 6H) 2 Cl 2,5-(CH₃)₂ 3.8(s, broad, 6H) 3 Cl 2-CH₃-4-C(CH₃)═N—OCH₃ 4.0(s, 3H); 3.8 (s, broad, EH) 4 Cl 2,5-(CH₃)₂-4-C(CH₃)═N—O- 3.8(s, broad, 6H) Allyl 5 CH₃ 2-CH₃-4-C(CH₃)═N—OCH₃ 4.0(s, 3H); 3.75 (s, broad, 6H) 6 CH₃ 2-CH₃ 3.75(s, broad, 6H) 7 CH₃ 2,5-(CH₃)₂ 3.75(s, broad, 6H) 8 CH₃ 2,5-(CH₃)₂-4-C(CH₃)═N—O- 3.75(s, broad, Allyl 6H)

Example 11 2-(2′-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

a) 2-(2′-Methylphenoxymethyl)-nitrobenzene

75 g (0.347 mol) of 2-nitrobenzyl bromide, 37 g (0.342 mol) of o-cresol and 56 g (0.405 mol) of potassium carbonate in 500 ml of dimethylformamide is stirred for 5 hours at room temperature (20° C.). The reaction mixture is diluted with water and the aqueous phase is extracted three times with ether. The ether phase is dried and evaporated down. The crystalline residue is stirred with methanol and suction filtered. There is obtained 73 g (0.300 mol=88%) of the title compound as a colorless solid.

Mp=83° C.

¹H-NMR, (CDCl₃; δ (ppm)): 8.15 (d, 1H, I=8 Hz, aromatic); 7.95 (d, 1H, I=8 Hz, aromatic); 7.7 (t, 1H, I=8 Hz, aromatic); 7.45 (t, 1H, I=8 Hz, aromatic); 7.15 (m, 2H, aromatic); 6.9 (m, 2H, aromatic); 5.45 (s, 2H, O—CH₂); 2.35 (s, 3H, CH₃)

b) 2-(2′-Methylphenoxymethyl)-aniline

75 g (0.308 mol) of 2-(2′-methylphenoxymethyl)-nitrobenzene (Example 11a) and 10 g of 5% Pt/C (platinum adsorbed on activated carbon) in 50 ml of methanol are stirred vigorously under a hydrogen blanket for 2 hours. A further 2 g of 5% Pt/C is added and the mixture is stirred overnight. The catalyst is filtered off and replaced by 10 g of fresh catalyst. The mixture is stirred overnight and suction filtered, and the filtrate is evaporated down under reduced pressure. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 61 g (0.286 mol=93%) of the title compound as a colorless solid.

Mp=56° C.

¹H-NMR (CDCl₃; δ (ppm)): 7.2 (m, 4H, aromatic); 6.95 (d, 1H, I=8 Hz, aromatic); 6.9 (t, 1H, I=6 Hz, aromatic); 6.7 (m, 2H, aromatic); 5.0 (S, 2H, O—CH₂); 4.05 (s, broad, 2H, NH₂); 2.2 (s, 3H, CH₃)

c) 2-(2′-Methylphenoxymethyl)-trichloroacetanilide (Table 38, No. 1)

At 10-15° C., a solution of 6 g of 2-(2′-methylphenoxymethyl)-aniline (Example 1b) in 20 ml of CH₂Cl₂ is added to a mixture of 6.6 g (36 mmol) of trichloroacetyl chloride and 3 g (38 mmol) of pyridine in 50 ml of CH₂Cl₂. The mixture is stirred for 1 hour at room temperature, and then extracted with water, dried over MgSO₄ and evaporated down. The residue is suction filtered over silica gel and the filtrate which is obtained is evaporated down. The residue crystallizes and is stirred with hexane. There is obtained 7.9 g (22 mmol=78%) of the title compound as a crystalline solid (mp=128° C.).

¹H-NMR (CDCl₃; δ (ppm)): 9.6 (s, broad, 1H, NH); 8.1 (d, 1H, I=8 Hz, phenyl); 7.5 (t, broad, 1H, phenyl); 7.4 (d, broad, 1H, phenyl); 7.2 (m, 3H, phenyl); 6.95 (m, 2H, phenyl); 5.1 (s, 2H, OCH₂); 2.2 (s, 3H, CH₃)

Example 12 N-Methyl-N′-(2-(2′-methylphenoxymethyl)-phenyl)-urea (Table 7, No. 2)

In a laboratory autoclave, about 10 ml of methylamine is added to 2 g (5.5 mmol) of the trichloroacetanilide from Example 1c. The autoclave is then closed and the reaction mixture is heated for about 6 hours at 80° C. The reaction mixture is cooled and the autoclave opened. The methylamine is allowed to evaporate off and the solid residue is stirred with methyl tert-butyl ether. The insoluble solid is filtered off and dried under reduced pressure. There is obtained 1.4 g (5.2 mmol=94%) of the title compound as a crystalline solid (mp=144° C.).

¹H-NMR (DMSO-d₆; δ (ppm)): 8.05 (s, 1H, NH); 7.8 (d, 1H, I=8 Hz, phenyl); 7.4 (d, 1H, I=8 Hz, phenyl); 6.8-7.3 (m, 6H, phenyl); 6.7 (s, 1H, NH); 5.1 (s, 2H, OCH₂); 2.65 (d, 3H, I=5 Hz, N—CH₃); 2.2 (s, 3H, CH₃)

Example 13 2-(2′-Methylphenoxymethyl)-propionyl anilide (Table 38, No. 3)

A mixture of 3 g (14.1 mmol) of the aniline from Example 11b, 1.35 g (17 mmol) of pyridine and 1.4 g (15.5 mmol) of propionyl chloride in 30 ml of methylene chloride is stirred for 1 hour at room temperature. The reaction mixture is then extracted with diluted hydrochloric acid and water, dried over MgSO₄ and evaporated down. There is obtained 3.8 g (quantitative yield) of the title compound.

¹H-NMR (COCl₃; δ (ppm)): 8.25 (s, broad, 1H, NH); 8.15 (d, 1H, I=8 Hz, phenyl); 6.9-7.5 (m, 7H, phenyl); 5.1 (s, 2H, OCH₂); 2.35 (q, 2H, I=8 Hz, CH₂); 2.25 (s, 3H, CH₃); 1.2 (t, 3H, I=8 Hz, CH₃)

Example 14 N-Propionyl-2-(2′-methylphenoxymethyl)-propionyl anilide (Table 38, No. 4)

0.41 g (17.1 mmol) of sodium hydride is added in portions to 3.8 g (14 mmol) of the propionyl anilide from Example 13 in 40 ml of dimethylformamide. Upon completion of gas evolution 1.4 g (15.9 mmol) of propionyl chloride is added and the mixture is stirred overnight at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2.6 g (8 mmol=57%) of the title compound as a yellow oil.

¹H-NMR (CDCl₃): δ (ppm): 7.6 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.15 (m, 3H, phenyl); 6.85 (m, 2H, phenyl); 4.85 (m, 2H, OCH₂); 2.6 (m, 4H, 2xCH₂); 2.2 (s, 3H, CH₃); 1.1 (t, 6H, I=8 Hz, 2xCH₃)

Example 15 N-Methyl-2-(2′-methylphenoxymethyl)-propionyl anilide (Table 38, No. 5)

0.45 g (19 mmol) of sodium hydride is added in portions to 4.0 g (14.8 mmol) of the propionyl anilide from Example 13 in 50 ml of dimethylformamide. Upon completion of gas evolution 3.0 g (21 mmol) of methyl iodide is added and the mixture is stirred for 2 hours at room temperature. The reaction mixture is then diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The residue crystallizes is stirred with hexane. There is obtained 3.7 g (11.7 mmol=90%) of the title compound as a colorless solid (mp=80° C.).

¹H-NMR (CDCl₃; δ (ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.2 (s, 3H, N—CH₃); 2.2 (s, 3H, CH₃); 2.0 (m, 2H, CH₂); 1.0 (t, 3H, I=8 Hz, CH₃)

Example 19 N-Methyl-2-(2′-methylphenoxymethyl)-acetanilide

a) N-Methyl-2-(2′-methylphenoxymethyl)-aniline

A mixture of 5 g (23 mmol) of 2-(2′-methylphenoxymethyl)-aniline (Example 1b), 5 g (36 mmol) of K₂CO₃ and 3.4 g (24 mmol) of methyl iodide in 50 ml of dimethylformamide is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. The reside is purified chromatographically using mixtures of hexane and methylene chloride. There is obtained 3.0 g (70% purity, about 40% yield) of the title compound as a yellow oil.

¹H-NMR (CDCl₃; δ in ppm): 6.6-7.4 (m, 8H, phenyl); 5.0 (s, 2H, OCH₂); 4.6 (s, broad, 1H, NH); 2.9 (d, 3H, N—CH₃); 2.2 (s, 3H, CH₃).

b) N-Methyl-2-(2′-methylphenoxymethyl)-acetanilide (Table 7, No. 9)

3 g (approx. 9.3 mmol) of N-methyl-2-(2′-methylphenoxymethyl)-aniline (from Example 5a is added to a mixture of 1.6 g (16 mmol) of acetoanhydride and 1.3 g (16 mmol) of pyridine in 20 ml of methylene chloride. The mixture is stirred for 1 hour at room temperature and is then extracted with dilute hydrochloric acid and water. The organic phase is evaporated down and the residue is purified by column chromatography with mixtures of hexane and ethyl acetate. There is obtained 2 g (80%) of the title compound as a colorless solid (mp=76° C.).

¹H-NMR (CDCl₃; δ in ppm): 7.7 (m, 1H, phenyl); 7.4 (m, 2H, phenyl); 7.2 (m, 3H, phenyl); 6.9 (m, 2H, phenyl); 5.0 (s, 2H, OCH₂); 3.25 (s, 3H, CH₃); 2.25 (s, 3H, CH₃); 1.8 (s, 3H, CH₃).

The compounds listed in the tables below may be prepared correspondingly.

Compound I from Table 32, No. 1 has for example the following structural formula:

The compounds described in the following tables may be prepared analogously.

TABLE 32

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CO—CH₃ 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CO—CH₂—CH₂—CH₃ 305 2-Me-4-CO—CH(CH₃)₂ 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CO—CH₃ 308 2,5-Me₂-4-CO—CH₂—CH₃ 309 2,5-Me₂-4-CH₂—CH₂—CO—CH₃ 310 2,5-Me₂-4-CO—CH(CH₃)₂ 311 2-Cl-4-CHO 312 2-Cl-4-CO—CH₃ 313 2-Cl-4-CO—CH₂—CH₃ 314 2-Cl-4-CO—CH(CH₃)₂ 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CO—CH₃ 317 2,5-Cl₂-4-CO—CH₂—CH₃ 318 2,5-Cl₂-4-CO—CH₂—CH₂—CH₃ 319 2,5-Cl₂-4-CO—CH(CH₃)₂ 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇) 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazoly1-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 33

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CO—CH₃ 303 2-Me-4-CO—CH₂—CH₃ 304 2-Me-4-CO—CH₂—CH₂—CH₃ 305 2-Me-4-CO—CH(CH₃)₂ 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CO—CH₃ 308 2,5-Me₂-4-CO—CH₂—CH₃ 309 2,5-Me₂-4-CH₂—CH₂—CO—CH₃ 310 2,5-Me₂-4-CO—CH(CH₃)₂ 311 2-Cl-4-CHO 312 2-Cl-4-CO—CH₃ 313 2-Cl-4-CO—CH₂—CH₃ 314 2-Cl-4-CO—CH(CH₃)₂ 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CO—CH₃ 317 2,5-Cl₂-4-CO—CH₂—CH₃ 318 2,5-Cl₂-4-CO—CH₂—CH₂—CH₃ 319 2,5-Cl₂-4-CO—CH(CH₃)₂ 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇) 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazoly1-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chlorallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chlorallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 34

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CO—CH₃ 303 2-Me-4-CO—CH₂—CH₃ 304 2-Me-4-CO—CH₂—CH₂—CH₃ 305 2-Me-4-CO—CH(CH₃)₂ 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CO—CH₃ 308 2,5-Me₂-4-CO—CH₂—CH₃ 309 2,5-Me₂-4-CH₂—CH₂—CO—CH₃ 310 2,5-Me₂-4-CO—CH(CH₃)₂ 311 2-Cl-4-CHO 312 2-Cl-4-CO—CH₃ 313 2-Cl-4-CO—CH₂—CH₃ 314 2-Cl-4-CO—CH(CH₃)₂ 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CO—CH₃ 317 2,5-Cl₂-4-CO—CH₂—CH₃ 318 2,5-Cl₂-4-CO—CH₂—CH₂—CH₃ 319 2,5-Cl₂-4-CO—CH(CH₃)₂ 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇) 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazoly1-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 35

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃CO 303 2-Me-4-CO—CH₂—CH₃ 304 2-Me-4-CO—CH₂—CH₂—CH₃ 305 2-Me-4-CO—CH(CH₃)₂ 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CO—CH₃ 308 2,5-Me₂-4-CO—CH₂—CH₃ 309 2,5-Me₂-4-CH₂—CH₂—CO—CH₃ 310 2,5-Me₂-4-CO—CH(CH₃)₂ 311 2-Cl-4-CHO 312 2-Cl-4-CO—CH₃ 313 2-Cl-4-CO—CH₂—CH₃ 314 2-Cl-4-CO—CH(CH₃)₂ 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CO—CH₃ 317 2,5-Cl₂-4-CO—CH₂—CH₃ 318 2,5-Cl₂-4-CO—CH₂—CH₂—CH₃ 319 2,5-Cl₂-4-CO—CH(CH₃)₂ 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇) 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazoly1-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N—O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 36

No. X_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 267 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CO—CH₂—CH₃ 304 2-Me-4-CO—CH₂—CH₂—CH₃ 305 2-Me-4-CO—CH(CH₃)₂ 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CO—CH₃ 308 2,5-Me₂-4-CO—CH₂—CH₃ 309 2,5-Me₂-4-CH₂—CH₂—CO—CH₃ 310 2,5-Me₂-4-CO—CH(CH₃)₂ 311 2-Cl-4-CHO 312 2-Cl-4-CO—CH₃ 313 2-Cl-4-CO—CH₂—CH₃ 314 2-Cl-4-CO—CH(CH₃)₂ 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CO—CH₃ 317 2,5-Cl₂-4-CO—CH₂—CH₃ 318 2,5-Cl₂-4-CO—CH₂—CH₂—CH₃ 319 2,5-Cl₂-4-CO—CH(CH₃)₂ 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chlorallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Propargyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄ 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 37

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N—(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N—(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N—(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N—(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N—(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N—(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N—(4′-CN—C₆H₄)-Pyrrolyl-3 14 N—(3′-CN—C₆H₄)-Pyrrolyl-3 15 N—(2′-CN—C₆H₄)-Pyrrolyl-3 16 N—(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N—(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N—(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N—(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N—(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N—(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N—(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N—(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N—(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N—(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N—(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N—(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N—(4′-CN—C₆H₄)-Pyrrolyl-2 32 N—(3′-CN—C₆H₄)-Pyrrolyl-2 33 N—(2′-CN—C₆H₄)-Pyrrolyl-2 34 N—(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N—(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N—(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N—(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N—(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N—(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N—(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N—(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N—(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N—(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N—(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N—(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N—(4′-CN—C₆H₄)-Pyrazolyl-4 138 N—(3′-CN—C₆H₄)-Pyrazolyl-4 139 N—(2′-CN—C₆H₄)-Pyrazolyl-4 140 N—(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N—(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N—(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH₃-Oxazolyl-4 234 3-C₆H₅-Oxazolyl-4 235 3-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 3-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 3-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 3-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 3-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 3-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 3-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 3-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 3-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 3-(4′-CN—C₆H₄)-Oxazolyl-4 245 3-(3′-CN—C₆H₄)-Oxazolyl-4 246 3-(2′-CN—C₆H₄)-Oxazolyl-4 247 3-(4′-Cl—C₆H₄)-Oxazolyl-4 248 3-(3′-Cl—C₆H₄)-Oxazolyl-4 249 3-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ = Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ VII: R¹ = CO—C₂H₅, Z = C₂H₅ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ = CH₂—OCH₃, Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃)

TABLE 38 Selected physical data of some compounds IR (cm⁻¹) or ¹H-NMR mp No. Compound (ppm) (° C.) 1

128 2

144 3

4

5

80 6

75 7

188 8

115 9

76 10

96 11

3.3 (s, 3H); 2.25 (s, 3H)

TABLE 58 Selected physical data of some compounds

IR (cm⁻¹) or No. X_(m) R¹ ¹H-NMR (ppm) mp (° C.) 1 2-CH₃ H 120 2 2-CH₃ CH₃ oil 3 2-CH₃ C₂H₅ oil 4 2-CH₃ Allyl oil 5 2-CH₃ Propargyl oil 6 2-CH₃ CH₂—OCH₃ oil 7 2,5-(CH₃)₂ H 170 8 2,5-(CH₃)₂ CH₃ oil 9 2,5-(CH₃)₂ C₂H₅ oil 10 2,5-(CH₃)₂ Allyl oil 11 2,5-(CH₃)₂ Propargyl oil 12 2,5-(CH₃)₂ CH₂—OCH₃ oil 13 2-CH₃-4-C(CH₃)═N—OCH₃ H 125 14 2-CH₃-4-C(CH₃)═N—OCH₃ CH₃ oil 15 2-CH₃-4-C(CH₃)═N—OCH₃ C₂H₅ oil 16 2-CH₃-4-C(CH₃)═N—OCH₃ Allyl  87 17 2-CH₃-4-C(CH₃)═N—OCH₃ Propargyl oil 18 2-CH₃-4-C(CH₃)═N—OCH₃ CH₂—OCH₃ oil 19 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl H  85 20 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl CH₃ oil 21 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl C₂H₅ oil 22 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl Allyl  87 23 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl Propargyl oil 24 2,5-(CH₃)₂-4-C(CH₃)═N—O-Allyl CH₂—OCH₃ oil

TABLE 59 Selected physical data of some compounds

IR (cm⁻¹) or ¹H-NMR No. X_(m) R¹ (ppm) mp (° C.) 1 4-CH₃ H 118 2 4-CH₃ CH₃ oil 3 4-CH₃ C₂H₅ oil 4 4-CH₃ Allyl oil 5 4-CH₃ Propargyl oil 6 4-CH₃ CH₂—OCH₃ oil 7 3,5-Cl₂ H 160 8 3,5-Cl₂ CH₃ oil 9 3,5-Cl₂ C₂H₅ oil 10 3,5-Cl₂ Allyl  85 11 3,5-Cl₂ Propargyl oil 12 3,5-Cl₂ CH₂—OCH₃ oil

TABLE 39

No. X R¹ Z A 1 H H CH₃ —CH₂O— 2 H H CH₃ —CH₂O—N═C(CH₃)— 3 H H CH₃ —CH═CH— 4 H H NH₂ —CH₂O— 5 H H NH₂ —CH₂O—N═C(CH₃)— 6 H H NH₂ —CH═CH— 7 H H N(CH₃)₂ —CH₂O— 8 H H N(CH₃)₂ —CH₂O—N═C(CH₃)— 9 H H N(CH₃)₂ —CH═CH— 10 H H CCl₃ —CH₂O— 11 H H CCl₃ —CH₂O—N═C(CH₃)— 12 H H CCl₃ —CH═CH— 13 H H CF₃ —CH₂O— 14 H H CF₃ —CH₂O—N═C(CH₃)— 15 H H CF₃ —CH═CH— 16 H Propargyl CH₃ —CH₂O— 17 H Propargyl CH₃ —CH₂O—N═C(CH₃)— 18 H Propargyl CH₃ —CH═CH— 19 H Propargyl NH₂ —CH₂O— 20 H Propargyl NH₂ —CH₂O—N═C(CH₃)— 21 H Propargyl NH₂ —CH═CH— 22 H Propargyl N(CH₃)₂ —CH₂O— 23 H Propargyl N(CH₃)₂ —CH₂O—N—═C(CH₃)— 24 H Propargyl N(CH₃)₂ —CH═CH— 25 H Propargyl CCl₃ —CH₂O— 26 H Propargyl CCl₃ —CH₂O—N═C(CH₃)— 27 H Propargyl CCl₃ —CH═CH— 28 H Propargyl CF₃ —CH₂O— 29 H Propargyl CF₃ —CH₂O—N═C(CH₃)— 30 H Propargyl CF₃ —CH═CH— 31 CH₃ H CH₃ —CH₂O— 32 CH₃ H CH₃ —CH₂O—N═C(CH₃)— 33 CH₃ H CH₃ —CH═CH— 34 CH₃ H NH₂ —CH₂O— 35 CH₃ H NH₂ —CH₂O—N═C(CH₃)— 36 CH₃ H NH₂ —CH═CH— 37 CH₃ H N(CH₃)₂ —CH₂O— 38 CH₃ H N(CH₃)₂ —CH₂O—N═C(CH₃)— 39 CH₃ H N(CH₃)₂ —CH═CH— 40 CH₃ H CCl₃ —CH₂O— 41 CH₃ H CCl₃ —CH₂O—N═C(CH₃)— 42 CH₃ H CCl₃ —CH═CH— 43 CH₃ H CF₃ —CH₂O— 44 CH₃ H CF₃ —CH₂O—N═C(CH₃)— 45 CH₃ H CF₃ —CH═CH— 46 CH₃ Propargyl CH₃ —CH₂O— 47 CH₃ Propargyl CH₃ —CH₂O—N═C(CH₃)— 48 CH₃ Propargyl CH₃ —CH═CH— 49 CH₃ Propargyl NH₂ —CH₂O— 50 CH₃ Propargyl NH₂ —CH₂O—N═C(CH₃)— 51 CH₃ Propargyl NH₂ —CH═CH— 52 CH₃ Propargyl N(CH₃)₂ —CH₂O— 53 CH₃ Propargyl N(CH₃)₂ —CH₂O—N═C(CH₃)— 54 CH₃ Propargyl N(CH₃)₂ —CH═CH— 55 CH₃ Propargyl CCl₃ —CH₂O— 56 CH₃ Propargyl CCl₃ —CH₂O—N═C(CH₃)— 57 CH₃ Propargyl CCl₃ —CH═CH— 58 CH₃ Propargyl CF₃ —CH₂O— 59 CH₃ Propargyl CF₃ —CH₂O—N═C(CH₃)— 60 CH₃ Propargyl CF₃ —CH═CH— 61 Cl H CH₃ —CH₂O— 62 Cl H CH₃ —CH₂O—N═C(CH₃)— 63 Cl H CH₃ —CH═CH— 64 Cl H NH₂ —CH₂O— 65 Cl H NH₂ —CH₂O—N═C(CH₃)— 66 Cl H NH₂ —CH═CH— 67 Cl H N(CH₃)₂ —CH₂O— 68 Cl H N(CH₃)₂ —CH₂O—N═C(CH₃)— 69 Cl H N(CH₃)₂ —CH═CH— 70 Cl H CCl₃ —CH₂O— 71 Cl H CCl₃ —CH₂O—N═C(CH₃)— 72 Cl H CCl₃ —CH═CH— 73 Cl H CF₃ —CH₂O— 74 Cl H CF₃ —CH₂O—N═C(CH₃)— 75 Cl H CF₃ —CH═CH— 76 Cl Propargyl CH₃ —CH₂O— 77 Cl Propargyl CH₃ —CH₂O—N═C(CH₃)— 78 Cl Propargyl CH₃ —CH═CH— 79 Cl Propargyl NH₂ —CH₂O— 80 Cl Propargyl NH₂ —CH₂O—N═C(CH₃)— 81 Cl Propargyl NH₂ —CH═CH— 82 Cl Propargyl N(CH₃)₂ —CH₂O— 83 Cl Propargyl N(CH₃)₂ —CH₂O—N═C(CH₃)— 84 Cl Propargyl N(CH₃)₂ —CH═CH— 85 Cl Propargyl CCl₃ —CH₂O— 86 Cl Propargyl CCl₃ —CH₂O—N═C(CH₃)— 87 Cl Propargyl CCl₃ —CH═CH— 88 Cl Propargyl CF₃ —CH₂O— 89 Cl Propargyl CF₃ —CH₂O—N═C(CH₃)— 90 Cl Propargyl CF₃ —CH═CH—

TABLE 40

I: R¹ = H, Z = C₂H₅ II: R¹ = CH₃, Z = C₂H₅ III: R¹ = C₂H₅, Z = C₂H₅ IV: R¹ Allyl, Z = C₂H₅ V: R¹ = Propargyl, Z = C₂H₅ VI: R¹ = CH₂—OCH₃, Z = C₂H₅ # VII: R¹ = CO—C₂ VIII: R¹ = H, Z = NH(CH₃) IX: R¹ = CH₃, Z = NH(CH₃) X: R¹ = C₂H₅, Z = NH(CH₃) XI: R¹ = Allyl, Z = NH(CH₃) XII: R¹ = Propargyl, Z = NH(CH₃) XIII: R¹ =CH₂—OCH₃, # Z = NH(CH₃) XIV: R¹ = CO—C₂H₅, Z = NH(CH₃) NO. B  1 2-Pyridyl  2 3-Trifluoromethyl-2-pyridyl  3 5-Trifluoromethyl-2-pyridyl  4 3,5-Bis-(trifluoromethyl)-2-pyridyl  5 3,5-Dichloro-2-pyridyl  6 3-Chloroo-5-trifluoromethyl-2-pyridyl  7 3,5-Dichloro-2-pyridyl  8 2-Chloroo-4-trifluoromethylphenyl  9 2-Benzothiazolyl 10 5-Chloroo-I-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimidazo- [5,4-a]-pyridin-2-yl 13 5-Chloroo-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl

Example 16 Methyl N-[2-(3″,4″-dichlorophenyl-1′-methyliminooxymethyl-4′)-6-methylphenyl]-carbamate (Table 47, No. 2)

a) 2-(Methanesulfonyloxymethyl)-6-methyl-nitrobenzene

At 10-15° C., 27 g (0.23 mol) of methanesulfonyl chloride dissolved in 20 ml of CH₂Cl₂ is dripped into a mixture of 34 g (0.2 mol) of 3-methyl-2-nitrobenzyl alcohol and 27 g (0.27 mol) of triethylamine in 100 ml of CH₂Cl₂. The reaction mixture is stirred for 1 hour at room temperature and is then extracted with water. The organic phase is dried over MgSO₄ and evaporated down. There is obtained as residue 48 g of the title compound as a yellow oil, containing about 10% of the corresponding benzyl chloride as impurity. The crude product is used for the next reaction without any further purification.

¹H-NMR(COCl₃; δ in ppm): 7.3-7.6 (m, 3H, phenyl); 5.3 (S, 2H, OCH₂); 3.0 (S, 3H, CH₃—SO₃); 2.4 (S, 3H, CH₃)

b) 2-(3″,4″-Dichlorophenyl-1′-methyl-iminooxymethyl-4′)-6-methyl-nitrobenzene

At room temperature, 1.8 g (75 mmol) of sodium hydride is added in portions to a solution of 13 g (64 mmol) of 3,4-dichloroacetophenonoxime in 100 ml of dimethylformamide. Upon conclusion of gas evolution, a solution of 16 g (65 mmol) of the mesylate from Example 1a in 30 ml of dimethylformamide is dripped in at 25-30° C., and the mixture is then stirred for 1 hour at room temperature. The reaction mixture is diluted with water and the aqueous phase is then extracted three times with methyl tert-butyl ether. The combined organic phases are washed with water, dried over MGSO₄ and evaporated down. The residue crystallizes and is stirred with methanol. The mother liquor is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained a total of 20.4 g (58 mmol=90%) of the title compound as pale yellow crystals.

¹H-NMR(CDCl₃; δ in ppm): 7.7 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.3 (S, 2H, OCH₂); 2.4 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

c) 2-(3″,4″-Dichlorophenyl-1′-methyl-iminooxymethyl-4′)-6-methyl-aniline

At 20-30° C., 53 g of 21.8% strength Na₂[Fe(CO)₄] solution (1 kg of the solution contains 633 g of water, 218 g of Na₂[Fe(CO)₄], 108 g of Na₂CO₃ and 41 g of NaOH) is added dropwise to 19 g (52.8 mmol) of the nitrobenzene from Example 16b in 150 ml of methanol. The brown suspension is stirred for 2 hours at room temperature, and the reaction mixture is then diluted with methylene chloride and the mixture is suction filtered using kieselguhr. The residue is again washed with CH₂Cl₂ and the combined extracts are extracted with water, dried over MgSO₄ and evaporated down. The brown residue is purified by column chromatography with mixtures of cyclohexane and ethyl acetate. There is obtained 14.3 g (44.3 mmol=82%) of the title compound as a beige solid.

¹H-NMR(CDCl₃; δ in ppm): 7.7 (S, 1H, phenyl); 7.5 (m, 2H, phenyl); 7.1 (t, broad, 2H, phenyl); 6.7 (t, 1H, I=8 Hz, phenyl); 5.2 (S, 2H, OCH₂); 4.15 (S, 2H, NH₂; 2.2 (S, 3H, CH₃)

d) Methyl N-[2-(3″,4″-dichlorophenyl-1′-methyl-iminooxymethyl-4′-6-methylphenyl]-carbamate (Table 47, No. 2)

At 20-30° C., 4.8 g (50 mmol) of methyl chloroformate a subsequently 4.8 g (60 mmol) of pyridine are dripped into a solution of 14.3 g (44 mmol) of the aniline from Example 1c in 150 ml of CH₂Cl₂. The mixture is stirred overnight at room temperature and is then extracted with dilute hydrochloric acid and water. The reaction mixture is suction filtered using silica gel, dried over MgSO₄ and evaporated down. The residue crystallizes and is stirred with cyclohexane. There is obtained 13.8 g (36 mmol=82%) of the title compound as a colorless solid (mp=109° C.).

¹H-NMR(CDCl₃; δ in ppm): 7.8 (S, 1H, phenyl); 7.6 (S, broad, 1H, NH); 7.4 (S, 2H, phenyl); 7.2 (m, 3H, phenyl); 5.2 (S, 2H, OCH₂); 3.8 (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.2 (S, 3H, CH₃)

Example 17 Methyl N-[2-(3″,4″-dichlorophenyl-1′-methyl-iminooxymethyl-4′)-6-methylphenyl]-N-propargyl-carbamate (Table 47, No. 13)

At 25-30° C., 0.15 g (6.3 mmol) of sodium hydride is added in portions to a solution of 1.9 g (5 mmol) of the carbamate from Example 16d in 20 ml of dimethylformamide. When no more gas evolves, 0.75 g (6.3 mmol) of propargyl bromide is added and the whole is stirred overnight at room temperature. The reaction mixture is diluted with water and the aqueous phase is extracted three times with methyl tert-butyl ether. The combined organic phases are extracted with water, dried over MgSO₄ and evaporated down. There is obtained 1.4 g (3.3 mmol=67%) of the title compound as a yellow oil.

¹H-NMR (CDCl₃; δ in ppm): 7.75 (S, broad, 1H, phenyl); 7.2-7.6 (m, 5H, phenyl); 5.2 (dd, 2H, I=12 Hz, OCH₂); 4.4 (dd, broad, I=16 Hz, NCH₂); (S, 3H, OCH₃); 2.3 (S, 3H, CH₃); 2.25 (S, broad, 1H, C≡CH); 2.2 (S, 3H, CH₃); the ¹H-NMR spectrum also contains signals of about 20% of the amide rotamer.

The compounds described in the following tables may be prepared analogously.

TABLE 41

I: II: III: IV: V: VI: VII: VIII: IX: X: XI: XII: XIII: XIV: R¹ = H, X = CH³ R¹ = CH₃, X = CH₃ R¹ = C₂H₅, X = CH₃ R¹ = Allyl, X = CH₃ # R¹ = Propargyl, X =CH₃ R¹ = CH₂—OCH₃, X = CH₃ R¹ = CO₂CH₃, X = CH₃ R¹ = H, X = Cl R¹ = CH₃, X = Cl R¹ = C₂H₅, X = Cl R¹ = Allyl, X = Cl R¹ = Propargyl, X = Cl # R¹ = CH₂—OCH₃, X = Cl R¹ = CO₂CH₃, X = Cl

Compound I from Table 41 has for instance the following structural formula:

NO. T_(m)  1 H  2 2-F  3 3-F  4 4-F  5 2,4-F₂  6 2,4,6-F₃  7 2,3,4,5,6-F₅  8 2,3-F₂  9 2-Cl  10 3-Cl  11 4-Cl  12 2,3-Cl₂  13 2,4-Cl₂  14 2,5-Cl₂  15 2,6-Cl₂  16 3,4-Cl₂  17 3,5-Cl₂  18 2,3,4-Cl₃  19 2,3,5-Cl₃  20 2,3,6-Cl₃  21 2,4,5-Cl₃  22 2,4,6-Cl₃  23 3,4,5-Cl₃  24 2,3,4,6-Cl₄  25 2,3,5,6-Cl₄  26 2,3,4,5,6-Cl₅  27 2-Br  28 3-Br  29 4-Br  30 2,4-Br₂  31 2,5-Br₂  32 2,6-Br₂  33 2,4,6-Br₃  34 2,3,4,5,6-Br₅  35 2-I  36 3-I  37 4-I  38 2,4-I₂  39 2-Cl, 3-F  40 2-Cl, 4-F  41 2-Cl, 5-F  42 2-Cl, 6-F  43 2-Cl, 3-Br  44 2-Cl, 4-Br  45 2-Cl, 5-Br  46 2-Cl, 6-Br  47 2-Br, 3-Cl  48 2-Br, 4-Cl  49 2-Br, 5-Cl  50 2-Br, 3-F  51 2-Br, 4-F  52 2-Br, 5-F  53 2-Br, 6-F  54 2-F, 3-Cl  55 2-F, 4-Cl  56 2-F, 5-Cl  57 3-Cl, 4-F  58 3-Cl, 5-F  59 3-Cl, 4-Br  60 3-Cl, 5-Br  61 3-F, 4-Cl  62 3-F, 4-Br  63 3-Br, 4-Cl  64 3-Br, 4-F  65 2,6-Cl₂, 4-Br  66 2-CH₃  67 3-CH₃  68 4-CH₃  69 2,3-(CH₃)₂  70 2,4-(CH₃)₂  71 2,5-(CH₃)₂  72 2,6-(CH₃)₂  73 3,4-(CH₃)₂  74 3,5-(CH₃)₂  75 2,3,5-(CH₃)₃  76 2,3,4-(CH₃)₃  77 2,3,6-(CH₃)₃  78 2,4,5-(CH₃)₃  79 2,4,6-(CH₃)₃  80 3,4,5-(CH₃)₃  81 2,3,4,6-(CH₃)₄  82 2,3,5,6-(CH₃)₄  83 2,3,4,5,6-(CH₃)₅  84 2-C₂H₅  85 3-C₂H₅  86 4-C₂H₅  87 2,4-(C₂H₅)₂  88 2,6-(C₂H₅)₂  89 3,5-(C₂H₅)₂  90 2,4,6-(C₂H₅)₃  91 2-n-C₃H₇  92 3-n-C₃H₇  93 4-n-C₃H₇  94 2-i-C₃H₇  95 3-i-C₃H₇  96 4-i-C₃H₇  97 2,4-(i-C₃H₇)₂  98 2,6-(i-C₃H₇)₂  99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H_(7, 5-CH) ₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—-C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H_(5, 4-Cl) 152 2-CH₂C₆H_(5, 4-Br) 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H_(11, 4-Cl) 156 2-cyclo-C₆H_(11, 4-Br) 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-O—C₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-9-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-COHCH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C (═NO-n-C₄H9)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NC-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O-C₆H₅ 475 3-O-C₆H₅ 476 4-O-C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N-OCH₃) 645 2-CH₃-4-(n-C₃H₇—C═N-OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N-O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N-O-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N-O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N-O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N-O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N-O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N-O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N-OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N-OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N-O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N-O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N-O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N-O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N-O-Proparoyl) 660 2-CH₃-4-(i-C₃H₇—C═N-O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N-O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-S-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃

TABLE 42

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 S-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH₃-Oxazolyl-4 234 3-C₆H₅-Oxazolyl-4 235 3-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 3-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 3-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 3-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 3-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 3-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 3-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 3-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 3-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 3-(4′-CN—C₆H₄)-Oxazolyl-4 245 3-(3′-CN—C₆H₄)-Oxazolyl-4 246 3-(2′-CN—C₆H₄)-Oxazolyl-4 247 3-(4′-Cl—C₆H₄)-Oxazolyl-4 248 3-(3′-Cl—C₆H₄)-Oxazolyl-4 249 3-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-l,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl I: R¹ = H, X = CH₃ II: R¹ = CH₃, X = CH₃ III: R¹ = C₂H₅, X = CH₃ IV: R¹ = Allyl, X = CH₃ V: R¹ = Propargyl, X = CH₃ VI: R¹ = CH₂—OCH₃, X = CH₃ VII: R¹ = CO₂CH₃, X = CH₃ VIII: R¹ = H, X = Cl IX: R¹ = CH₃, X = Cl X: R¹ = C₂H₅, X = Cl XI: R¹ = Allyl, X = Cl XII: R¹ = Propargyl, X = Cl XIII: R¹ = CH₂—OCH₃, X = Cl XIV: R¹ = CO₂CH₃, X = Cl

TABLE 43

No. T_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O—CH₂C₆H₅ 178 3-O—CH₂C₆H₅ 179 4-O—CH₂C₆H₅ 180 2-O—(CH₂)₃C₆H₅ 181 3-O—(CH₂)₃C₆H₅ 182 4-O—(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br₂, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅₎ 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)-CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Propargyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO—CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O-C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N-C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N-C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₄) 561 2-O-(3′-CF₃—C₆H₄) 562 2-O-(4′-CF₃—C₆H₄) 563 3-O-(2′-CF₃—C₆H₄) 564 3-O-(3′-CF₃—C₆H₄) 565 3-O-(4′-CF₃—C₆H₄) 566 4-O-(2′-CF₃—C₆H₄) 567 4-O-(3′-CF₃—C₆H₄) 568 4-O-(4′-CF₃—C₆H₄) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ 641 2-CH₃-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 642 2-CH₃-4-(C₂H₅—C═N—O—CH₂—CH₂—OCH₃) 643 2,5-(CH₃)₂-4-(CH₃—C═N—O—CH₂—CH₂—OCH₃) 644 2-CH₃-4-(n-C₃H₇—C═N—COH₃) 645 2-CH₃-4-(n-C₃H₇—C═N—OC₂H₅) 646 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₃H₇) 647 2-CH₃-4-(n-C₃H₇—C═N-i-C₃H₇) 648 2-CH₃-4-(n-C₃H₇—C═N—O-Allyl) 649 2-CH₃-4-(n-C₃H₇—C═N—O-trans-Chloroallyl) 650 2-CH₃-4-(n-C₃H₇—C═N—O-Propargyl) 651 2-CH₃-4-(n-C₃H₇—C═N—O-n-C₄H₉) 652 2-CH₃-4-(n-C₃H₇—C═N—O—CH₂—C₆H₅) 653 2-CH₃-4-(i-C₃H₇—C═N—OCH₃) 654 2-CH₃-4-(i-C₃H₇—C═N—OC₂H₅) 655 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₃H₇) 656 2-CH₃-4-(i-C₃H₇—C═N—O-i-C₃H₇) 657 2-CH₃-4-(i-C₃H₇—C═N—O-Allyl) 658 2-CH₃-4-(i-C₃H₇—C═N—O-trans-Chloroallyl) 659 2-CH₃-4-(i-C₃H₇—C═N—O-Propargyl) 660 2-CH₃-4-(i-C₃H₇—C═N—O-n-C₄H₉) 661 2-CH₃-4-(i-C₃H₇—C═N—O—CH₂—C₆H₅) 662 2-O-n-C₄H₉ 663 2-O-i-C₄H₉ 664 2-O-s-C₄H₉ 665 2-O-t-C₄H₉ 666 2-Neopentyloxy 667 3-O-n-C₄H₉ 668 3-O-i-C₄H₉ 669 3-O-s-C₄H₉ 670 3-O-t-C₄H₉ 671 3-Neopentyloxy 672 4-O-n-C₄H₉ 673 4-O-i-C₄H₉ 674 4-O-s-C₄H₉ 675 4-O-t-C₄H₉ 676 4-Neopentyloxy 677 3-CH₃-4-OCH₃ 678 3-CH₃-4-OC₂H₅ 679 3-CH₃-4-O-n-C₃H₇ 680 3-CH₃-4-O-n-C₄H₉ 681 3-CH₃-4-O-i-C₄H₉ 682 3-CH₃-4-O-s-C₄H₉ 683 3-CH₃-4-O-t-C₄H₉ 684 3-CH₃-4-Neopentyloxy 685 2-CH₃-3-OCH₃ 686 2-CH₃-4-OCH₃ 687 2-CH₃-5-OCH₃ 688 2-CH₃-6-OCH₃ 689 3-CH₃-4-OCH₃ 690 3-CH₃-5-OCH₃ 691 3-CH₃-6-OCH₃ 692 4-CH₃-5-O—CH₃ 693 4-CH₃-6-O—CH₃ 694 4-CH₃-6-OCH₃ 695 2-CH₃-3-O-i-C₃H₇ 696 2-CH₃-4-O-i-C₃H₇ 697 2-CH₃-5-O-i-C₃H₇ 698 2-CH₃-6-O-i-C₃H₇ 699 3-CH₃-4-O-i-C₃H₇ 700 3-CH₃-5-O-i-C₃H₇ 701 3-CH₃-6-O-i-C₃H₇ 702 4-CH₃-5-O-i-C₃H₇ 703 4-CH₃-6-O-i-C₃H₇ 704 5-CH₃-6-O-i-C₃H₇ 705 2-Cl-3-OCH₃ 706 2-Cl-4-OCH₃ 707 2-Cl-5-OCH₃ 708 2-Cl-6-OCH₃ 709 3-Cl-4-OCH₃ 710 3-Cl-5-OCH₃ 711 3-Cl-6-OCH₃ 712 4-Cl-5-OCH₃ 713 4-Cl-6-OCH₃ 714 5-Cl-6-OCH₃ I: R¹ = H, X = CH₃ II: R¹ = CH₃, X = CH₃ III: R¹ = C₂H₅, X = CH₃ IV: R¹ = Allyl, X = CH₃ V: R¹ = Propargyl, X = CH₃ VI: R¹ = CH₂—OCH₃, X = CH₃ VII: R¹ = CO₂CH₃, X = CH₃ VIII: R¹ = H, X = Cl IX: R¹ = CH₃, X = Cl X: R¹ = C₂H₅, X = Cl XI: R¹ = Allyl, X = Cl XII: R¹ = Propargyl, X = Cl XIII: R¹ = CH₂—OCH₃, X = Cl XIV: R¹ = CO₂CH₃, X = Cl

TABLE 44

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄)-Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4-(2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)—N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)—N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)—N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)—N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)—N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)—N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)—N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)—N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄)—N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazolyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH₃-Oxazolyl-4 234 3-C₆H₅-Oxazolyl-4 235 3-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 3-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 3-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 3-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 3-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 3-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 3-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 3-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 3-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 3-(4′-CN—C₆H₄)-Oxazolyl-4 245 3-(3′-CN—C₆H₄)-Oxazolyl-4 246 3-(2′-CN—C₆H₄)-Oxazolyl-4 247 3-(4′-Cl—C₆H₄)-Oxazolyl-4 248 3-(3′-Cl—C₆H₄)-Oxazolyl-4 249 3-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 384 1-Naphthyl 385 2-Naphthyl I: R¹ = H, X = CH₃ II: R¹ = CH₃, X = CH₃ III: R¹ = C₂H₅, X = CH₃ IV: R¹ = Allyl, X = CH₃ V: R¹ = Propargyl, X = CH₃ VI: R¹ = CH₂—OCH₃, X = CH₃ VII: R¹ = CO₂CH₃, X = CH₃ VIII: R¹ = H, X = Cl IX: R¹ = CH₃, X = Cl X: R¹ = C₂H₅, X = Cl XI: R¹ = Allyl, X = Cl XII: R¹ = Propargyl, X = Cl XIII: R¹ = CH₂—OCH₃, X = Cl XIV: R¹ = CO₂CH₃, X = Cl

TABLE 45

No. T_(m) 1 H 2 2-F 3 3-F 4 4-F 5 2,4-F₂ 6 2,4,6-F₃ 7 2,3,4,5,6-F₅ 8 2,3-F₂ 9 2-Cl 10 3-Cl 11 4-Cl 12 2,3-Cl₂ 13 2,4-Cl₂ 14 2,5-Cl₂ 15 2,6-Cl₂ 16 3,4-Cl₂ 17 3,5-Cl₂ 18 2,3,4-Cl₃ 19 2,3,5-Cl₃ 20 2,3,6-Cl₃ 21 2,4,5-Cl₃ 22 2,4,6-Cl₃ 23 3,4,5-Cl₃ 24 2,3,4,6-Cl₄ 25 2,3,5,6-Cl₄ 26 2,3,4,5,6-Cl₅ 27 2-Br 28 3-Br 29 4-Br 30 2,4-Br₂ 31 2,5-Br₂ 32 2,6-Br₂ 33 2,4,6-Br₃ 34 2,3,4,5,6-Br₅ 35 2-I 36 3-I 37 4-I 38 2,4-I₂ 39 2-Cl, 3-F 40 2-Cl, 4-F 41 2-Cl, 5-F 42 2-Cl, 6-F 43 2-Cl, 3-Br 44 2-Cl, 4-Br 45 2-Cl, 5-Br 46 2-Cl, 6-Br 47 2-Br, 3-Cl 48 2-Br, 4-Cl 49 2-Br, 5-Cl 50 2-Br, 3-F 51 2-Br, 4-F 52 2-Br, 5-F 53 2-Br, 6-F 54 2-F, 3-Cl 55 2-F, 4-Cl 56 2-F, 5-Cl 57 3-Cl, 4-F 58 3-Cl, 5-F 59 3-Cl, 4-Br 60 3-Cl, 5-Br 61 3-F, 4-Cl 62 3-F, 4-Br 63 3-Br, 4-Cl 64 3-Br, 4-F 65 2,6-Cl₂, 4-Br 66 2-CH₃ 67 3-CH₃ 68 4-CH₃ 69 2,3-(CH₃)₂ 70 2,4-(CH₃)₂ 71 2,5-(CH₃)₂ 72 2,6-(CH₃)₂ 73 3,4-(CH₃)₂ 74 3,5-(CH₃)₂ 75 2,3,5-(CH₃)₃ 76 2,3,4-(CH₃)₃ 77 2,3,6-(CH₃)₃ 78 2,4,5-(CH₃)₃ 79 2,4,6-(CH₃)₃ 80 3,4,5-(CH₃)₃ 81 2,3,4,6-(CH₃)₄ 82 2,3,5,6-(CH₃)₄ 83 2,3,4,5,6-(CH₃)₅ 84 2-C₂H₅ 85 3-C₂H₅ 86 4-C₂H₅ 87 2,4-(C₂H₅)₂ 88 2,6-(C₂H₅)₂ 89 3,5-(C₂H₅)₂ 90 2,4,6-(C₂H₅)₃ 91 2-n-C₃H₇ 92 3-n-C₃H₇ 93 4-n-C₃H₇ 94 2-i-C₃H₇ 95 3-i-C₃H₇ 96 4-i-C₃H₇ 97 2,4-(i-C₃H₇)₂ 98 2,6-(i-C₃H₇)₂ 99 3,5-(i-C₃H₇)₂ 100 2,4,6-(i-C₃H₇)₃ 101 2-s-C₄H₉ 102 3-s-C₄H₉ 103 4-s-C₄H₉ 104 2-t-C₄H₉ 105 3-t-C₄H₉ 106 4-t-C₄H₉ 107 2,3-(t-C₄H₉)₂ 108 2,4-(t-C₄H₉)₂ 109 2,5-(t-C₄H₉)₂ 110 2,6-(t-C₄H₉)₂ 111 3,4-(t-C₄H₉)₂ 112 2,4,6-(t-C₄H₉)₃ 113 4-n-C₉H₁₉ 114 4-n-C₁₂H₂₅ 115 4-n-C₁₅H₃₁ 116 4-(1,1,3,3-Tetramethylbutyl) 117 4-(2,4,4-Trimethylpropyl) 118 2-t-C₄H₉, 4-CH₃ 119 2-t-C₄H₉, 5-CH₃ 120 2,6-(t-C₄H₉)₂, 4-CH₃ 121 2-CH₃, 4-t-C₄H₉ 122 2-CH₃, 6-t-C₄H₉ 123 2-CH₃, 4-i-C₃H₇ 124 2-CH₃, 5-i-C₃H₇ 125 3-CH₃, 4-i-C₃H₇ 126 2-i-C₃H₇, 5-CH₃ 127 2,4-(t-C₄H₉)₂, 6-i-C₃H₇ 128 2-Allyl 129 3-Allyl 130 4-Allyl 131 2-Allyl, 6-CH₃ 132 2-cyclo-C₆H₁₁ 133 3-cyclo-C₆H₁₁ 134 4-cyclo-C₆H₁₁ 135 2,4-(cyclo-C₆H₁₁)₂, 6-CH₃ 136 2-CH₃, 4-cyclo-C₆H₁₁ 137 2-CH₂—C₆H₅ 138 3-CH₂—C₆H₅ 139 4-CH₂—C₆H₅ 140 2-CH₂—C₆H₅, 4-CH₃ 141 2-CH₃, 4-CH₂—C₆H₅ 142 2-C₆H₅ 143 3-C₆H₅ 144 4-C₆H₅ 145 4-(2-i-C₃H₇—C₆H₄) 146 4-C₆H₅, 2,6-(CH₃)₂ 147 2-Cl, 4-C₆H₅ 148 2-Br, 4-C₆H₅ 149 2-C₆H₅, 4-Cl 150 2-C₆H₅, 4-Br 151 2-CH₂C₆H₅, 4-Cl 152 2-CH₂C₆H₅, 4-Br 153 2-Cl, 4-CH₂C₆H₅ 154 2-Br, 4-CH₂C₆H₅ 155 2-cyclo-C₆H₁₁, 4-Cl 156 2-cyclo-C₆H₁₁, 4-Br 157 2-Cl, 4-cyclo-C₆H₁₁ 158 2-Br, 4-cyclo-C₆H₁₁ 159 2-OCH₃ 160 3-OCH₃ 161 4-OCH₃ 162 2-OC₂H₅ 163 3-O—C₂H₅ 164 4-O—C₂H₅ 165 2-O-n-C₃H₇ 166 3-O-n-C₃H₇ 167 4-O-n-C₃H₇ 168 2-O-i-C₃H₇ 169 3-O-i-C₃H₇ 170 4-O-i-C₃H₇ 171 2-O-n-C₆H₁₃ 172 3-O-n-C₆H₁₃ 173 4-O-n-C₆H₁₃ 174 2-O-n-C₈H₁₇ 175 3-O-n-C₈H₁₇ 176 4-O-n-C₈H₁₇ 177 2-O-CH₂C₆H₅ 178 3-O-CH₂C₆H₅ 179 4-O-CH₂C₆H₅ 180 2-O-(CH₂)₃C₆H₅ 181 3-O-(CH₂)₃C₆H₅ 182 4-O-(CH₂)₃C₆H₅ 183 2,4-(OCH₃)₂ 184 2-CF₃ 185 3-CF₃ 186 4-CF₃ 187 2-OCF₃ 188 3-OCF₃ 189 4-OCF₃ 190 3-OCH₂CHF₂ 191 2-NO₂ 192 3-NO₂ 193 4-NO₂ 194 2-CN 195 3-CN 196 4-CN 197 2-CH₃, 3-Cl 198 2-CH₃, 4-Cl 199 2-CH₃, 5-Cl 200 2-CH₃, 6-Cl 201 2-CH₃, 3-F 202 2-CH₃, 4-F 203 2-CH₃, 5-F 204 2-CH₃, 6-F 205 2-CH₃, 3-Br 206 2-CH₃, 4-Br 207 2-CH₃, 5-Br 208 2-CH₃, 6-Br 209 2-Cl, 3-CH₃ 210 2-Cl, 4-CH₃ 211 2-Cl, 5-CH₃ 212 2-F, 3-CH₃ 213 2-F, 4-CH₃ 214 2-F, 5-CH₃ 215 2-Br, 3-CH₃ 216 2-Br, 4-CH₃ 217 2-Br, 5-CH₃ 218 3-CH₃, 4-Cl 219 3-CH₃, 5-Cl 220 3-CH₃, 4-F 221 3-CH₃, 5-F 222 3-CH₃, 4-Br 223 3-CH₃, 5-Br 224 3-F, 4-CH₃ 225 3-Cl, 4-CH₃ 226 3-Br, 4-CH₃ 227 2-Cl, 4,5-(CH₃)₂ 228 2-Br, 4,5-(CH₃)₂ 229 2-Cl, 3,5-(CH₃)₂ 230 2-Br, 3,5-(CH₃)₂ 231 2,6-Cl₂, 4-CH₃ 232 2,6-F₂, 4-CH₃ 233 2,6-Br₂, 4-CH₃ 234 2,4-Br, 6-CH₃ 235 2,4-F₂, 6-CH₃ 236 2,4-Br₂, 6-CH₃ 237 2,6-(CH₃)₂, 4-F 238 2,6-(CH₃)₂, 4-Cl 239 2,6-(CH₃)₂, 4-Br 240 3,5-(CH₃)₂, 4-F 241 3,5-(CH₃)₂, 4-Cl 242 3,5-(CH₃)₂, 4-Br 243 2,3,6-(CH₃)₃, 4-F 244 2,3,6-(CH₃)₃, 4-Cl 245 2,3,6-(CH₃)₃, 4-Br 246 2,4-(CH₃)₂, 6-F 247 2,4-(CH₃)₂, 6-Cl 248 2,4-(CH₃)₂, 6-Br 249 2-i-C₃H₇, 4-Cl, 5-CH₃ 250 2-Cl, 4-NO₂ 251 2-NO₂, 4-Cl 252 2-OCH₃, 5-NO₂ 253 2,4-Cl₂, 5-NO₂ 254 2,4-Cl₂, 6-NO₂ 255 2,6-Cl₂, 4-NO₂ 256 2,6-Br₂, 4-NO₂ 257 2,6-I₂, 4-NO₂ 258 2-CH₃, 5-i-C₃H₇, 4-Cl 259 2-CO₂CH₃ 260 3-CO₂CH₃ 261 4-CO₂CH₃ 262 2-CO₂(C₂H₅) 263 3-CO₂(C₂H₅) 264 4-CO₂(C₂H₅) 265 2-CO₂(n-C₃H₇) 266 3-CO₂(n-C₃H₇) 267 4-CO₂(n-C₃H₇) 268 2-CO₂(i-C₃H₇) 269 3-CO₂(i-C₃H₇) 270 4-CO₂(i-C₃H₇) 271 2-CO₂(n-C₆H₁₃) 272 3-CO₂(n-C₆H₁₃) 273 4-CO₂(n-C₆H₁₃) 274 2-CH₂—OCH₃ 275 3-CH₂—OCH₃ 276 4-CH₂—OCH₃ 277 2-CH₂O(C₂H₅) 278 3-CH₂O(C₂H₅) 279 4-CH₂O(C₂H₅) 280 2-CH₂O(n-C₃H₇) 281 3-CH₂O(n-C₃H₇) 282 4-CH₂O(n-C₃H₇) 283 2-CH₂O(i-C₃H₇) 284 3-CH₂O(i-C₃H₇) 285 4-CH₂O(i-C₃H₇) 286 2-CHO 287 3-CHO 288 4-CHO 289 2-CO—CH₃ 290 3-CO—CH₃ 291 4-CO—CH₃ 292 2-CO—CH₂—CH₃ 293 3-CO—CH₂—CH₃ 294 4-CO—CH₂—CH₃ 295 2-CO—CH₂—CH₂—CH₃ 296 3-CO—CH₂—CH₂—CH₃ 297 4-CO—CH₂—CH₂—CH₃ 298 2-CO—CH(CH₃)—CH₃ 299 3-CO—CH(CH₃)—CH₃ 300 4-CO—CH(CH₃)—CH₃ 301 2-Me-4-CHO 302 2-Me-4-CH₃—CO 303 2-Me-4-CH₃—CH₂—CO 304 2-Me-4-CH₃—CH₂—CH₂—CO 305 2-Me-4-CH₃—CH(CH₃)—CO 306 2,5-Me₂-4-CHO 307 2,5-Me₂-4-CH₃—CO 308 2,5-Me₂-4-CH₃—CH₂—CO 309 2,5-Me₂-4-CH₃—CH₂—CH₂—CO 310 2,5-Me₂-4-CH₃—CH(CH₃)—CO 311 2-Cl-4-CHO 312 2-Cl-4-CH₃—CO 313 2-Cl-4-CH₃—CH₂—CO 314 2-Cl-4-CH₃—CH(CH₃)—CO 315 2,5-Cl₂-4-CHO 316 2,5-Cl₂-4-CH₃—CO 317 2,5-Cl₂-4-CH₃—CH₂—CO 318 2,5-Cl₂-4-CH₃—CH₂—CH₂—CO 319 2,5-Cl₂-4-CH₃—CH(CH₃)—CO 320 2-C(═NOCH₃)—CH₃ 321 3-C(═NOCH₃)—CH₃ 322 4-C(═NOCH₃)—CH₃ 323 2-C(═NOC₂H₅)—CH₃ 324 3-C(═NOC₂H₅)—CH₃ 325 4-C(═NOC₂H₅)—CH₃ 326 2-C(═NO-n-C₃H₇)—CH₃ 327 3-C(═NO-n-C₃H₇)—CH₃ 328 4-C(═NO-n-C₃H₇)—CH₃ 329 2-C(═NO-i-C₃H₇)—CH₃ 330 3-C(═NO-i-C₃H₇)—CH₃ 331 4-C(═NO-i-C₃H₇)—CH₃ 332 2-C(═NO-Allyl)—CH₃ 333 3-C(═NO-Allyl)-CH₃ 334 4-C(═NO-Allyl)-CH₃ 335 2-C(═NO-trans-Chloroallyl)-CH₃ 336 3-C(═NO-trans-Chloroallyl)-CH₃ 337 4-C(═NO-trans-Chloroallyl)-CH₃ 338 2-C(═NO-Propargyl)-CH₃ 339 3-C(═NO-Propargyl)-CH₃ 340 4-C(═NO-Proparoyl)-CH₃ 341 2-C(═NO-n-C₄H₉)—CH₃ 342 3-C(═NO-n-C₄H₉)—CH₃ 343 4-C(═NO-n-C₄H₉)—CH₃ 344 2-C(═NO—CH₂—C₆H₅)—CH₃ 345 3-C(═NO—CH₂—C₆H₅)—CH₃ 346 4-C(═NO—CH₂—C₆H₅)—CH₃ 347 2-CH₃-4-CH═NOCH₃ 348 2-CH₃-4-CH═NOC₂H₅ 349 2-CH₃-4-CH═NO-n-C₃H₇ 350 2-CH₃-4-CH═NO-i-C₃H₇ 351 2-CH₃-4-CH═NO-Allyl 352 2-CH₃-4-CH═NO-(trans-Chloroallyl) 353 2-CH₃-4-CH═NO-Propargyl 354 2-CH₃-4-CH═NO-n-C₄H₉ 355 2-CH₃-4-CH═NO—CH₂—C₆H₅ 356 2-CH₃-4-(CH₃—C═NOCH₃) 357 2-CH₃-4-(CH₃—C═NOC₂H₅) 358 2-CH₃-4-(CH₃—C═NO-n-C₃H₇) 359 2-CH₃-4-(CH₃—C═NO-i-C₃H₇) 360 2-CH₃-4-(CH₃—C═NO-Allyl) 361 2-CH₃-4-(CH₃—C═NO-trans-Chloroallyl) 362 2-CH₃-4-(CH₃—C═NO-Propargyl) 363 2-CH₃-4-(CH₃—C═NO-n-C₄H₉) 364 2-CH₃-4-(CH₃—C═NO—CH₂—C₆H₅) 365 2-CH₃-4-(C₂H₅—C═NO—CH₃) 366 2-CH₃-4-(C₂H₅—C═NO—C₂H₅) 367 2-CH₃-4-(C₂H₅—C═NO-n-C₃H₇) 368 2-CH₃-4-(C₂H₅—C═NO-i-C₃H₇ 369 2-CH₃-4-(C₂H₅—C═NO-Allyl) 370 2-CH₃-4-(C₂H₅—C═NO-trans-Chloroallyl) 371 2-CH₃-4-(C₂H₅—C═NO-Propargyl) 372 2-CH₃-4-(C₂H₅—C═NO-n-C₄H₉) 373 2-CH₃-4-(C₂H₅—C═NO—CH₂—C₆H₅) 374 2,5-(CH₃)₂-4-(CH₃—C═NOCH₃) 375 2,5-(CH₃)₂-4-(CH₃—C═NOC₂H₅) 376 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₃H₇) 377 2,5-(CH₃)₂-4-(CH₃—C═NO-i-C₃H₇) 378 2,5-(CH₃)₂-4-(CH₃—C═NO-Allyl) 379 2,5-(CH₃)₂-4-(CH₃—C═NO-trans-Chloroallyl) 380 2,5-(CH₃)₂-4-(CH₃—C═NO-Proparyl) 381 2,5-(CH₃)₂-4-(CH₃—C═NO-n-C₄H₉) 382 2,5-(CH₃)₂-4-(CH₃—C═NO-CH₂—C₆H₅) 383 2-C₆H₅ 384 3-C₆H₅ 385 4-C₆H₅ 386 2-(2′-F—C₆H₄) 387 2-(3′-F—C₆H₄) 388 2-(4′-F—C₆H₄) 389 3-(2′-F—C₆H₄) 390 3-(3′-F—C₆H₄) 391 3-(4′-F—C₆H₄) 392 4-(2′-F—C₆H₄) 393 4-(3′-F—C₆H₄) 394 4-(4′-F—C₆H₄) 395 2-(2′-Cl—C₆H₄) 396 2-(3′-Cl—C₆H₄) 397 2-(4′-Cl—C₆H₄) 398 3-(2′-Cl—C₆H₄) 399 3-(3′-Cl—C₆H₄) 400 3-(4′-Cl—C₆H₄) 401 4-(2′-Cl—C₆H₄) 402 4-(3′-Cl—C₆H₄) 403 4-(4′-Cl—C₆H₄) 405 2-(2′-CH₃—C₆H₄) 406 2-(3′-CH₃—C₆H₄) 407 2-(4′-CH₃—C₆H₄) 408 3-(2′-CH₃—C₆H₄) 409 3-(3′-CH₃—C₆H₄) 410 3-(4′-CH₃—C₆H₄) 411 4-(2′-CH₃—C₆H₄) 412 4-(3′-CH₃—C₆H₄) 413 4-(4′-CH₃—C₆H₄) 414 2-(2′-CH₃—CO—C₆H₄) 415 2-(3′-CH₃—CO—C₆H₄) 416 2-(4′-CH₃—CO—C₆H₄) 417 3-(2′-CH₃—CO—C₆H₄) 418 3-(3′-CH₃—CO—C₆H₄) 419 3-(4′-CH₃—CO—C₆H₄) 420 4-(2′-CH₃—CO—C₆H₄) 421 4-(3′-CH₃—CO—C₆H₄) 422 4-(4′-CH₃—CO—C₆H₄) 423 2-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 424 2-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 425 2-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 426 3-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 427 3-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 428 3-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 429 4-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 430 4-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 431 4-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 432 2-(2′-CH₃O₂C—C₆H₄) 433 2-(3′-CH₃O₂C—C₆H₄) 434 2-(4′-CH₃O₂C—C₆H₄) 435 3-(2′-CH₃O₂C—C₆H₄) 436 3-(3′-CH₃O₂C—C₆H₄) 437 3-(4′-CH₃O₂C—C₆H₄) 438 4-(2′-CH₃O₂C—C₆H₄) 439 4-(3′-CH₃O₂C—C₆H₄) 440 4-(4′-CH₃O₂C—C₆H₄) 441 2-(2′-CH₃O—C₆H₄) 442 2-(3′-CH₃O—C₆H₄) 443 2-(4′-CH₃O—C₆H₄) 444 3-(2′-CH₃O—C₆H₄) 445 3-(3′-CH₃O—C₆H₄) 446 3-(4′-CH₃O—C₆H₄) 447 4-(2′-CH₃O—C₆H₄) 448 4-(3′-CH₃O—C₆H₄) 449 4-(4′-CH₃O—C₆H₄) 450 2-(2′-O₂N—C₆H₄) 451 2-(3′-O₂N—C₆H₄) 452 2-(4′-O₂N—C₆H₄) 453 3-(2′-O₂N—C₆H₄) 454 3-(3′-O₂N—C₆H₄) 455 3-(4′-O₂N—C₆H₄) 456 4-(2′-O₂N—C₆H₄) 457 4-(3′-O₂N—C₆H₄) 458 4-(4′-O₂N—C₆H₄) 459 2-(2′-NC—C₆H₄) 460 2-(3′-NC—C₆H₄) 461 2-(4′-NC—C₆H₄) 462 3-(2′-NC—C₆H₄) 463 3-(3′-NC—C₆H₄) 464 3-(4′-NC—C₆H₄) 465 4-(2′-NC—C₆H₄) 466 4-(3′-NC—C₆H₄) 467 4-(4′-NC—C₆H₄) 468 2-(2′-CF₃—C₆H₄) 469 2-(3′-CF₃—C₆H₄) 470 2-(4′-CF₃—C₆H₄) 471 3-(2′-CF₃—C₆H₄) 472 3-(3′-CF₃—C₆H₄) 473 3-(4′-CF₃—C₆H₄) 474 4-(2′-CF₃—C₆H₄) 475 4-(3′-CF₃—C₆H₄) 476 4-(4′-CF₃—C₆H₄) 477 2-O—C₆H₅ 475 3-O—C₆H₅ 476 4-O—C₆H₅ 478 2-O-(2′-F—C₆H₄) 479 2-O-(3′-F—C₆H₄) 480 2-O-(4′-F—C₆H₄) 481 3-O-(2′-F—C₆H₄) 482 3-O-(3′-F—C₆H₄) 483 3-O-(4′-F—C₆H₄) 484 4-O-(2′-F—C₆H₄) 485 4-O-(3′-F—C₆H₄) 486 4-O-(4′-F—C₆H₄) 487 2-O-(2′-Cl—C₆H₄) 488 2-O-(3′-Cl—C₆H₄) 489 2-O-(4′-Cl—C₆H₄) 490 3-O-(2′-Cl—C₆H₄) 491 3-O-(3′-Cl—C₆H₄) 492 3-O-(4′-Cl—C₆H₄) 493 3-O-(4′-Cl—C₆H₄) 494 4-O-(2′-Cl—C₆H₄) 495 4-O-(3′-Cl—C₆H₄) 496 4-O-(4′-Cl—C₆H₄) 497 2-O-(2′-CH₃—C₆H₄) 498 2-O-(3′-CH₃—C₆H₄) 499 2-O-(4′-CH₃—C₆H₄) 500 3-O-(2′-CH₃—C₆H₄) 501 3-O-(3′-CH₃—C₆H₄) 502 3-O-(4′-CH₃—C₆H₄) 503 4-O-(2′-CH₃—C₆H₄) 504 4-O-(3′-CH₃—C₆H₄) 505 4-O-(4′-CH₃—C₆H₄) 506 2-O-(2′-CH₃—CO—C₆H₄) 507 2-O-(3′-CH₃—CO—C₆H₄) 508 2-O-(4′-CH₃—CO—C₆H₄) 509 3-O-(2′-CH₃—CO—C₆H₄) 510 3-O-(3′-CH₃—CO—C₆H₄) 511 3-O-(4′-CH₃—CO—C₆H₄) 512 4-O-(2′-CH₃—CO—C₆H₄) 513 4-O-(3′-CH₃—CO—C₆H₄) 514 4-O-(4′-CH₃—CO—C₆H₄) 515 2-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 516 2-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 517 2-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 518 3-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 519 3-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 520 3-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 521 4-O-(2′-(CH₃—C(═NOAllyl))-C₆H₄) 522 4-O-(3′-(CH₃—C(═NOAllyl))-C₆H₄) 523 4-O-(4′-(CH₃—C(═NOAllyl))-C₆H₄) 524 2-O-(2′-CH₃O₂C—C₆H₄) 525 2-O-(3′-CH₃O₂C—C₆H₄) 526 2-O-(4′-CH₃O₂C—C₆H₄) 527 3-O-(2′-CH₃O₂C—C₆H₄) 528 3-O-(3′-CH₃O₂C—C₆H₄) 529 3-O-(4′-CH₃O₂C—C₆H₄) 530 4-O-(2′-CH₃O₂C—C₆H₄) 531 4-O-(3′-CH₃O₂C—C₆H₄) 532 4-O-(4′-CH₃O₂C—C₆H₄) 533 2-O-(2′-CH₃O—C₆H₄) 534 2-O-(3′-CH₃O—C₆H₄) 535 2-O-(4′-CH₃O—C₆H₄) 536 3-O-(2′-CH₃O—C₆H₄) 537 3-O-(3′-CH₃O—C₆H₄) 538 3-O-(4′-CH₃O—C₆H₄) 539 4-O-(2′-CH₃O—C₆H₄) 540 4-O-(3′-CH₃O—C₆H₄) 541 4-O-(4′-CH₃O—C₆H₄) 542 2-O-(2′-O₂N—C₆H₄) 543 2-O-(3′-O₂N—C₆H₄) 544 2-O-(4′-O₂N—C₆H₄) 545 3-O-(2′-O₂N—C₆H₄) 546 3-O-(3′-O₂N—C₆H₄) 547 3-O-(4′-O₂N—C₆H₄) 548 4-O-(2′-O₂N—C₆H₄) 549 4-O-(3′-O₂N—C₆H₄) 550 4-O-(4′-O₂N—C₆H₄) 551 2-O-(2′-NC—C₆H₄) 552 2-O-(3′-NC—C₆H₄) 553 2-O-(4′-NC—C₆H₄) 554 3-O-(2′-NC—C₆H₄) 555 3-O-(3′-NC—C₆H₄) 556 3-O-(4′-NC—C₆H₄) 557 4-O-(2′-NC—C₆H₄) 558 4-O-(3′-NC—C₆H₄) 559 4-O-(4′-NC—C₆H₄) 560 2-O-(2′-CF₃—C₆H₅) 561 2-O-(3′-CF₃—C₆H₅) 562 2-O-(4′-CF₃—C₆H₅) 563 3-O-(2′-CF₃—C₆H₅) 564 3-O-(3′-CF₃—C₆H₅) 565 3-O-(4′-CF₃—C₆H₅) 566 4-O-(2′-CF₃—C₆H₅) 567 4-O-(3′-CF₃—C₆H₅) 568 4-O-(4′-CF₃—C₆H₅) 569 2-Pyridinyl-2′ 570 2-Pyridinyl-3′ 571 2-Pyridinyl-4′ 572 3-Pyridinyl-2′ 573 3-Pyridinyl-3′ 574 3-Pyridinyl-4′ 575 4-Pyridinyl-2′ 576 4-Pyridinyl-3′ 577 4-Pyridinyl-4′ 578 2-Pyrimidinyl-2′ 579 2-Pyrimidinyl-3′ 580 2-Pyrimidinyl-4′ 581 3-Pyrimidinyl-2′ 582 3-Pyrimidinyl-3′ 583 3-Pyrimidinyl-4′ 584 4-Pyrimidinyl-2′ 585 4-Pyrimidinyl-3′ 586 4-Pyrimidinyl-4′ 587 2-Pyrazolyl-1′ 588 2-Pyrazolyl-3′ 589 2-Pyrazolyl-4′ 590 3-Pyrazolyl-1′ 591 3-Pyrazolyl-3′ 592 3-Pyrazolyl-4′ 593 4-Pyrazolyl-1′ 594 4-Pyrazolyl-3′ 595 4-Pyrazolyl-4′ 596 2-Isoxazolyl-3′ 597 2-Isoxazolyl-4′ 598 2-Isoxazolyl-5′ 599 3-Isoxazolyl-3′ 600 3-Isoxazolyl-4′ 601 3-Isoxazolyl-5′ 602 4-Isoxazolyl-3′ 603 4-Isoxazolyl-4′ 604 4-Isoxazolyl-5′ 605 2-Isothiazolyl-3′ 606 2-Isothiazolyl-4′ 607 2-Isothiazolyl-5′ 608 3-Isothiazolyl-3′ 609 3-Isothiazolyl-4′ 610 3-Isothiazolyl-5′ 611 4-Isothiazolyl-3′ 612 4-Isothiazolyl-4′ 613 4-Isothiazolyl-5′ 614 2-Imidazolyl-1′ 615 2-Imidazolyl-2′ 616 2-Imidazolyl-4′ 617 3-Imidazolyl-1′ 618 3-Imidazolyl-2′ 619 3-Imidazolyl-4′ 620 4-Imidazolyl-1′ 621 4-Imidazolyl-2′ 622 4-Imidazolyl-4′ 623 2-Oxazolyl-2′ 624 2-Oxazolyl-4′ 625 2-Oxazolyl-5′ 626 3-Oxazolyl-2′ 627 3-Oxazolyl-4′ 628 3-Oxazolyl-5′ 629 4-Oxazolyl-2′ 630 4-Oxazolyl-4′ 631 4-Oxazolyl-5′ 632 2-Thiazolyl-2′ 633 2-Thiazolyl-4′ 634 2-Thiazolyl-5′ 635 3-Thiazolyl-2′ 636 3-Thiazolyl-4′ 637 3-Thiazolyl-5′ 638 4-Thiazolyl-2′ 639 4-Thiazolyl-4′ 640 4-Thiazolyl-5′ I: R¹ = H, X = CH₃ II: R¹ = CH₃, X = CH₃ III: R¹ = C₂H₅, X = CH₃ IV: R¹ = Allyl, X = CH₃ V: R¹ = Propargyl, X = CH₃ VI: R¹ = CH₂—OCH₃, X = CH₃ VII: R¹ = CO₂CH₃, X = CH₃ VIII: R¹ = H, X = Cl IX: R¹ = CH₃, X = Cl X: R¹ = C₂H₅, X = Cl XI: R¹ = Allyl, X = Cl XII: R¹ = Propargyl, X = Cl XIII: R¹ = CH₂—OCH₃, X = Cl XIV: R¹ = CO₂CH₃, X = Cl

TABLE 46

No. B 1 Pyrrolyl-3 2 N—CH₃-Pyrrolyl-3 3 N—C₆H₅-Pyrrolyl-3 4 N-(4′-CH₃—C₆H₄)-Pyrrolyl-3 5 N-(3′-CH₃—C₆H₄)-Pyrrolyl-3 6 N-(2′-CH₃—C₆H₄)-Pyrrolyl-3 7 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-3 8 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-3 9 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-3 10 N-(4′-NO₂—C₆H₄)-Pyrrolyl-3 11 N-(3′-NO₂—C₆H₄)-Pyrrolyl-3 12 N-(2′-NO₂—C₆H₄)-Pyrrolyl-3 13 N-(4′-CN—C₆H₄)-Pyrrolyl-3 14 N-(3′-CN—C₆H₄)-Pyrrolyl-3 15 N-(2′-CN—C₆H₄)-Pyrrolyl-3 16 N-(4′-Cl—C₆H₄)-Pyrrolyl-3 17 N-(3′-Cl—C₆H₄)-Pyrrolyl-3 18 N-(2′-Cl—C₆H₄)-Pyrrolyl-3 19 Pyrrolyl-2 20 N—CH₃-Pyrrolyl-2 21 N—C₆H₅-Pyrrolyl-2 22 N-(4′-CH₃—C₆H₄)-Pyrrolyl-2 23 N-(3′-CH₃—C₆H₄)-Pyrrolyl-2 24 N-(2′-CH₃—C₆H₄)-Pyrrolyl-2 25 N-(4′-CH₃O—C₆H₄)-Pyrrolyl-2 26 N-(3′-CH₃O—C₆H₄)-Pyrrolyl-2 27 N-(2′-CH₃O—C₆H₄)-Pyrrolyl-2 28 N-(4′-NO₂—C₆H₄)-Pyrrolyl-2 29 N-(3′-NO₂—C₆H₄)-Pyrrolyl-2 30 N-(2′-NO₂—C₆H₄)-Pyrrolyl-2 31 N-(4′-CN—C₆H₄)-Pyrrolyl-2 32 N-(3′-CN—C₆H₄)-Pyrrolyl-2 33 N-(2′-CN—C₆H₄)-Pyrrolyl-2 34 N-(4′-Cl—C₆H₄)-Pyrrolyl-2 35 N-(3′-Cl—C₆H₄)-Pyrrolyl-2 36 N-(2′-Cl—C₆H₄)-Pyrrolyl-2 37 Furyl-2 38 5-CH₃-Furyl-2 39 5-C₆H₅-Furyl-2 40 5-(4′-CH₃—C₆H₄)-Furyl-2 41 5-(3′-CH₃—C₆H₄)-Furyl-2 42 5-(2′-CH₃—C₆H₄)-Furyl-2 43 5-(4′-CH₃O—C₆H₄)-Furyl-2 44 5-(3′-CH₃O—C₆H₄)-Furyl-2 45 5-(2′-CH₃O—C₆H₄)-Furyl-2 46 5-(4′-NO₂—C₆H₄)-Furyl-2 47 5-(3′-NO₂—C₆H₄)-Furyl-2 48 5-(2′-NO₂—C₆H₄)-Furyl-2 49 5-(4′-CN—C₆H₄)-Furyl-2 50 5-(3′-CN—C₆H₄)-Furyl-2 51 5-(2′-CN—C₆H₄)-Furyl-2 52 5-(4′-Cl—C₆H₄)-Furyl-2 53 5-(3′-Cl—C₆H₄)-Furyl-2 54 5-(2′-Cl—C₆H₄)-Furyl-2 55 4-CH₃-Furyl-2 56 4-C₆H₅-Furyl-2 57 4-(4′-CH₃—C₆H₄)-Furyl-2 58 4-(3′-CH₃—C₆H₄)-Furyl-2 59 4-(2′-CH₃—C₆H₄)-Furyl-2 60 4-(4′-CH₃O—C₆H₄)-Furyl-2 61 4-(3′-CH₃O—C₆H₄)-Furyl-2 62 4-(2′-CH₃O—C₆H₄)-Furyl-2 63 4-(4′-NO₂—C₆H₄)-Furyl-2 64 4-(3′-NO₂—C₆H₄)-Furyl-2 65 4-(2′-NO₂—C₆H₄)-Furyl-2 66 4-(4′-CN—C₆H₄)-Furyl-2 67 4-(3′-CN—C₆H₄)-Furyl-2 68 4-(2′-CN—C₆H₄)-Furyl-2 69 4-(4′-Cl—C₆H₄)-Furyl-2 70 4-(3′-Cl—C₆H₄)-Furyl-2 71 4-(2′-Cl—C₆H₄)-Furyl-2 72 Thienyl-2 73 5-CH₃-Thienyl-2 74 5-C₆H₅-Thienyl-2 75 5-(4′-CH₃—C₆H₄)-Thienyl-2 76 5-(3′-CH₃—C₆H₄)-Thienyl-2 77 5-(2′-CH₃—C₆H₄)-Thienyl-2 78 5-(4′-CH₃O—C₆H₄)-Thienyl-2 79 5-(3′-CH₃O—C₆H₄)-Thienyl-2 80 5-(2′-CH₃O—C₆H₄)-Thienyl-2 81 5-(4′-NO₂—C₆H₄)-Thienyl-2 82 5-(3′-NO₂—C₆H₄)-Thienyl-2 83 5-(2′-NO₂—C₆H₄)-Thienyl-2 84 5-(4′-CN—C₆H₄)-Thienyl-2 85 5-(3′-CN—C₆H₄)-Thienyl-2 86 5-(2′-CN—C₆H₄)-Thienyl-2 87 5-(4′-Cl—C₆H₄)-Thienyl-2 88 5-(3′-Cl—C₆H₄)-Thienyl-2 89 5-(2′-Cl—C₆H₄)-Thienyl-2 90 4-CH₃-Thienyl-2 91 4-C₆H₅-Thienyl-2 92 4-(4′-CH₃—C₆H₄)-Thienyl-2 93 4-(3′-CH₃—C₆H₄)-Thienyl-2 94 4-(2′-CH₃—C₆H₄) Thienyl-2 95 4-(4′-CH₃O—C₆H₄)-Thienyl-2 96 4-(3′-CH₃O—C₆H₄)-Thienyl-2 97 4-(2′-CH₃O—C₆H₄)-Thienyl-2 98 4-(4′-NO₂—C₆H₄)-Thienyl-2 99 4-(3′-NO₂—C₆H₄)-Thienyl-2 100 4 (2′-NO₂—C₆H₄)-Thienyl-2 101 4-(4′-CN—C₆H₄)-Thienyl-2 102 4-(3′-CN—C₆H₄)-Thienyl-2 103 4-(2′-CN—C₆H₄)-Thienyl-2 104 4-(4′-Cl—C₆H₄)-Thienyl-2 105 4-(3′-Cl—C₆H₄)-Thienyl-2 106 4-(2′-Cl—C₆H₄)-Thienyl-2 107 Thienyl-3 108 5-CH₃-Thienyl-3 109 5-C₆H₅-Thienyl-3 110 5-(4′-CH₃—C₆H₄)-Thienyl-3 111 5-(3′-CH₃—C₆H₄)-Thienyl-3 112 5-(2′-CH₃—C₆H₄)-Thienyl-3 113 5-(4′-CH₃O—C₆H₄)-Thienyl-3 114 5-(3′-CH₃O—C₆H₄)-Thienyl-3 115 5-(2′-CH₃O—C₆H₄)-Thienyl-3 116 5-(4′-NO₂—C₆H₄)-Thienyl-3 117 5-(3′-NO₂—C₆H₄)-Thienyl-3 118 5-(2′-NO₂—C₆H₄)-Thienyl-3 119 5-(4′-CN—C₆H₄)-Thienyl-3 120 5-(3′-CN—C₆H₄)-Thienyl-3 121 5-(2′-CN—C₆H₄)-Thienyl-3 122 5-(4′-Cl—C₆H₄)-Thienyl-3 123 5-(3′-Cl—C₆H₄)-Thienyl-3 124 5-(2′-Cl—C₆H₄)-Thienyl-3 125 Pyrazolyl-4 126 N—CH₃-Pyrazolyl-4 127 N—C₆H₅-Pyrazolyl-4 128 N-(4′-CH₃—C₆H₄)-Pyrazolyl-4 129 N-(3′-CH₃—C₆H₄)-Pyrazolyl-4 130 N-(2′-CH₃—C₆H₄)-Pyrazolyl-4 131 N-(4′-CH₃O—C₆H₄)-Pyrazolyl-4 132 N-(3′-CH₃O—C₆H₄)-Pyrazolyl-4 133 N-(2′-CH₃O—C₆H₄)-Pyrazolyl-4 134 N-(4′-NO₂—C₆H₄)-Pyrazolyl-4 135 N-(3′-NO₂—C₆H₄)-Pyrazolyl-4 136 N-(2′-NO₂—C₆H₄)-Pyrazolyl-4 137 N-(4′-CN—C₆H₄)-Pyrazolyl-4 138 N-(3′-CN—C₆H₄)-Pyrazolyl-4 139 N-(2′-CN—C₆H₄)-Pyrazolyl-4 140 N-(4′-Cl—C₆H₄)-Pyrazolyl-4 141 N-(3′-Cl—C₆H₄)-Pyrazolyl-4 142 N-(2′-Cl—C₆H₄)-Pyrazolyl-4 143 3-CH₃—N-Methylpyrazolyl-4 144 3-C₆H₅—N-Methylpyrazolyl-4 145 3-(4′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 146 3-(3′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 147 3-(2′-CH₃—C₆H₄)-N-Methylpyrazolyl-4 148 3-(4′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 149 3-(3′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 150 3-(2′-CH₃O—C₆H₄)-N-Methylpyrazolyl-4 151 3-(4′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 152 3-(3′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 153 3-(2′-NO₂—C₆H₄)-N-Methylpyrazolyl-4 154 3-(4′-CN—C₆H₄)-N-Methylpyrazolyl-4 155 3-(3′-CN—C₆H₄)-N-Methylpyrazolyl-4 156 3-(2′-CN—C₆H₄)-N-Methylpyrazolyl-4 157 3-(4′-Cl—C₆H₄)-N-Methylpyrazolyl-4 158 3-(3′-Cl—C₆H₄)-N-Methylpyrazolyl-4 159 3-(2′-Cl—C₆H₄) N-Methylpyrazolyl-4 160 Isoxazolyl-5 161 3-CH₃-Isoxazolyl-5 162 3-C₆H₅-Isoxazolyl-5 163 3-(4′-CH₃—C₆H₄)-Isoxazolyl-5 164 3-(3′-CH₃—C₆H₄)-Isoxazolyl-5 165 3-(2′-CH₃—C₆H₄)-Isoxazolyl-5 166 3-(4′-CH₃O—C₆H₄)-Isoxazolyl-5 167 3-(3′-CH₃O—C₆H₄)-Isoxazolyl-5 168 3-(2′-CH₃O—C₆H₄)-Isoxazolyl-5 169 3-(4′-NO₂—C₆H₄)-Isoxazolyl-5 170 3-(3′-NO₂—C₆H₄)-Isoxazolyl-5 171 3-(2′-NO₂—C₆H₄)-Isoxazolyl-5 172 3-(4′-CN—C₆H₄)-Isoxazolyl-5 173 3-(3′-CN—C₆H₄)-Isoxazolyl-5 174 3-(2′-CN—C₆H₄)-Isoxazolyl-5 175 3-(4′-Cl—C₆H₄)-Isoxazolyl-5 176 3-(3′-Cl—C₆H₄)-Isoxazolyl-5 177 3-(2′-Cl—C₆H₄)-Isoxazolyl-5 178 4-Chloroisoxazolyl-5 179 3-CH₃-4-Chloroisoxazolyl-5 180 3-C₆H₅-4-Chloroisoxazoyl-5 181 3-(4′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 182 3-(3′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 183 3-(2′-CH₃—C₆H₄)-4-Chloroisoxazolyl-5 184 3-(4′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 185 3-(3′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 186 3-(2′-CH₃O—C₆H₄)-4-Chloroisoxazolyl-5 187 3-(4′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 188 3-(3′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 189 3-(2′-NO₂—C₆H₄)-4-Chloroisoxazolyl-5 190 3-(4′-CN—C₆H₄)-4-Chloroisoxazolyl-5 191 3-(3′-CN—C₆H₄)-4-Chloroisoxazolyl-5 192 3-(2′-CN—C₆H₄)-4-Chloroisoxazolyl-5 193 3-(4′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 194 3-(3′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 195 3-(2′-Cl—C₆H₄)-4-Chloroisoxazolyl-5 196 Isoxazolyl-3 197 5-CH₃-Isoxazolyl-3 198 5-C₆H₅-Isoxazolyl-3 199 5-(4′-CH₃—C₆H₄)-Isoxazolyl-3 200 5-(3′-CH₃—C₆H₄)-Isoxazolyl-3 201 5-(2′-CH₃—C₆H₄)-Isoxazolyl-3 202 5-(4′-CH₃O—C₆H₄)-Isoxazolyl-3 203 5-(3′-CH₃O—C₆H₄)-Isoxazolyl-3 204 5-(2′-CH₃O—C₆H₄)-Isoxazolyl-3 205 5-(4′-NO₂—C₆H₄)-Isoxazolyl-3 206 5-(3′-NO₂—C₆H₄)-Isoxazolyl-3 207 5-(2′-NO₂—C₆H₄)-Isoxazolyl-3 208 5-(4′-CN—C₆H₄)-Isoxazolyl-3 209 5-(3′-CN—C₆H₄)-Isoxazolyl-3 210 5-(2′-CN—C₆H₄)-Isoxazolyl-3 211 5-(4′-Cl—C₆H₄)-Isoxazolyl-3 212 5-(3′-Cl—C₆H₄)-Isoxazolyl-3 213 5-(2′-Cl—C₆H₄)-Isoxazolyl-3 214 Isothiazolyl-5 215 3-CH₃-Isothiazolyl-5 216 3-C₆H₅-Isothiazolyl-5 217 3-(4′-CH₃—C₆H₄)-Isothiazolyl-5 218 3-(3′-CH₃—C₆H₄)-Isothiazolyl-5 219 3-(2′-CH₃—C₆H₄)-Isothiazolyl-5 220 3-(4′-CH₃O—C₆H₄)-Isothiazolyl-5 221 3-(3′-CH₃O—C₆H₄)-Isothiazolyl-5 222 3-(2′-CH₃O—C₆H₄)-Isothiazolyl-5 223 3-(4′-NO₂—C₆H₄)-Isothiazolyl-5 224 3-(3′-NO₂—C₆H₄)-Isothiazolyl-5 225 3-(2′-NO₂—C₆H₄)-Isothiazolyl-5 226 3-(4′-CN—C₆H₄)-Isothiazolyl-5 227 3-(3′-CN—C₆H₄)-Isothiazolyl-5 228 3-(2′-CN—C₆H₄)-Isothiazolyl-5 229 3-(4′-Cl—C₆H₄)-Isothiazolyl-5 230 3-(3′-Cl—C₆H₄)-Isothiazolyl-5 231 3-(2′-Cl—C₆H₄)-Isothiazolyl-5 232 Oxazolyl-4 233 3-CH₃-Oxazolyl-4 234 3-C₆H₅-Oxazolyl-4 235 3-(4′-CH₃—C₆H₄)-Oxazolyl-4 236 3-(3′-CH₃—C₆H₄)-Oxazolyl-4 237 3-(2′-CH₃—C₆H₄)-Oxazolyl-4 238 3-(4′-CH₃O—C₆H₄)-Oxazolyl-4 239 3-(3′-CH₃O—C₆H₄)-Oxazolyl-4 240 3-(2′-CH₃O—C₆H₄)-Oxazolyl-4 241 3-(4′-NO₂—C₆H₄)-Oxazolyl-4 242 3-(3′-NO₂—C₆H₄)-Oxazolyl-4 243 3-(2′-NO₂—C₆H₄)-Oxazolyl-4 244 3-(4′-CN—C₆H₄)-Oxazolyl-4 245 3-(3′-CN—C₆H₄)-Oxazolyl-4 246 3-(2′-CN—C₆H₄)-Oxazolyl-4 247 3-(4′-Cl—C₆H₄)-Oxazolyl-4 248 3-(3′-Cl—C₆H₄)-Oxazolyl-4 249 3-(2′-Cl—C₆H₄)-Oxazolyl-4 250 Thiazolyl-4 251 2-CH₃-Thiazolyl-4 252 2-C₆H₅-Thiazolyl-4 253 2-(4′-CH₃—C₆H₄)-Thiazolyl-4 254 2-(3′-CH₃—C₆H₄)-Thiazolyl-4 255 2-(2′-CH₃—C₆H₄)-Thiazolyl-4 256 2-(4′-CH₃O—C₆H₄)-Thiazolyl-4 267 2-(3′-CH₃O—C₆H₄)-Thiazolyl-4 258 2-(2′-CH₃O—C₆H₄)-Thiazolyl-4 259 2-(4′-NO₂—C₆H₄)-Thiazolyl-4 260 2-(3′-NO₂—C₆H₄)-Thiazolyl-4 261 2-(2′-NO₂—C₆H₄)-Thiazolyl-4 262 2-(4′-CN—C₆H₄)-Thiazolyl-4 263 2-(3′-CN—C₆H₄)-Thiazolyl-4 264 2-(2′-CN—C₆H₄)-Thiazolyl-4 265 2-(4′-Cl—C₆H₄)-Thiazolyl-4 266 2-(3′-Cl—C₆H₄)-Thiazolyl-4 267 2-(2′-Cl—C₆H₄)-Thiazolyl-4 268 N—CH₃-1,2,4-Triazolyl-5 269 3-CH₃—N—CH₃-1,2,4-Triazolyl-5 270 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5 271 3-(4′-CH₃—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 272 3-(3′-CH₃—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 273 3-(2′-CH₃—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 274 3-(4′-CH₃O—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 275 3-(3′-CH₃O—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 276 3-(2′-CH₃O—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 277 3-(4′-NO₂—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 278 3-(3′-NO₂—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 279 3-(2′-NO₂—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 280 3-(4′-CN—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 281 3-(3′-CN—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 282 3-(2′-CN—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 283 3-(4′-Cl—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 284 3-(3′-Cl—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 285 3-(2′-Cl—C₆H₄)-N—CH₃-1,2,4-Triazolyl-5 286 1,3,4-Oxadiazolyl-2 287 5-CH₃-1,3,4-Oxadiazolyl-2 288 5-C₆H₅-1,3,4-Oxadiazolyl-2 289 5-(4′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 290 5-(3′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 291 5-(2′-CH₃—C₆H₄)-1,3,4-Oxadiazolyl-2 292 5-(4′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 293 5-(3′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 294 5-(2′-CH₃O—C₆H₄)-1,3,4-Oxadiazolyl-2 295 5-(4′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 296 5-(3′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 297 5-(2′-NO₂—C₆H₄)-1,3,4-Oxadiazolyl-2 298 5-(4′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 299 5-(3′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 300 5-(2′-CN—C₆H₄)-1,3,4-Oxadiazolyl-2 301 5-(4′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 302 5-(3′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 303 5-(2′-Cl—C₆H₄)-1,3,4-Oxadiazolyl-2 304 1,2,4-Oxadiazolyl-3 305 5-CH₃-1,2,4-Oxadiazolyl-3 306 5-C₆H₅-1,2,4-Oxadiazolyl-3 307 5-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 308 5-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 309 5-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-3 310 5-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 311 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 312 5-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-3 313 5-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 314 5-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 315 5-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-3 316 5-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 317 5-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 318 5-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-3 319 5-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 320 5-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 321 5-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-3 322 1,2,4-Oxadiazolyl-5 323 3-CH₃-1,2,4-Oxadiazolyl-5 324 3-C₆H₅-1,2,4-Oxadiazolyl-5 325 3-(4′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 326 3-(3′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 327 3-(2′-CH₃—C₆H₄)-1,2,4-Oxadiazolyl-5 328 3-(4′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 329 3-(3′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 330 3-(2′-CH₃O—C₆H₄)-1,2,4-Oxadiazolyl-5 331 3-(4′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 332 3-(3′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 333 3-(2′-NO₂—C₆H₄)-1,2,4-Oxadiazolyl-5 334 3-(4′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 335 3-(3′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 336 3-(2′-CN—C₆H₄)-1,2,4-Oxadiazolyl-5 337 3-(4′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 338 3-(3′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 339 3-(2′-Cl—C₆H₄)-1,2,4-Oxadiazolyl-5 340 1,2,4-Thiadiazolyl-3 341 5-CH₃-1,2,4-Thiadiazolyl-3 342 5-C₆H₅-1,2,4-Thiadiazolyl-3 343 5-(4′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 344 5-(3′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 345 5-(2′-CH₃—C₆H₄)-1,2,4-Thiadiazolyl-3 346 5-(4′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 347 5-(3′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 348 5-(2′-CH₃O—C₆H₄)-1,2,4-Thiadiazolyl-3 349 5-(4′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 350 5-(3′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 351 5-(2′-NO₂—C₆H₄)-1,2,4-Thiadiazolyl-3 352 5-(4′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 353 5-(3′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 354 5-(2′-CN—C₆H₄)-1,2,4-Thiadiazolyl-3 355 5-(4′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 356 5-(3′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 357 5-(2′-Cl—C₆H₄)-1,2,4-Thiadiazolyl-3 358 1,3,4-Thiadiazolyl-2 359 5-CH₃-1,3,4-Thiadiazolyl-2 360 5-C₆H₅-1,3,4-Thiadiazolyl-2 361 5-(4′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 362 5-(3′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 363 5-(2′-CH₃—C₆H₄)-1,3,4-Thiadiazolyl-2 364 5-(4′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 365 5-(3′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 366 5-(2′-CH₃O—C₆H₄)-1,3,4-Thiadiazolyl-2 367 5-(4′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 368 5-(3′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 369 5-(2′-NO₂—C₆H₄)-1,3,4-Thiadiazolyl-2 370 5-(4′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 371 5-(3′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 372 5-(2′-CN—C₆H₄)-1,3,4-Thiadiazolyl-2 373 5-(4′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 374 5-(3′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 375 5-(2′-Cl—C₆H₄)-1,3,4-Thiadiazolyl-2 376 Pyridinyl-2 377 Pyridinyl-4 378 Pyridazinyl-3 379 Pyridazinyl-4 380 Pyridazinyl-2 381 Pyrimidinyl-4 382 Pyrimidinyl-5 383 Pyrimidinyl-2 I: R¹ = H, X = CH₃ II: R¹ = CH₃, X = CH₃ III: R¹ = C₂H₅, X = CH₃ IV: R¹ = Allyl, X = CH₃ V: R¹ = Propargyl, X = CH₃ VI: R¹ = CH₂—OCH₃, X = CH₃ VII: R¹ = CO₂CH₃, X = CH₃ VIII: R¹ = H, X = Cl IX: : R¹ = CH₃, X = Cl X: R¹ = C₂H₅, X = Cl XI: R¹ = Allyl, X = Cl XII: R¹ = Propargyl, X = Cl XIII: R¹ = CH₂—OCH₃, X = Cl XIV: R¹ = CO₂CH₃, X = Cl

TABLE 47 Selected physical data of some compounds

IR (cm⁻¹) or No. X_(m) R¹ ¹H-NMR (ppm) mp 1 4-Cl H 133 2 3,4-Cl₂ H 109 3 4-t-C₄H₉ H 86 4 4-CH₃ H 117 5 4-CF₃ H 103 6 3-Br H 99 7 3-Cl H 93 8 3-CF₃ H 88 9 3,5-Cl₂ H 100 10 3,4-(CH₃)₂ H 127 11 3,4-Cl₂ CH₃ 74 12 3,4-Cl₂ Allyl 3.65(S, 3H); 2.2(S, 6H) 13 3,4-Cl₂ Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 14 3,4-Cl₂ CH₂—OCH₃ 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 15 3,4-Cl₂ CO—OCH₃ 137 16 4-t-C₄H₉ CH₃ 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 17 4-t-C₄H₉ Allyl 69 18 4-t-C₄H₉ Propargyl 117 19 4-t-C₄H₉ CH₂—OCH₃ 3.65(S, 3H); 2.25(S, 3H); 117 2.2(S, 3H) 20 4-t-C₄H₉ CO—OCH₃ 3.65; 2.1 119 21 4-CH₃ CH₃ 69 22 4-CH₃ Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 23 4-CH₃ Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 24 4-CH₃ CH₂—OCH₃ 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 25 4-CH₃ CO—OCH₃ 97 26 4-CF₃ CH₃ 76 27 4-CF₃ Allyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 28 4-CF₃ Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 29 4-CF₃ CH₂—OCH₃ 3.65(S, 3H); 2.25(S, 6H) 30 4-CF₃ CO—OCH₃ 103 31 4-Cl CH₃ 106 32 4-Cl Allyl 3.65(S, 3H); 2.2(2S, each 3H) 33 4-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H; 2.2(S, 3H) 34 4-Cl CH₂—OCH₃ 3.65(S, 3H); 2.25(S, 3H; 2.2(S, 3H) 35 4-Cl CO—OCH₃ 109 36 3-Br CH₃ 75 37 3-Br Allyl 3.65(S, 3H); 2.2(2S, each 3H 38 3-Br Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 39 3-Br CH₂—OCH₃ 72 40 3-Br CO—OCH₃ 131 41 3-Cl CH₃ 84 42 3-Cl Allyl 3.65(S, 3H); 2.25(S, 3H); 2.2(S, 3H) 43 3-Cl Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.2(S, 3H) 44 3-Cl CH₂—OCH₃ 66 45 3-Cl CO—OCH₃ 123 46 3-CF₃ CH₃ 63 47 3-CF₃ Allyl 64 48 3-CF₃ Propargyl 3.65(S, 3H); 2.3(S, 3H); 2.25(S, 3H) 49 3-CF₃ CH₂—OCH₃ 89 50 3-CF₃ CO—OCH₃ 136 51 4-Br CO—OCH₃ 103 52 4-Br H 108 53 4-Br Propargyl 1710,1486,1469,1447,1376, 1299,1252,1026,1008,774 54 4-Br CH₂—OCH₃ 1715,1468,1445,1370,1301, 1274,1090,1059,1008,775 55 3,4-(CH₃)₂ CH₃ oil 56 3,4-(CH₃)₂ Allyl oil 57 3,4-(CH₃)₂ Propargyl oil 58 3,4-(CH₃)₂ CH₂—OCH₃ oil 59 3,4-(CH₃)₂ CO—OCH₃ 135 60 3,5-Cl₂ CH₃ 95 61 3,5-Cl₂ Allyl 97 62 3,5-Cl₂ Propargyl 100 63 3,5-Cl₂ CH₂—OCH₃ 112 64 3,5-Cl₂ CO—OCH₃ 160

TABLE 48 Selected physical data of some compounds

IR (cm⁻¹) or ¹H-NMR No. X_(m) R¹ (ppm) mp 1 2-CH₃-4-C(CH₃)= H 82 N—OCH₃ 2 2,4-(CH₃)₂ H 131 3 2,5-(CH₃)₂ H 124 4 2-CH₃-4-C(CH₃)= H 102 N—OC₂H₅ 5 2,5-(CH₃)₂-4-C(CH₃)═ H 116 N—OC₂H₅ 6 2,5-(CH₃)₂-4-C(CH₃)═ H 122 N—OCH₃ 7 2-CH₃-4-C(CH₃)═ CH₃ 4.0(S, 3H); N—OCH₃ 3.65(S, 3H) 8 2-CH₃-4-C(CH₃)═ Allyl 101 N—OCH₃ 9 2-CH₃-4-C(CH₃)═ Propargyl 4.0(S, 3H); N—OCH₃ 3.65(S, 3H) 10 2-CH₃-4-C(CH₃)═ CH₂—OCH₃ 4.0(S, 3H); N—OCH₃ 3.65(S, 3H) 11 2-CH₃-4-C(CH₃)═ CO-OCH₃ 122 N—OCH₃ 12 2,4-(CH₃)₂ CH₃ 3.65(S, 3H); 2.25(2s, each 3H) 13 2,4-(CH₃)₂ Allyl 59 14 2,4-(CH₃)₂ Propargyl 3.65(S, 3H); 2.25(3s, each 3H) 15 2,4-(CH₃)₂ CH₂—OCH₃ 76 16 2,4-(CH₃)₂ CO—OCH₃ 133 17 2,5-(CH₃)₂ CH₃ 3.65(S, 3H); 2.3(s, 3H) 18 2,5-(CH₃)₂ Allyl 56 19 2,5-(CH₃)₂ Propargyl 80 20 2,5-(CH₃)₂ CH₂—OCH₃ 3.65(S, 3H); 80 2.3(S, 3H) 21 2,5-(CH₃)₂ CH₂—CCH₃ 140 22 2-CH₃ H 107 23 2-CH₃ Propargyl oil 24 2-CH₃ CO—OCH₃ 135 25 2-CH₃ CH₂—OCH₃ oil 26 2-CH₃-4-C(CH₃)═ H 97 B—O-Allyl 27 2-CH₃-4-C(CH₃)═ Propargyl oil N—O-Allyl 28 2-CH₃-4-C(CH₃)═ CO—OCH₃ 130 N—O-Allyl 29 2-CH₃-4-C(CH₃)═ CH₂—OCH₃ oil N—O-Allyl 30 2-CH₃-4-C(CH₃)═ CH₃ oil N—O—C₂H₅ 31 2-CH₃-4-C(CH₃)═ Allyl 75 N—O—C₂H₅ 32 2-CH₃-4-C(CH₃)═ Propargyl 77 N—O—C₂H₅ 33 2-CH₃-4-C(CH₃)═ CH₂—OCH₃ oil N—O—C₂H₅ 34 2-CH₃-4-C(CH₃)═ CO—OCH₃ oil N—O—C₂H₅ 35 2,5-(CH₃)²⁻4-C(CH₃)═ CH₃ oil N—OCH₃ 36 2,5-(CH₃)²⁻4-C(CH₃)═ Allyl 104 N—OCH₃ 37 2,5-(CH₃)²⁻4-C(CH₃)═ Propargyl oil N—OCH₃ 38 2,5-(CH₃)²⁻4-C(CH₃)═ CH₂—OCH₃ oil N—OCH₃ 39 2,5-(CH₃)²⁻4-C(CH₃)═ CO—OCH₃ 158 N—OCH₃ 40 2,5-(CH₃)₂-4-C(CH₃)═ CH₃ oil N—OC₂H₅ 41 2,5-(CH₃)²⁻4-C(CH₃)═ Allyl 71 N—OC₂H₅ 42 2,5-(CH₃)²⁻4-C(CH₃)═ Propargyl oil N—OC₂H₅ 43 2,5-(CH₃)²⁻4-C(CH₃)═ CH₂—OCH₃ oil N—OC₂H₅ 44 2,5-(CH₃)²⁻4-C(CH₃)═ CO—CCH₃ 128 N—OC₂H₅

TABLE 49

No. B 1 2-Pyridyl 2 3-Trifluoromethyl-2-pyridyl 3 5-Trifluoromethyl-2-pyridyl 4 3,5-Bis-(trifluoromethyl)-2-pyridyl 5 3,5-Dichloro-2-pyridyl 6 3-Chloro-5-trifluoromethyl-2-pyridyl 7 3,5-Dichloro-2-pyridyl 8 2-Chloro-4-trifluoromethylphenyl 9 2-Benzothiazolyl 10 5-Chloro-1-methyl-2-benzimidazolyl 11 2-Benzoxazolyl 12 1-Methyl-5-trifluoromethylimide-azo [5,4-a]- pyridin-2-yl 13 5-Chloro-2-pyrimidinyl 14 4-Methyl-5-phenyl-2-thiazolin-2-yl 15 4-Methyl-5-phenyl-2-oxazolin-2-yl 16 7-Trifluoromethyl-4-quinolinyl I: R¹ = H, X═CH₃ II: R¹ = CH₃, X═CH₃ II: R¹ = C₂H₅, X═CH₃ IV: R¹ = Allyl, X═CH₃ V: R¹ = Propargyl, X═CH₃ VI: R¹ = CH₂—OCH₃, X═CH₃ VII: R¹ = CO₂CH₃, X═CH₃ VIII: R¹ =H, X═Cl IX: R¹ = CH₃, X═Cl X: R¹ = C₂C₅, X═Cl XI: R¹ = Allyl, X═Cl XII: R¹ = Propargyl, X═Cl XIII: R¹ = CH₂—OCH₃, X═Cl XIV: R¹ = CO₂CH₃, X═Cl

TABLE 50 Selected physical data of some compounds

No. X_(m) IR (cm⁻¹) or ¹H-NMR (ppm) mp 1 4-NO₂ 112 2 3,4-Cl₂ 3.8 (s, 3H); 3.75 (s, 3H) 3 2,4-(CH₃)₂ 3.75 (s, 3H); 3.7 (s, 3H) 4 H 3.75 (2s, each 3H) 5 4-i-C₃H₇ 3.8 (s, 3H); 3.75 (s, 3H) 6 3,4-(CH₃)₂ 3.8 (s, 3H); 3.75 (s, 3H) 7 3-CH₃-4-OCH₃ 3.85 (s, 3H); 3.8 (s, 3H); 3.75 (s, 3H) 8 3-CH₃-4-O- 3.8 (2s, each 3H) i-C₃H₇ 9 4-CF₃ 3.8 (s, 3H); 3.75 (s, 3H) 10 3-CH₃ 3.8 (2s, each 3H) 11 3-CF₃ 3.8 (s, 3H); 3.75 (s, 3H) 12 4-F 3.8 (s, 3H); 3.75 (s, 3H) 13 4-Br 3.8 (s, 3H); 3.75 (s, 3H) 14 3-Br 3.8 (s, 3H); 3.75 (s, 3H) 15 4-t-Bu 3.8 (s, 3H); 3.75 (s, 3H) 16 4-OCH₃ 3.85 (s, 3H); 3.8 (s, 3H); 3.75 (s, 3H) 17 2-CH₃ 3.8 (s, 3H); 3.75 (s, 3H) 18 3-Cl 3.8 (s, 3H); 3.75 (s, 3H) 19 4-CN 3.8 (s, 3H); 3.75 (s, 3H) 20 4-C₂H₅ 3.8 (s, 3H); 3.75 (s, 3H)

TABLE 51 Selected physical data of some compounds

No. X_(m) IR (cm⁻¹) or ¹H-NMR (ppm) mp 1 4-Cl 3.8 (s, 3H); 3.75 (s, 3H) 2 2-Cl 3.8 (s, 3H); 3.75 (s, 3H) 3 2,5-(CH₃)₂-4-C(C₂H₅)═ 3.8 (s, 3H); 3.75 (s, 3H) N—O-Allyl 4 2,5-(CH₃)₂-4-C(C₂H₅)═ 3.9 (s, 3H); 3.8 (s, 3H); N—O—CH₃ 3.75 (s, 3H) 5 2-CH₃-4-C(C₂H₅)═ 3.8 (s, 3H); 3.75 (s, 3H) N—O-trans-Cl-Allyl 6 2-CH₃-4-C(C₂H₅)═ 3.8 (s, 3H); 3.75 (s, 3H) N—O-Allyl 7 2-CH₃-4-Cl 3.8 (s, 3H); 3.75 (s, 3H) 8 2-Cl-4-CH₃ 3.8 (s, 3H); 3.75 (s, 3H) 9 2-Cl-5-CH₃ 3.8 (s, 3H); 3.75 (s, 3H) 10 2-CH₃-4-C(C₂H₅)═ 4.2 (q, 2H); 3.8 (s, 3H); N—O—C₂H₅ 3.75 (s, 3H) 11 2-CH₃-4-C(C₂H₅)═ 3.95 (s, 3H); 3.8 (s, 3H); N—O—CH₃ 3.75 (s, 3H) 12 2,5-(CH₃)₂-4-C(CH₃)═ 3.8 (s, 3H); 3.75 (s, 3H) N—O-trans-Cl-Allyl 13 2,5-(CH₃)₂-4-C(CH₃)═ 4.2 (t, 2H); 3.8 (s, 3H); —N—O—C₂H₅ 3.75 (s, 3H) 14 2,5-(CH₃)₂-4-C(CH₃)═ 3.95 (s, 3H); 3.8 (s, 3H); N—O—CH₃ 3.75 (s, 3H) 15 2-CH₃-4-C(CH₃)═ 3.8 (s, 3H); 3.75 (s, 3H) N—O-trans-Cl-Allyl 16 2-CH₃-4-C(CH₃)═ 4.2 (t, 2H); 3.8 (s, 3H); N—O—C₂H₅ 3.75 (s, 3H) 17 2,5-(CH₃)₂-4-C(C₂H₅)═ 4.2 (t, 2H); 3.8 (s, 3H); N—O—C₂H₅ 3.75 (s, 3H)

TABLE 60

No. B 1 Phenyl 2 3-Phenoxyphenyl 3 3-(2-Cyanophenoxy)-phenyl 4 4-Chlorophenyl 5 3-Trifluoromethylphenyl 6 3-tert.-Butoxyphenyl 7 3,5-Dichlorophenyl 8 3,5-Diethylphenyl 9 2-Pyridyl 10 4-Pyrimidinyl 11 6-Phenoxy-pyrimidin-4-yl 12 6-Chloropyrimidin-4-yl 13 6-(2-Fluorophenoxy)-pyrimidin-4-yl 14 6-(2-Methylphenoxy)-pyrimidin-4-yl 15 6-(2-Cyanophenoxy)-pyrimidin-4-yl 16 6-(2,6-Difluorophenoxy)-pyrimidin-4-yl The novel compounds are suitable as fungicides.

The fungicidal compounds according to the invention, or agents containing them, may be applied for instance in the form of directly sprayable solutions, powders, suspensions (including high-percentage aqueous, oily or other suspensions), dispersions, emulsions, oil dispersions, pastes, dusts, broadcasting agents, or granules by spraying, atomizing, dusting, broadcasting or watering. The forms of application depend entirely on the purpose for which the agents are being used, but they must ensure as fine a distribution of the active ingredients according to the invention as possible.

Normally, the plants are sprayed or dusted with the active ingredients, or the seeds of the plants are treated with the active ingredients.

The formulations are produced in known manner, for example by extending the active ingredient with solvents and/or carriers, with or without the use of emulsifiers and dispersants; if water is used as solvent, it is also possible to employ other organic solvents as auxiliary solvents. Suitable auxiliaries for this purpose are solvents such as aromatics (e.g., xylene), chlorinated aromatics (e.g., chlorobenzenes), paraffins (e.g., crude oil fractions), alcohols (e.g., methanol, butanol), ketones (e.g., cyclohexanone), amines (e.g., ethanolamine, dimethylformamide), and water; carriers such as ground natural minerals (e.g., kaolins, aluminas, talc and chalk) and ground synthetic minerals (e.g., highly disperse silica and silicates); emulsifiers such as nonionic and anionic emulsifiers (e.g., polyoxyethylene fatty alcohol ethers, alkyl sulfonates and aryl sulfonates); and dispersants such as lignin-sulfite waste liquors and methylcellulose.

Examples of surfactants are: alkali metal, alkaline earth metal and ammonium salts of aromatic sulfonic acids, e.g. ligninsulfonic acid, phenolsulfonic acid, naphthalenesulfonic acid and dibutylnaphthalenesulfonic acid, and of fatty acids, alkyl and alkylaryl sulfonates, and alkyl, lauryl ether and fatty alcohol sulfates, and salts of sulfated hexadecanols, heptadecanols, and octadecanols, salts of fatty alcohol glycol ethers, condensation products of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensation products of naphthalene or naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ethers, ethoxylated isooctylphenol, ethoxylated octylphenol and ethoxylated nonylphenol, alkylphenol polyglycol ethers, tributylphenyl polyglycol ethers, alkylaryl polyether alcohols, isotridecyl alcohol fatty alcohol ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters, lignin-sulfite waste liquors and methyl cellulose.

Powders, dusts and broadcasting agents may be prepared by mixing or grinding the active ingredients with a solid carrier.

Granules, e.g., coated, impregnated or homogeneous granules may be prepared by bonding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silicic acids, silica gels, silicates, talc, kaolin, attapulgus clay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground plastics, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate, and ureas, and vegetable products such as grain meals, bark meal, wood meal, and nutshell meal, cellulosic powders, etc.

Examples of Formulations are Given Below:

I. A solution of 90 parts by weight of the compound from Table 7, No. 1 (7/1) and 10 parts by weight of N-methyl-α-pyrrolidone, which is suitable for application in the form of very fine drops.

II. A mixture of 20 parts by weight of compound 7/2, 80 parts by weight of xylene, 10 parts by weight of the adduct of 8 to 10 moles of ethylene oxide and 1 mole of oleic acid-N-monoethanolamide, 5 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, and 5 parts weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil. By finely dispersing the mixture in water, a dispersion is obtained.

III. An aqueous dispersion of 20 parts by weight of compound 7/3, 40 parts by weight of cyclohexanone, 30 parts weight of isobutanol, 20 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

IV. An aqueous dispersion of 20 parts by weight of compound 7/4, 25 parts by weight of cyclohexanol, 65 parts by weight of a mineral oil fraction having a boiling point between 210 and 280° C., and 10 parts by weight of the adduct of 40 moles of ethylene oxide and 1 mole of castor oil.

V. A hammer-milled mixture of 80 parts by weight of compound 7/5, 3 parts by weight of the sodium salt of diisobutylnaphthalene-α-sulfonic acid, 10 parts by weight of the sodium salt of a lignin-sulfonic acid obtained from a sulfite waste liquor, and 7 parts by weight of powdered silica gel. By finely dispersing the mixture in water, a spray liquor is obtained.

VI. An intimate mixture of 3 parts by weight of compound 7/6 and 97 parts by weight of particulate kaolin. The dust contains 3 wt % of the active ingredient.

VII. An intimate mixture of 30 parts by weight of compound 7/7, 92 parts by weight of powdered silica gel and 8 parts by weight of paraffin oil sprayed onto the surface of this silica gel. This formulation of the active ingredient exhibits good adherence.

VIII. A stable aqueous dispersion of 40 parts by weight of compound 7/8, 10 parts of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate, 2 parts of silica gel and 48 parts of water, which dispersion can be further diluted.

IX. A stable oily dispersion of 20 parts by weight of compound 7/9, 2 parts by weight of the calcium salt of dodecylbenzenesulfonic acid, 8 parts by weight of a fatty alcohol polyglycol ether, 2 parts by weight of the sodium salt of a phenolsulfonic acid-urea-formaldehyde condensate and 68 parts by weight of a paraffinic mineral oil.

The novel compounds are extremely effective on a broad spectrum of phytopathogenic fungi, in particular those from the class consisting of the Ascomycetes and Basidiomycetes. Some of them have a systemic action and can be used as foliar and soil fungicides.

The fungicidal compounds are of particular interest for controlling a large number of fungi in various crops or their seeds, especially wheat, rye, barley, oats, rice, Indian corn, lawns, cotton, soybeans, coffee, sugar cane, fruit and ornamentals in horticulture and viticulture, and in vegetables such as cucumbers, beans and cucurbits.

The compounds are applied by treating the fungi, or the seeds, plants, materials or soil to be protected against fungus attack with a fungicidally effective amount of the active ingredients.

The agents may be applied before or after infection of the materials, plants or seed by the fungi.

The compounds I are particularly useful for controlling the following plant diseases:

Erysiphe graminis in cereals,

Erysiphe cichoracearum and Sphaerotheca fuliginea in cucurbits,

Podosphaera leucotricha in apples,

Uncinula necator in vines,

Puccinia species in cereals,

Rhizoctonia solani in cotton,

Ustilago species in cereals and sugar cane,

Venturia inaequalis (scab) in apples,

Helminthosporium species in cereals,

Septoria nodorum in wheat,

Botrytis cinerea (gray mold) in strawberries and grapes,

Cercospora arachidicola in groundnuts,

Pseudocercosporella herpotrichoides in wheat and barley,

Pyricularia oryzae in rice,

Phytophthora infestans in potatoes and tomatoes,

Fusarium and Verticillium species in various plants,

Plasmopara viticola in grapes,

Alternaria species in fruit and vegetables.

The novel compounds may also be used for protecting materials (timber), for instance against Paecilomyces variotii

The fungicidal agents generally contain from 0.1 to 95, preferably from 0.5 to 90, wt % of active ingredient.

The application rates depend on the effect desired, and from 0.02 to 3 kg of active ingredient per hectare.

When the active ingredients are used for treating seed, amounts of from 0.001 to 50, and preferably from 0.01 to 10, g per kg of seed are generally needed.

When the agents according to the invention are used as fungicides, they may be present together with other active ingredients, e.g., herbicides, insecticides, growth regulators, other fungicides, and fertilizers.

When they are mixed with other fungicides, the spectrum of fungicidal action is in many cases increased.

Use Examples

The active ingredients used for comparison purposes were isopropyl N-phenylcarbamate (A)—known from GB 574 995—, isopropyl N-3-chlorophenylcarbamate (B)—known from GB 574 995—and methyl N-3,4-dichlorophenylcarbamate (C)—known from BE 612 550.

Example 1

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the “Frühgold” variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredients nos. 1, 2, 3, 4, 8, 9, 20, 23, 31, 33, 34, 35, 36, 42, 43, 44, 47, 48, 52, 53, 54, 55, 56, 57, 60, 61, 62, 63, 64, 67, 69, 70, 71, 72, 74, 78, 79, 85, 87, 89, 90, 91, 92, 93, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal 40 action (95%) than prior art comparative agents A (45%), B (45%) and C (45%).

Example 2

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the “Bahia” variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredients nos. 1, 2, 12, 18, 19, 22, 29, 39, 40, 42, 47, 49, 50, 52, 53, 54, 60, 61, 62, 63, 69, 70, 71, 72, 73, 74, 81, 83, 85, 87, 89, 90, 91, 92, 94, 95, 104, 105, 106 and 107 from Table 7 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (95%) than prior art con parative agents A (30%), B (30%) and C (30%).

Example 3

Action on Wheat Mildew

Leaves of pot-grown wheat seedlings of the “Frühgold” variety were sprayed with aqueous liquors containing (dry basis) 80% of active ingredient and 20% of emulsifier, and dusted, 24 hours after the sprayed-on layer had dried, with spores of wheat mildew (Erysiphe graminis var. tritici). The plants were then set up in the greenhouse at from 20 to 22° C. and a relative humidity of from 75 to 80%. The extent of mildew spread was assessed after 7 days.

The results show that active ingredient no. 3 from Table 14, nos. 3 and 4 from Table 21, nos. 1, 3, 4, 5, 6, 7, 8, 9, 10, 11, 15, 17, 18, 19, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40 41, 42, 43 and 44 from Table 48, nos. 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20 and 23 from Table 14, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18 and 19 from Table 52, and nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (15%).

Example 4

Action on Pyricularia oryzae (Protective)

Leaves of pot-grown rice seedlings of the “Bahia” variety were sprayed to runoff with aqueous emulsions containing (dry basis) 80% of active ingredient and 20% of emulsifier, and inoculated 24 hours later with an aqueous spore suspension of Pyricularia oryzae. The plants were then set up in climatic cabinets at 22 to 24° C. and 95 to 99% relative humidity. The extent of fungus attack was assessed after 6 days.

The results show that active ingredient nos. 3, 7, 8, 9, 10, 11, 13, 14, 15, 16, 17, 18, 20, 21, 22 and 24 from Table 14, nos. 1, 2, 3, 4, 5. 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16, 17, 18, 19 and 20 from Table 52, nos. 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13, 14, 15, 16 and 17 from Table 53, nos. 3 and 4 from Table 21, nos. 4 and 5 from Table 38, nos. 4, 7, 10, 16, 20, 21, 22, 23, 24, 25, 41, 42, 55, 56, 57, 58 and 59 from Table 47, and nos. 1, 4, 5, 6, 7, 8, 11, 20, 21, 22, 23, 24, 25, 26, 27, 28, 29, 30, 31, 32, 33, 34, 35, 36, 37, 38, 39, 40, 41, 42, 43 and 44 from Table 48 have, when applied as spray liquors containing 250 ppm of active ingredient, a better fungicidal action (100%) than prior art comparative agents A, B and C (0%).

Use Example 5

Action on Botrytis cinerea

Paprika seedlings of the “Neusiedler Ideal Elite” variety were sprayed, after 4 to 5 leaves were well developed, to runoff with aqueous suspensions containing (dry basis) 80 of active ingredient and 20% of emulsifier. After the sprayed-on layer had dried, the plants were sprinkled with a conidial suspension of the fungus Botrytis cinerea, and placed at 22 to 24° C. in a chamber of high humidity. After 5 days, the disease had spread to such a great extent on the untreated plants that the necroses covered the major portion of the leaves.

Percentage leaf attack after spraying with aqueous formulations containing 500 ppm Active ingredient of active ingredient Table 30, active ingr. no. 2 5 Comparative substance A 100 Comparative substance B 100 Comparative substance C 100 Untreated 100

Use Example 6

Action on Plasmopara viticola

Leaves of potted vines of the Muller-Thurgau variety were sprayed with aqueous suspensions containing (dry basis) 80% of active ingredient and 20% of emulsifier. To assess the duration of action, the plants were set up, after the sprayed-on layer had dried, for 8 days in the greenhouse. Then the leaves were infected with a zoospore suspension of Plasmopara viticola. The plants were first placed for 48 hours in a water vapor-saturated chamber at 24° C. and then a greenhouse for 5 days at from 20 to 300° C. To accelerate and intensify the sporangiophore discharge, the plants were then again placed in the moist chamber for 16 hours. The extent of fungus attack was then assessed on the undersides of the leaves.

Percentage leaf attack after applying aqueous formulations containing 500 ppm of Active ingredient active ingredient Table 21, active ingr. no. 3 5 Table 21, active ingr. no. 4 0 Table 30, active ingr. no. 1 15 Comparative substance A 65 Comparative substance B 40 Comparative substance C 25 Untreated 65 

What is claimed is:
 1. A carbamate of the formula VII

where the substituents have the following meanings: X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, R¹ is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or —CO₂-alkyl, A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or plant-tolerated acid and base adducts.
 2. The carbamate of claim 1, wherein X and Y are hydrogen, R¹ is alkyl, A is CHR²—O wherein R² is hydrogen.
 3. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is N—C₆H₅-Pyrazolyl-4.
 4. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is N-(4′-CH₃—C₆H₄)-Pyrazolyl-4.
 5. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is N-(4′-Cl—C₆H₄)-Pyrazolyl-4.
 6. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is 3-C₆H₅—N-Methylpyrazolyl-4.
 7. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is 3-(4′-Cl—C₆H₄)-N-Methylpyrazolyl-4.
 8. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is 3-C₆H₅—N—CH₃-1,2,4-Triazolyl-5.
 9. The carbamate of claim 2, wherein R¹ is methyl or ethyl, and B is 3-(4′-Cl—C₆H₄)—N—CH₃-1,2,4-Triazolyl-5.
 10. A carbamate of the formula VIII

where A, B, and R¹ have the meanings given in claim
 1. 11. A carbamate of the formula IX

where R¹ and B have the meanings given in claim
 1. 12. A carbamate of the formula X

where R¹ and B have the meanings given in claim
 1. 13. Hydroxylamine derivatives of the formula XIV

where the substituents have the following meanings: Z is NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂H₅, CF₃ or CCl₃, X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or together may be condensed form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic partially or completely hydrogenated ring, R¹ is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or —CO₂-alkyl, A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or its plant-tolerated acid and base adducts.
 14. A compound of the formula XV

where A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, Z is methoxy, NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂H₅, CF₃ or CCl₃, R¹ is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or —CO₂-alkyl and X and Y are identical or different and each is hydrogen, F, Cl, Br, C₁-C₄-alkyl, C₁-C₄-alkoxy or cyano.
 15. A compound of the formula XV as set forth in claim 14, where Y is hydrogen.
 16. A compound of the formula XV as set forth in claim 14, where X and Y are hydrogen.
 17. A compound of the formula XVI

where R¹, X, Y, Z and B have the meanings given in claim
 14. 18. A compound of the formula XVI as set forth in claim 17, Y denoting hydrogen.
 19. A compound of the formula XVI as set forth in claim 17, X and Y denoting hydrogen.
 20. A compound of the formula XVII

where R¹, X, Y, Z and B have the meanings given in claim
 14. 21. A compound of the formula XIX

where R¹, X, Y, Z and B have the meanings given in claim
 14. 22. A compound of the formula XIX

where R¹ is hydrogen, alkyl, alkenyl, alkynyl, cyclopropyl, cyclopropylmethyl, cyclobutyl, —CH₂—CN, —CH₂—O—CH₃, or —CO₂CH₃, X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl, or may be condensed together to form a phenyl ring, Z is methoxy, B is substituted or unsubstituted hetaryl.
 23. An intermediate of the formula XXII

where Z is NH₂, NHCH₃, N(CH₃)₂, CH₃, C₂H₅, CF₃, CCl₃, or methoxy, X and Y are identical or different and each is hydrogen, F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or together may be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, and R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy.
 24. An intermediate of the formula XXIII

where A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, X and Y are identical or different and each is hydrogen, F, Cl, Br, C₁-C₄-alkyl, C₁-C₄-alkoxy or cyano, W is phenoxy, p-nitrophenoxy, Cl₃C—O—, Cl₃C— or halide, and R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl, and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy.
 25. A compound of the formula XXV

where the substituents have the following meanings: X and Y are identical or different and each is F, Cl, Br, CF₃, CN, NO₂, alkoxy, alkenyloxy, alkynyloxy, alkyl, alkenyl or alkynyl or may together be condensed to form a substituted or unsubstituted aromatic or heteroaromatic, alicyclic or heterocyclic, partially or completely hydrogenated ring, or Y is hydrogen, R¹ is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or —CO₂-alkyl, A is —O—, —S—, —CR²═CR³—, CHR²—O—, —CHR²—S—, —CHR²—O—N═C(R⁴)—, —CR²═N—O—, —O—N═C(R⁴)—, —C≡C—, —CHR²—CHR³—, —CHR²—O—CO—, —O—CHR²— or a single bond, B is substituted or unsubstituted hetaryl, R² and R³ are identical or different and each is hydrogen, alkyl, alkenyl, alkynyl or cycloalkyl and R⁴ is hydrogen, cyano, alkyl, alkenyl, alkynyl, cycloalkyl or alkoxy, or its plant-tolerated acid and base adducts.
 26. A compound of the formula XXVI

where A, B and R¹ have the meanings given in claim 25 and X and Y are identical or different and each is F, Cl, Br, C₁-C₄-alkyl, C₁-C₄-alkoxy or cyano.
 27. A compound of the formula XXVI as set forth in claim 26, Y denoting hydrogen.
 28. A compound of the formula XXVII

where R¹, X, Y and B have the meanings given in claim
 25. 29. A compound of the formula XXVII as set forth in claim 28, Y denoting hydrogen.
 30. A compound of the formula XXVIII

where R¹, X, Y and B have the meanings given in claim
 25. 31. A compound of the formula XXIX

where R¹, X, Y and B have the meanings given in claim
 25. 32. A compound of the formula XXX

where R¹, X, Y and B have the meanings given in claim
 25. 